UA80601C2 - The pyrimidin derivatives for the prevention of hiv infection - Google Patents
The pyrimidin derivatives for the prevention of hiv infection Download PDFInfo
- Publication number
- UA80601C2 UA80601C2 UAA200508362A UA2005008362A UA80601C2 UA 80601 C2 UA80601 C2 UA 80601C2 UA A200508362 A UAA200508362 A UA A200508362A UA 2005008362 A UA2005008362 A UA 2005008362A UA 80601 C2 UA80601 C2 UA 80601C2
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- UA
- Ukraine
- Prior art keywords
- alkyl
- group
- substituted
- cyano group
- amino
- Prior art date
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Classifications
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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- C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
- C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
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- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
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- C07D409/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
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| EP0301291 | 2003-02-07 | ||
| PCT/EP2004/001011 WO2004069812A1 (fr) | 2003-02-07 | 2004-02-04 | Derives de pyrimidine utilises dans la prevention des infections par le vih |
Publications (1)
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| UA80601C2 true UA80601C2 (en) | 2007-10-10 |
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| EP (1) | EP1597237B1 (fr) |
| JP (2) | JP5602333B2 (fr) |
| KR (2) | KR101185048B1 (fr) |
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| BR (1) | BRPI0407329A (fr) |
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| ES (1) | ES2598404T3 (fr) |
| HR (1) | HRP20050688B1 (fr) |
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| NO (1) | NO334178B1 (fr) |
| NZ (1) | NZ541902A (fr) |
| PL (1) | PL227577B1 (fr) |
| UA (1) | UA80601C2 (fr) |
| WO (1) | WO2004069812A1 (fr) |
| ZA (1) | ZA200506253B (fr) |
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| RU2260592C9 (ru) | 1999-04-15 | 2017-04-07 | Бристол-Маерс Сквибб Ко. | Циклические ингибиторы протеинтирозинкиназ |
| AU5328500A (en) * | 1999-06-11 | 2001-01-02 | Merck & Co., Inc. | N-cyclopentyl modulators of chemokine receptor activity |
| GB9914258D0 (en) | 1999-06-18 | 1999-08-18 | Celltech Therapeutics Ltd | Chemical compounds |
| OA12029A (en) * | 1999-09-24 | 2006-04-28 | Janssen Pharmaceutica Nv | Antiviral compositions. |
| WO2001085700A2 (fr) | 2000-05-08 | 2001-11-15 | Janssen Pharmaceutica N.V. | Inhibiteurs de la replication du vih |
| US6596729B2 (en) * | 2000-07-20 | 2003-07-22 | Bristol-Myers Squibb Company | Tricyclic-2-pyridone compounds useful as HIV reverse transcriptase inhibitors |
| CN1494528A (zh) * | 2001-03-02 | 2004-05-05 | ʷ��˿�������ȳ�ķ����˾ | 作为逆转录酶抑制剂的二苯酮 |
| JO3429B1 (ar) * | 2001-08-13 | 2019-10-20 | Janssen Pharmaceutica Nv | مشتقات برميدينات مثبطة فيروس الايدز |
| TW200306192A (en) | 2002-01-18 | 2003-11-16 | Bristol Myers Squibb Co | Tricyclic 2-pyrimidone compounds useful as HIV reverse transcriptase inhibitors |
| AR039540A1 (es) | 2002-05-13 | 2005-02-23 | Tibotec Pharm Ltd | Compuestos microbicidas con contenido de pirimidina o triazina |
| AU2002350719A1 (en) | 2002-11-29 | 2004-06-23 | Janssen Pharmaceutica N.V. | Pharmaceutical compositions comprising a basic respectively acidic drug compound, a surfactant and a physiologically tolerable water-soluble acid respectively base |
| CL2004000192A1 (es) | 2003-02-07 | 2005-03-18 | Janssen Pharmaceutica Nv | Uso de compuestos derivados de 2-aminopirimidina para preparar un medicamento para la prevencion de una infeccion por vih relaciones sexuales o un contacto intimo en la pareja. |
-
2004
- 2004-02-04 CL CL200400192A patent/CL2004000192A1/es unknown
- 2004-02-04 EP EP04707937.1A patent/EP1597237B1/fr not_active Expired - Lifetime
- 2004-02-04 KR KR1020057013837A patent/KR101185048B1/ko active IP Right Grant
- 2004-02-04 WO PCT/EP2004/001011 patent/WO2004069812A1/fr active Application Filing
- 2004-02-04 MX MXPA05008364A patent/MXPA05008364A/es active IP Right Grant
- 2004-02-04 AU AU2004210081A patent/AU2004210081B2/en not_active Expired
- 2004-02-04 NZ NZ541902A patent/NZ541902A/en not_active IP Right Cessation
- 2004-02-04 JP JP2006501729A patent/JP5602333B2/ja not_active Expired - Lifetime
- 2004-02-04 CN CNA2004800034604A patent/CN1747937A/zh active Pending
- 2004-02-04 AP AP2005003366A patent/AP2065A/en active
- 2004-02-04 BR BR0407329-0A patent/BRPI0407329A/pt not_active Application Discontinuation
- 2004-02-04 ES ES04707937.1T patent/ES2598404T3/es not_active Expired - Lifetime
- 2004-02-04 US US10/544,735 patent/US20070021449A1/en not_active Abandoned
- 2004-02-04 EA EA200501265A patent/EA011164B1/ru unknown
- 2004-02-04 CN CN2011100443222A patent/CN102151270A/zh active Pending
- 2004-02-04 PL PL378144A patent/PL227577B1/pl unknown
- 2004-02-04 KR KR1020117026076A patent/KR20110132482A/ko not_active Application Discontinuation
- 2004-02-04 CA CA2513527A patent/CA2513527C/fr not_active Expired - Lifetime
- 2004-02-05 MY MYPI20040342A patent/MY176490A/en unknown
- 2004-04-02 UA UAA200508362A patent/UA80601C2/uk unknown
-
2005
- 2005-08-01 HR HRP20050688AA patent/HRP20050688B1/hr not_active IP Right Cessation
- 2005-08-04 IL IL170114A patent/IL170114A/en active IP Right Grant
- 2005-08-04 ZA ZA200506253A patent/ZA200506253B/xx unknown
- 2005-09-06 NO NO20054143A patent/NO334178B1/no not_active IP Right Cessation
-
2009
- 2009-09-25 US US12/567,051 patent/US8828982B2/en active Active
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2014
- 2014-05-21 JP JP2014105248A patent/JP5799133B2/ja not_active Expired - Lifetime
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