TWI357899B - Process for producing 5-hydroxy-4-thiomethylpyrazo - Google Patents
Process for producing 5-hydroxy-4-thiomethylpyrazo Download PDFInfo
- Publication number
- TWI357899B TWI357899B TW094110223A TW94110223A TWI357899B TW I357899 B TWI357899 B TW I357899B TW 094110223 A TW094110223 A TW 094110223A TW 94110223 A TW94110223 A TW 94110223A TW I357899 B TWI357899 B TW I357899B
- Authority
- TW
- Taiwan
- Prior art keywords
- group
- hydroxy
- reaction
- mmol
- compound
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D231/18—One oxygen or sulfur atom
- C07D231/20—One oxygen atom attached in position 3 or 5
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D231/28—Two oxygen or sulfur atoms
- C07D231/30—Two oxygen or sulfur atoms attached in positions 3 and 5
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Plural Heterocyclic Compounds (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2004102963A JP4621939B2 (ja) | 2004-03-31 | 2004-03-31 | ５−ヒドロキシ−４−チオメチルピラゾール化合物の製造方法 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| TW200536832A TW200536832A (en) | 2005-11-16 |
| TWI357899B true TWI357899B (en) | 2012-02-11 |
Family
ID=35063690
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| TW094110223A TWI357899B (en) | 2004-03-31 | 2005-03-31 | Process for producing 5-hydroxy-4-thiomethylpyrazo |
Country Status (19)
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| TWI848950B (zh) * | 2018-05-31 | 2024-07-21 | 日商組合化學工業股份有限公司 | 含氟之吡唑衍生物之製造方法及其中間物 |
Families Citing this family (24)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AU2005291117B2 (en) | 2004-10-05 | 2011-06-09 | Syngenta Limited | Isoxazoline derivatives and their use as herbicides |
| AR052058A1 (es) * | 2004-12-20 | 2007-02-28 | Ihara Chemical Ind Co | Metodo para producir un compuesto de sal (4.5-dihidroisoxasol-3-yl) tiocarboxamidina |
| JP2007031342A (ja) * | 2005-07-27 | 2007-02-08 | Ihara Chem Ind Co Ltd | ５−ヒドロキシ−１−アルキルピラゾール誘導体の製造方法 |
| NZ570495A (en) | 2006-02-14 | 2011-10-28 | Ihara Chemical Ind Co | Process for production of 5-alkoxy-4-hydroxymethylpyrazole compound |
| KR20100017372A (ko) * | 2007-05-25 | 2010-02-16 | 애보트 게엠베하 운트 콤파니 카게 | 향대사성 글루타메이트 수용체 2（ｍｇｌｕ2 수용체）의 포지티브 조절자로서의 헤테로사이클릭 화합물 |
| GB0916267D0 (en) | 2009-09-16 | 2009-10-28 | Syngenta Ltd | Herbicidal compounds |
| CA2781404A1 (en) * | 2009-11-26 | 2011-06-03 | Basf Se | Method for producing 5,5-disubstituted 4,5-dihydroisoxazol-3-thiocarboxamidine salts |
| DK2504321T3 (da) | 2009-11-26 | 2014-07-14 | Basf Se | Fremgangsmåde til fremstilling af 5,5-disubstituerede 2-isoxazoliner |
| EP2571854B1 (en) * | 2010-05-20 | 2014-11-05 | Bayer Intellectual Property GmbH | Method for manufacturing 1-alkyl-3-difluormethyl-5-hydroxypyrazoles |
| WO2013016815A1 (en) | 2011-07-29 | 2013-02-07 | Rashidian Atabak | Polymer-based resonator antennas |
| CN103387541B (zh) * | 2012-05-10 | 2016-02-10 | 中国中化股份有限公司 | 一种取代吡唑醚类化合物的制备方法 |
| CN108026051A (zh) * | 2015-11-16 | 2018-05-11 | 隆萨有限公司 | 制备1-甲基-3-（三氟甲基）-1h-吡唑-5-醇的方法 |
| TW201835036A (zh) | 2017-02-27 | 2018-10-01 | 瑞士商隆薩有限公司 | 製備1-甲基-3-(三氟甲基)-1h-吡唑-5-醇的方法 |
| WO2019131715A1 (ja) * | 2017-12-27 | 2019-07-04 | クミアイ化学工業株式会社 | チオカルボキサミジン塩化合物の製造方法 |
| WO2021019537A1 (en) | 2019-07-30 | 2021-02-04 | Adama Agan Ltd. | Process and intermediates for the preparation of pyroxasulfone |
| US20230012374A1 (en) | 2019-10-31 | 2023-01-12 | Kumiai Chemical Industry Co., Ltd. | Process for producing herbicide and intermediate thereof |
| BR112022017794A2 (pt) | 2020-03-05 | 2022-10-25 | Adama Agan Ltd | Processo e intermediários para a preparação de piroxassulfona |
| CN111574511A (zh) * | 2020-06-28 | 2020-08-25 | 安徽久易农业股份有限公司 | 一种砜吡草唑的合成方法及其应用 |
| EP4177244A3 (en) | 2020-07-10 | 2023-08-09 | Adama Agan Ltd. | Process and intermediates for the preparation of pyroxasulfone and fenoxasulfone |
| CN112110912B (zh) * | 2020-07-31 | 2022-07-05 | 绍兴贝斯美化工股份有限公司 | 一种合成硫醚类中间体的方法 |
| TW202334128A (zh) | 2021-10-29 | 2023-09-01 | 日商組合化學工業股份有限公司 | 二硫化物化合物、多硫化物化合物及其用途 |
| AR127776A1 (es) | 2021-11-28 | 2024-02-28 | Adama Agan Ltd | Composiciones de concentrado en suspensión de alta carga |
| CN114716428B (zh) * | 2022-05-06 | 2024-02-06 | 山东潍坊润丰化工股份有限公司 | 制备砜吡草唑中间体的方法 |
| CN115850178B (zh) * | 2022-12-28 | 2025-04-04 | 宁夏格瑞精细化工有限公司 | 一种1-甲基-3-(三氟甲基)-1h-吡唑-5-醇的制备方法 |
Family Cites Families (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4918085A (en) * | 1989-03-02 | 1990-04-17 | Rhone-Poulenc Ag Company | Pesticidal 3-cyano-5-alkoxy-1-arylpyrazoles, compositions and use |
| AR035912A1 (es) * | 2000-03-02 | 2004-07-28 | Aventis Cropscience Sa | Compuestos de 4-tiometilpirazol, composicion plaguicida, metodo para el control de plagas en un lugar, semillas tratadas o recubiertas,uso de estos compuestos o composiciones para el control de plagas, uso de estos compuestos para preparar un medicamento veterinario, y,proceso para la preparacion de |
| JP4465133B2 (ja) * | 2001-02-08 | 2010-05-19 | クミアイ化学工業株式会社 | イソオキサゾリン誘導体及びこれを有効成分とする除草剤 |
| JP4317445B2 (ja) * | 2001-06-21 | 2009-08-19 | クミアイ化学工業株式会社 | イソオキサゾリン誘導体及び除草剤 |
| EP1541561B1 (en) * | 2002-08-01 | 2014-07-23 | Ihara Chemical Industry Co., Ltd. | Pyrazole derivatives and process for the production thereof |
| UA78071C2 (en) * | 2002-08-07 | 2007-02-15 | Kumiai Chemical Industry Co | Herbicidal composition |
-
2004
- 2004-03-31 JP JP2004102963A patent/JP4621939B2/ja not_active Expired - Lifetime
-
2005
- 2005-03-31 NZ NZ550143A patent/NZ550143A/en not_active IP Right Cessation
- 2005-03-31 WO PCT/JP2005/006806 patent/WO2005095352A1/ja active Application Filing
- 2005-03-31 RU RU2006138241/04A patent/RU2386619C2/ru active
- 2005-03-31 EP EP05728918.3A patent/EP1767528B1/en not_active Expired - Lifetime
- 2005-03-31 ES ES05728918.3T patent/ES2508765T3/es not_active Expired - Lifetime
- 2005-03-31 AU AU2005228017A patent/AU2005228017B2/en not_active Expired
- 2005-03-31 CA CA2560936A patent/CA2560936C/en not_active Expired - Lifetime
- 2005-03-31 US US10/594,710 patent/US7488831B2/en active Active
- 2005-03-31 TW TW094110223A patent/TWI357899B/zh not_active IP Right Cessation
- 2005-03-31 UA UAA200611331A patent/UA83910C2/ru unknown
- 2005-03-31 MX MXPA06011130 patent/MX280092B/es active IP Right Grant
- 2005-03-31 BR BRPI0509353A patent/BRPI0509353B1/pt active IP Right Grant
- 2005-03-31 CN CN2005800106359A patent/CN1938278B/zh not_active Expired - Lifetime
- 2005-03-31 PL PL05728918T patent/PL1767528T3/pl unknown
- 2005-03-31 KR KR1020067019480A patent/KR101205731B1/ko not_active Expired - Lifetime
-
2006
- 2006-09-20 CR CR8640A patent/CR8640A/es unknown
- 2006-09-21 IL IL178233A patent/IL178233A/en active IP Right Grant
- 2006-09-25 IN IN5581DE2006 patent/IN2006DE05581A/en unknown
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| TWI848950B (zh) * | 2018-05-31 | 2024-07-21 | 日商組合化學工業股份有限公司 | 含氟之吡唑衍生物之製造方法及其中間物 |
Also Published As
| Publication number | Publication date |
|---|---|
| PL1767528T3 (pl) | 2015-03-31 |
| KR101205731B1 (ko) | 2012-11-28 |
| AU2005228017B2 (en) | 2010-09-30 |
| CA2560936C (en) | 2013-01-08 |
| EP1767528B1 (en) | 2014-09-17 |
| NZ550143A (en) | 2010-04-30 |
| US20070185334A1 (en) | 2007-08-09 |
| JP4621939B2 (ja) | 2011-02-02 |
| US7488831B2 (en) | 2009-02-10 |
| BRPI0509353A (pt) | 2007-09-11 |
| IL178233A (en) | 2014-02-27 |
| WO2005095352A1 (ja) | 2005-10-13 |
| BRPI0509353A8 (pt) | 2017-09-19 |
| CR8640A (es) | 2007-08-28 |
| ES2508765T3 (es) | 2014-10-16 |
| CA2560936A1 (en) | 2005-10-13 |
| EP1767528A4 (en) | 2010-04-21 |
| CN1938278B (zh) | 2012-12-12 |
| RU2386619C2 (ru) | 2010-04-20 |
| AU2005228017A1 (en) | 2005-10-13 |
| JP2005289824A (ja) | 2005-10-20 |
| IN2006DE05581A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) | 2007-08-31 |
| MX280092B (es) | 2010-10-18 |
| MXPA06011130A (es) | 2007-01-25 |
| CN1938278A (zh) | 2007-03-28 |
| BRPI0509353B1 (pt) | 2019-01-02 |
| IL178233A0 (en) | 2006-12-31 |
| RU2006138241A (ru) | 2008-05-10 |
| UA83910C2 (ru) | 2008-08-26 |
| TW200536832A (en) | 2005-11-16 |
| KR20070003964A (ko) | 2007-01-05 |
| EP1767528A1 (en) | 2007-03-28 |
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| MK4A | Expiration of patent term of an invention patent |