TWI295670B - Vanilloid receptor ligands and their use in treatments - Google Patents
Vanilloid receptor ligands and their use in treatments Download PDFInfo
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- TWI295670B TWI295670B TW094104222A TW94104222A TWI295670B TW I295670 B TWI295670 B TW I295670B TW 094104222 A TW094104222 A TW 094104222A TW 94104222 A TW94104222 A TW 94104222A TW I295670 B TWI295670 B TW I295670B
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- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
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- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
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- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
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| KR101042490B1 (ko) | 2004-07-15 | 2011-06-16 | 니뽄 다바코 산교 가부시키가이샤 | 축합 벤즈아미드 화합물 및 바닐로이드 수용체 1형(vr1)활성 저해제 |
| WO2006089311A1 (en) * | 2005-02-15 | 2006-08-24 | Amgen Inc. | Vanilloid receptor ligands and their use in treatments |
| CA2632508A1 (en) * | 2005-12-28 | 2008-06-05 | Japan Tobacco Inc. | 3,4-dihydrobenzoxazine compound and inhibitor of vanilloid receptor type 1 (vr1) activity |
| US7906508B2 (en) * | 2005-12-28 | 2011-03-15 | Japan Tobacco Inc. | 3,4-dihydrobenzoxazine compounds and inhibitors of vanilloid receptor subtype 1 (VRI) activity |
| MX2010004246A (es) * | 2007-10-18 | 2010-04-30 | Novartis Ag | Inhibidores de csf-1r para el tratamiento de cancer y de enfermedades oseas. |
| US7938903B2 (en) * | 2008-03-07 | 2011-05-10 | Xerox Corporation | Nanosized particles of benzimidazolone pigments |
| US8012254B2 (en) | 2008-03-07 | 2011-09-06 | Xerox Corporation | Nanosized particles of benzimidazolone pigments |
| US8025723B2 (en) | 2008-03-07 | 2011-09-27 | Xerox Corporation | Nonpolar liquid and solid phase change ink compositions comprising nanosized particles of benzimidazolone pigments |
| US7985290B2 (en) | 2008-03-07 | 2011-07-26 | Xerox Corporation | Nonpolar liquid and solid phase change ink compositions comprising nanosized particles of benzimidazolone pigments |
| US7883574B2 (en) * | 2008-03-07 | 2011-02-08 | Xerox Corporation | Methods of making nanosized particles of benzimidazolone pigments |
| US7857901B2 (en) * | 2008-03-07 | 2010-12-28 | Xerox Corporation | Nonpolar liquid and solid phase change ink compositions comprising nanosized particles of benzimidazolone pigments |
| US7905954B2 (en) * | 2008-03-07 | 2011-03-15 | Xerox Corporation | Nanosized particles of benzimidazolone pigments |
| PL2285786T3 (pl) * | 2008-06-16 | 2014-01-31 | Merck Patent Gmbh | Pochodne chinoksalinodionowe |
| KR101676375B1 (ko) | 2009-04-09 | 2016-11-15 | 시므라이즈 아게 | 피부 자극-완화제로서 트랜스-텔트-부틸 사이클로헥사놀을 포함하는 조성물 |
| EP2322512B1 (en) | 2009-10-19 | 2015-10-21 | Xerox Corporation | Alkylated benzimidazolone compounds and self-assembled nanostructures generated therefrom |
| US8703988B2 (en) | 2010-06-22 | 2014-04-22 | Xerox Corporation | Self-assembled nanostructures |
| US8362270B2 (en) | 2010-05-11 | 2013-01-29 | Xerox Corporation | Self-assembled nanostructures |
| HRP20200992T1 (hr) * | 2012-05-17 | 2020-10-16 | Genentech, Inc. | Amorfni oblik pirimidinil-ciklopentanskog spoja koji inhibira akt, te njegovi pripravci i postupci |
| CN103923033B (zh) * | 2013-01-14 | 2015-11-18 | 天津药物研究院 | 具有抗胃溃疡作用的哌嗪类衍生物 |
| US10537552B2 (en) | 2015-05-05 | 2020-01-21 | Carafe Drug Innovation, Llc | Substituted 5-hydroxyoxindoles and their use as analgesics and fever reducers |
| CN108863949B (zh) * | 2018-07-09 | 2021-01-15 | 湖南博隽生物医药有限公司 | 一种用于治疗慢性炎性痛的辣椒素受体拮抗剂及合成方法 |
| PY2311120A (es) * | 2022-03-01 | 2023-09-14 | Syngenta Crop Protection Ag | Compuestos herbicidas |
| CN120398870A (zh) * | 2024-01-31 | 2025-08-01 | 深圳晶蛋生物医药科技有限公司 | 一种苯并吗啉类化合物及其应用 |
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- 2005-02-11 JP JP2006553265A patent/JP2007522235A/ja not_active Withdrawn
- 2005-02-11 BR BRPI0507927-6A patent/BRPI0507927A/pt not_active IP Right Cessation
- 2005-02-11 EP EP05722962A patent/EP1720868B1/en not_active Expired - Lifetime
- 2005-02-11 KR KR1020067018172A patent/KR100813093B1/ko not_active Expired - Fee Related
- 2005-02-11 AT AT05722962T patent/ATE447570T1/de not_active IP Right Cessation
- 2005-02-11 CN CNA200580008675XA patent/CN1953976A/zh active Pending
- 2005-02-11 US US11/056,568 patent/US7511044B2/en not_active Expired - Fee Related
- 2005-02-11 WO PCT/US2005/004378 patent/WO2005077944A1/en not_active Ceased
- 2005-02-11 AU AU2005212517A patent/AU2005212517B2/en not_active Ceased
- 2005-02-11 AR ARP050100490A patent/AR049771A1/es not_active Application Discontinuation
- 2005-02-11 DE DE602005017468T patent/DE602005017468D1/de not_active Expired - Fee Related
- 2005-02-14 TW TW094104222A patent/TWI295670B/zh active
-
2006
- 2006-08-08 IL IL177369A patent/IL177369A0/en unknown
- 2006-09-08 NO NO20064055A patent/NO20064055L/no not_active Application Discontinuation
- 2006-09-08 ZA ZA200607518A patent/ZA200607518B/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| EA200601426A1 (ru) | 2007-02-27 |
| AR049771A1 (es) | 2006-09-06 |
| ES2333973T3 (es) | 2010-03-03 |
| US20050176726A1 (en) | 2005-08-11 |
| DE602005017468D1 (de) | 2009-12-17 |
| ZA200607518B (en) | 2008-07-30 |
| KR20070033325A (ko) | 2007-03-26 |
| AU2005212517A1 (en) | 2005-08-25 |
| EP1720868B1 (en) | 2009-11-04 |
| US7511044B2 (en) | 2009-03-31 |
| EP1720868A1 (en) | 2006-11-15 |
| ATE447570T1 (de) | 2009-11-15 |
| IL177369A0 (en) | 2006-12-10 |
| CN1953976A (zh) | 2007-04-25 |
| WO2005077944A1 (en) | 2005-08-25 |
| EA010265B1 (ru) | 2008-06-30 |
| KR100813093B1 (ko) | 2008-03-17 |
| NO20064055L (no) | 2006-10-24 |
| JP2007522235A (ja) | 2007-08-09 |
| BRPI0507927A (pt) | 2007-07-17 |
| CA2555685A1 (en) | 2005-08-25 |
| AU2005212517B2 (en) | 2009-05-21 |
| MY139645A (en) | 2009-10-30 |
| TW200534858A (en) | 2005-11-01 |
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