EA200400762A1 - Новые соединения, их использование в медицине, способ их изготовления и содержащие их фармацевтические композиции - Google Patents

Новые соединения, их использование в медицине, способ их изготовления и содержащие их фармацевтические композиции

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Publication number
EA200400762A1
EA200400762A1 EA200400762A EA200400762A EA200400762A1 EA 200400762 A1 EA200400762 A1 EA 200400762A1 EA 200400762 A EA200400762 A EA 200400762A EA 200400762 A EA200400762 A EA 200400762A EA 200400762 A1 EA200400762 A1 EA 200400762A1
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Eurasian Patent Office
Prior art keywords
pharmaceutically acceptable
compounds
new
relates
medicine
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EA200400762A
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English (en)
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EA008947B1 (ru
Inventor
Дебназ Бхуния
Сайбал Кумар Дас
Гуррам Ранга Мадхаван
Джавед Икбал
Ранджан Чакрабарти
Риба Каннимел Викрамадитян
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Д-Р Редди'С Лабораторис Лтд.
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Publication of EA200400762A1 publication Critical patent/EA200400762A1/ru
Publication of EA008947B1 publication Critical patent/EA008947B1/ru

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    • A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/35—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom
    • A61K31/352—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom condensed with carbocyclic rings, e.g. methantheline 
    • A61K31/353—3,4-Dihydrobenzopyrans, e.g. chroman, catechin
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Abstract

Изобретение касается новых антидиабетических, гиполипидемических, гипохолестеринемических соединений и средств против ожирения с формулой (I), их производных, их аналогов, их таутомерных форм, их стереоизомеров, их полиморфов, их фармацевтически приемлемых солей, их фармацевтически приемлемых сольватов и содержащих их фармацевтически приемлемых композиций. Конкретнее, данное изобретение касается соединений с общей формулой (I), являющихся преимущественно агонистами PPARα, их производных, их аналогов, их таутомерных форм, их стереоизомеров, их полиморфов, их фармацевтически приемлемых солей, их фармацевтически приемлемых сольватов, и содержащих их фармацевтически приемлемых композиций. Изобретение также касается способов получения новых соединений формулы (I), новых промежуточных соединений, способов их получения, использования новых промежуточных соединений в синтезе указанных выше соединений и их использования в качестве антидиабетических, гиполипидемических, гипохолестеринемических соединений и средств против ожирения.Отчет о международном поиске был опубликован 2004.06.10.
EA200400762A 2001-12-03 2002-12-02 АГОНИСТЫ PPARα И ИХ ПРИМЕНЕНИЕ EA008947B1 (ru)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
IN971MA2001 2001-12-03
PCT/IB2002/005064 WO2003048116A2 (en) 2001-12-03 2002-12-02 Esters and amides as ppar-alpha agonists ____________

Publications (2)

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EA200400762A1 true EA200400762A1 (ru) 2004-12-30
EA008947B1 EA008947B1 (ru) 2007-10-26

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EA200400762A EA008947B1 (ru) 2001-12-03 2002-12-02 АГОНИСТЫ PPARα И ИХ ПРИМЕНЕНИЕ

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US (2) US7314889B2 (ru)
EP (1) EP1453795A2 (ru)
JP (1) JP2005511686A (ru)
KR (1) KR20040066866A (ru)
CN (1) CN1697828A (ru)
AU (1) AU2002351069A1 (ru)
BR (1) BR0214675A (ru)
CA (1) CA2469227A1 (ru)
CO (1) CO5580760A2 (ru)
EA (1) EA008947B1 (ru)
HR (1) HRP20040485A2 (ru)
HU (1) HUP0402550A3 (ru)
IL (1) IL162185A0 (ru)
MX (1) MXPA04005257A (ru)
NO (1) NO20042805L (ru)
NZ (1) NZ533311A (ru)
PL (1) PL370554A1 (ru)
RS (1) RS48104A (ru)
UA (1) UA82835C2 (ru)
WO (1) WO2003048116A2 (ru)
ZA (1) ZA200404261B (ru)

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CN110627690A (zh) * 2019-10-03 2019-12-31 南京施倍泰生物科技有限公司 一类新型对香豆酸磺酸酯衍生物及其制备方法和应用
CN110590615A (zh) * 2019-10-03 2019-12-20 南京施倍泰生物科技有限公司 一类新型阿魏酸磺酸酯衍生物及其制备方法和应用
CN113968781A (zh) * 2021-11-11 2022-01-25 上海吉奉生物科技有限公司 一种(s)-2-羟基-3-邻甲基丙酸的合成方法
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US7598293B2 (en) 2009-10-06
IL162185A0 (en) 2005-11-20
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US20070142470A1 (en) 2007-06-21
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US20030229083A1 (en) 2003-12-11
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