UA80601C2 - The pyrimidin derivatives for the prevention of hiv infection - Google Patents
The pyrimidin derivatives for the prevention of hiv infection Download PDFInfo
- Publication number
- UA80601C2 UA80601C2 UAA200508362A UA2005008362A UA80601C2 UA 80601 C2 UA80601 C2 UA 80601C2 UA A200508362 A UAA200508362 A UA A200508362A UA 2005008362 A UA2005008362 A UA 2005008362A UA 80601 C2 UA80601 C2 UA 80601C2
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- UA
- Ukraine
- Prior art keywords
- alkyl
- group
- substituted
- cyano group
- amino
- Prior art date
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Classifications
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
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- C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
- C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
- C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
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- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
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- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
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- C07D409/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
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- Chemical & Material Sciences (AREA)
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Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP0301291 | 2003-02-07 | ||
| PCT/EP2004/001011 WO2004069812A1 (fr) | 2003-02-07 | 2004-02-04 | Derives de pyrimidine utilises dans la prevention des infections par le vih |
Publications (1)
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| UA80601C2 true UA80601C2 (en) | 2007-10-10 |
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| EP (1) | EP1597237B1 (fr) |
| JP (2) | JP5602333B2 (fr) |
| KR (2) | KR20110132482A (fr) |
| CN (2) | CN1747937A (fr) |
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| BR (1) | BRPI0407329A (fr) |
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| CL (1) | CL2004000192A1 (fr) |
| EA (1) | EA011164B1 (fr) |
| ES (1) | ES2598404T3 (fr) |
| HR (1) | HRP20050688B1 (fr) |
| IL (1) | IL170114A (fr) |
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| NO (1) | NO334178B1 (fr) |
| NZ (1) | NZ541902A (fr) |
| PL (1) | PL227577B1 (fr) |
| UA (1) | UA80601C2 (fr) |
| WO (1) | WO2004069812A1 (fr) |
| ZA (1) | ZA200506253B (fr) |
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| CZ299380B6 (cs) * | 1998-03-27 | 2008-07-09 | Janssen Pharmaceutica N. V. | Pyrimidinová sloucenina, použití této slouceniny pro prípravu léciva, farmaceutický prostredek tutoslouceninu obsahující, zpusob prípravy tohoto prostredku a uvedené slouceniny a kombinace a produktuvedenou slouceninu obsahující |
| HU230394B1 (hu) | 1998-11-10 | 2016-04-28 | Janssen Pharmaceutica N.V. | HIV-vírus szaporodását gátló pirimidin-származékok |
| ES2391550T3 (es) | 1999-04-15 | 2012-11-27 | Bristol-Myers Squibb Company | Inhibidores cíclicos de la proteína tirosina quinasa |
| AU5328500A (en) * | 1999-06-11 | 2001-01-02 | Merck & Co., Inc. | N-cyclopentyl modulators of chemokine receptor activity |
| GB9914258D0 (en) | 1999-06-18 | 1999-08-18 | Celltech Therapeutics Ltd | Chemical compounds |
| BRPI0014271B1 (pt) * | 1999-09-24 | 2021-06-22 | Janssen Pharmaceutica N.V. | Partícula consistindo em uma dispersão de sólidos, uso da dita partícula, dispersão de sólidos, forma de dosagem farmacêutica, bem como processos de preparação de dita partícula, dispersão e forma de dosagem |
| CA2406562C (fr) | 2000-05-08 | 2009-09-15 | Janssen Pharmaceutica N.V. | Pyrimidines et triazines inhibant la replication du vih |
| US6596729B2 (en) * | 2000-07-20 | 2003-07-22 | Bristol-Myers Squibb Company | Tricyclic-2-pyridone compounds useful as HIV reverse transcriptase inhibitors |
| JP2004525914A (ja) * | 2001-03-02 | 2004-08-26 | スミスクライン ビーチャム コーポレーション | 逆転写酵素阻害剤としてのベンゾフェノン類 |
| JO3429B1 (ar) * | 2001-08-13 | 2019-10-20 | Janssen Pharmaceutica Nv | مشتقات برميدينات مثبطة فيروس الايدز |
| TW200306192A (en) * | 2002-01-18 | 2003-11-16 | Bristol Myers Squibb Co | Tricyclic 2-pyrimidone compounds useful as HIV reverse transcriptase inhibitors |
| AR039540A1 (es) * | 2002-05-13 | 2005-02-23 | Tibotec Pharm Ltd | Compuestos microbicidas con contenido de pirimidina o triazina |
| AU2002350719A1 (en) * | 2002-11-29 | 2004-06-23 | Janssen Pharmaceutica N.V. | Pharmaceutical compositions comprising a basic respectively acidic drug compound, a surfactant and a physiologically tolerable water-soluble acid respectively base |
| BRPI0407329A (pt) | 2003-02-07 | 2006-01-10 | Janssen Pharmaceutica Nv | Derivados de pirimidina para a prevenção de infecção de hiv |
-
2004
- 2004-02-04 BR BR0407329-0A patent/BRPI0407329A/pt not_active Application Discontinuation
- 2004-02-04 JP JP2006501729A patent/JP5602333B2/ja not_active Expired - Lifetime
- 2004-02-04 PL PL378144A patent/PL227577B1/pl unknown
- 2004-02-04 NZ NZ541902A patent/NZ541902A/en not_active IP Right Cessation
- 2004-02-04 AP AP2005003366A patent/AP2065A/en active
- 2004-02-04 WO PCT/EP2004/001011 patent/WO2004069812A1/fr active Application Filing
- 2004-02-04 CN CNA2004800034604A patent/CN1747937A/zh active Pending
- 2004-02-04 CN CN2011100443222A patent/CN102151270A/zh active Pending
- 2004-02-04 KR KR1020117026076A patent/KR20110132482A/ko not_active Application Discontinuation
- 2004-02-04 ES ES04707937.1T patent/ES2598404T3/es not_active Expired - Lifetime
- 2004-02-04 CL CL200400192A patent/CL2004000192A1/es unknown
- 2004-02-04 KR KR1020057013837A patent/KR101185048B1/ko active IP Right Grant
- 2004-02-04 US US10/544,735 patent/US20070021449A1/en not_active Abandoned
- 2004-02-04 AU AU2004210081A patent/AU2004210081B2/en not_active Expired
- 2004-02-04 EA EA200501265A patent/EA011164B1/ru unknown
- 2004-02-04 CA CA2513527A patent/CA2513527C/fr not_active Expired - Lifetime
- 2004-02-04 EP EP04707937.1A patent/EP1597237B1/fr not_active Expired - Lifetime
- 2004-02-04 MX MXPA05008364A patent/MXPA05008364A/es active IP Right Grant
- 2004-02-05 MY MYPI20040342A patent/MY176490A/en unknown
- 2004-04-02 UA UAA200508362A patent/UA80601C2/uk unknown
-
2005
- 2005-08-01 HR HRP20050688AA patent/HRP20050688B1/hr not_active IP Right Cessation
- 2005-08-04 IL IL170114A patent/IL170114A/en active IP Right Grant
- 2005-08-04 ZA ZA200506253A patent/ZA200506253B/xx unknown
- 2005-09-06 NO NO20054143A patent/NO334178B1/no not_active IP Right Cessation
-
2009
- 2009-09-25 US US12/567,051 patent/US8828982B2/en active Active
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2014
- 2014-05-21 JP JP2014105248A patent/JP5799133B2/ja not_active Expired - Lifetime
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