TWI359141B - Preparation of fluoromethyl-substituted heterocycl - Google Patents

Preparation of fluoromethyl-substituted heterocycl Download PDF

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Publication number
TWI359141B
TWI359141B TW093132853A TW93132853A TWI359141B TW I359141 B TWI359141 B TW I359141B TW 093132853 A TW093132853 A TW 093132853A TW 93132853 A TW93132853 A TW 93132853A TW I359141 B TWI359141 B TW I359141B
Authority
TW
Taiwan
Prior art keywords
group
formula
alkyl
heterocyclic ring
substituted heterocyclic
Prior art date
Application number
TW093132853A
Other languages
English (en)
Chinese (zh)
Other versions
TW200530189A (en
Inventor
Reinhard Lantzsch
Sergiy Pazenok
Frank Memmel
Original Assignee
Bayer Cropscience Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Cropscience Ag filed Critical Bayer Cropscience Ag
Publication of TW200530189A publication Critical patent/TW200530189A/zh
Application granted granted Critical
Publication of TWI359141B publication Critical patent/TWI359141B/zh

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
    • C07D263/02—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings
    • C07D263/30—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D263/34—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D277/22—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • C07D277/30—Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
TW093132853A 2003-10-31 2004-10-29 Preparation of fluoromethyl-substituted heterocycl TWI359141B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE10351088A DE10351088A1 (de) 2003-10-31 2003-10-31 Verfahren zum Herstellen von fluormethyl-substituierten Heterocyclen

Publications (2)

Publication Number Publication Date
TW200530189A TW200530189A (en) 2005-09-16
TWI359141B true TWI359141B (en) 2012-03-01

Family

ID=34530016

Family Applications (1)

Application Number Title Priority Date Filing Date
TW093132853A TWI359141B (en) 2003-10-31 2004-10-29 Preparation of fluoromethyl-substituted heterocycl

Country Status (14)

Country Link
US (1) US7501527B2 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
EP (1) EP1682515B1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
JP (1) JP4936895B2 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
KR (1) KR101123745B1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
CN (1) CN1875006B (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
BR (1) BRPI0416112A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
DE (1) DE10351088A1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
DK (1) DK1682515T3 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
ES (1) ES2524597T3 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
IL (1) IL175148A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
IN (1) IN2006DE01990A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
MX (1) MXPA06004605A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
TW (1) TWI359141B (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
WO (1) WO2005044804A1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)

Families Citing this family (19)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DK2086944T3 (da) 2006-11-03 2010-05-03 Basf Se Fremgangsmåde til fremstilling af difluormethylpyrazolylcarboxylater
EP2121618A1 (de) * 2006-12-21 2009-11-25 Basf Se Verfahren zur herstellung fluormethylsubstituierter heterocyclischer verbindungen
MX2009012020A (es) 2007-06-01 2009-11-18 Basf Se Procedimiento para la preparacion de (3-dihalometil-1-metil-pirazo l-4-il) carboxamidas n-sustituidas.
BRPI0812958A2 (pt) * 2007-06-15 2014-12-09 Basf Se Processo para preparar compostos, uso de compostos, e, compostos
CN105732376A (zh) 2007-08-16 2016-07-06 索尔维公司 制备4-氟取代的3-氧代-烷酸酯的方法
WO2009106619A1 (en) 2008-02-29 2009-09-03 Basf Se Process for preparing alkyl 2-alkoxymethylene-4,4-difluoro-3-oxobutyrates
US8314233B2 (en) 2008-05-02 2012-11-20 Basf Se Process for preparing 2-(aminomethylidene)-4,4-difluoro-3-oxobutyric esters
BRPI0911897A2 (pt) * 2008-05-02 2015-07-28 Basf Se Processo para a preparação de compostos, e, composto
JP5587293B2 (ja) 2008-05-05 2014-09-10 ビーエーエスエフ ソシエタス・ヨーロピア １，３，４−置換ピラゾール化合物の調製方法
EA018518B1 (ru) * 2008-05-08 2013-08-30 Басф Се Способ получения арилкарбоксамидов
MX2011000209A (es) 2008-07-21 2011-03-01 Basf Se Procedimiento para la obtencion de esteres de acido pirazolcarboxilicos disustituidos en 1,3.
JP5889299B2 (ja) * 2010-07-23 2016-03-22 ソルヴェイ（ソシエテ アノニム） １−置換−３−フルオロアルキル−ピラゾール−４−カルボン酸のエステルの調製方法
FR2975990B1 (fr) * 2011-06-01 2013-05-24 Rhodia Operations Procede de preparation d'un compose organique fluore
FR2975992B1 (fr) * 2011-06-01 2013-11-08 Rhodia Operations Procede de preparation d'un compose fluoromethylpyrazole sous forme acide carboxylique ou derivee
US20140128617A1 (en) * 2011-06-21 2014-05-08 Wahed Ahmed Moradi Method for producing pyrazolylcarboxanilides
US20150376135A1 (en) * 2013-02-15 2015-12-31 Syngenta Participations Ag Process for the preparation of bis-dihaloalkyl pyrazoles
DK3046908T3 (en) * 2013-09-20 2017-10-02 Bayer Cropscience Ag METHOD FOR PREPARING 5-FLOUR-1-ALKYL-3-FLOURALKYL-1H-PYRAZOL-4-CARBALDEHYDE.
CN106045910B (zh) * 2016-08-15 2017-10-10 浙江永太科技股份有限公司 一种3‑(二氟甲基)‑1‑甲基‑1h‑吡唑‑4‑羧酸的合成方法
CN115572210B (zh) * 2022-12-08 2023-03-21 暨南大学 一种(1,2,2,2-四氟乙基)芳烃衍生物及其制备方法和应用

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS6357568A (ja) * 1982-04-16 1988-03-12 ザ　ダウ　ケミカル　カンパニ− 液相ハロゲン交換反応における触媒再使用
DE3400168A1 (de) * 1984-01-04 1985-07-11 Bayer Ag, 5090 Leverkusen 5-halogenalkyl-1,3,4-thiadiazol-2-yloxyacetamide
DE3934924C2 (de) * 1989-10-20 1994-01-27 Huels Chemische Werke Ag Verfahren zur Herstellung von 4-Alkoxycarbonyl-3-chlormethyl-2H-pyrazolen
US5126275A (en) * 1990-09-19 1992-06-30 Miles Inc. Analytical method using tetrazolium salt indicators having a reflectance plateau
US5093347A (en) 1991-01-28 1992-03-03 Monsanto Company 3-difluoromethylpyrazolecarboxamide fungicides, compositions and use
US5223526A (en) 1991-12-06 1993-06-29 Monsanto Company Pyrazole carboxanilide fungicides and use
DE4231517A1 (de) 1992-09-21 1994-03-24 Basf Ag Carbonsäureanilide, Verfahren zu ihrer Herstellung und sie enthaltende Mittel zur Bekämpfung von Schadpilzen
DE19544800A1 (de) * 1995-12-01 1997-06-05 Bayer Ag Verfahren zur Herstellung von 1,3-Dimethyl-5-fluor-pyrazol-4-carboxaniliden
DE19629828A1 (de) 1996-07-24 1998-01-29 Bayer Ag Carbanilide
JP3533134B2 (ja) * 1999-02-15 2004-05-31 三井化学株式会社 フッ素化剤及びその製法と使用
DE10215292A1 (de) * 2002-02-19 2003-08-28 Bayer Cropscience Ag Disubstitutierte Pyrazolylcarbocanilide

Also Published As

Publication number Publication date
CN1875006B (zh) 2011-12-21
IL175148A (en) 2015-03-31
TW200530189A (en) 2005-09-16
JP2007509871A (ja) 2007-04-19
JP4936895B2 (ja) 2012-05-23
IN2006DE01990A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) 2007-07-13
WO2005044804A1 (de) 2005-05-19
DK1682515T3 (en) 2014-11-17
CN1875006A (zh) 2006-12-06
KR101123745B1 (ko) 2012-03-15
IL175148A0 (en) 2006-09-05
MXPA06004605A (es) 2006-07-20
DE10351088A1 (de) 2005-06-02
US7501527B2 (en) 2009-03-10
EP1682515B1 (de) 2014-10-01
EP1682515A1 (de) 2006-07-26
US20060276656A1 (en) 2006-12-07
BRPI0416112A (pt) 2007-01-02
KR20060094534A (ko) 2006-08-29
ES2524597T3 (es) 2014-12-10

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