TW200813067A - Nicotinic acetylcholine receptor ligands - Google Patents
Nicotinic acetylcholine receptor ligands Download PDFInfo
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- TW200813067A TW200813067A TW096116654A TW96116654A TW200813067A TW 200813067 A TW200813067 A TW 200813067A TW 096116654 A TW096116654 A TW 096116654A TW 96116654 A TW96116654 A TW 96116654A TW 200813067 A TW200813067 A TW 200813067A
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Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
- C07D491/22—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains four or more hetero rings
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- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/439—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom the ring forming part of a bridged ring system, e.g. quinuclidine
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- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
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- A—HUMAN NECESSITIES
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- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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- A61P25/00—Drugs for disorders of the nervous system
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
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- Addiction (AREA)
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- Anesthesiology (AREA)
- Psychology (AREA)
- Hospice & Palliative Care (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Steroid Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
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| US74747606P | 2006-05-17 | 2006-05-17 | |
| US82497506P | 2006-09-08 | 2006-09-08 |
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| TW200813067A true TW200813067A (en) | 2008-03-16 |
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| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| TW096116654A TW200813067A (en) | 2006-05-17 | 2007-05-10 | Nicotinic acetylcholine receptor ligands |
Country Status (19)
| Country | Link |
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| US (2) | US7842803B2 (enExample) |
| EP (1) | EP2019831B1 (enExample) |
| JP (1) | JP2009537517A (enExample) |
| KR (1) | KR20090007753A (enExample) |
| AR (1) | AR060914A1 (enExample) |
| AU (1) | AU2007250560B2 (enExample) |
| BR (1) | BRPI0711941A2 (enExample) |
| CA (1) | CA2652610A1 (enExample) |
| CL (1) | CL2007001405A1 (enExample) |
| EC (1) | ECSP088971A (enExample) |
| ES (1) | ES2392997T3 (enExample) |
| IL (1) | IL195019A0 (enExample) |
| MX (1) | MX2008014436A (enExample) |
| NO (1) | NO20084915L (enExample) |
| RU (1) | RU2441007C2 (enExample) |
| SA (1) | SA07280244B1 (enExample) |
| TW (1) | TW200813067A (enExample) |
| UY (1) | UY30349A1 (enExample) |
| WO (1) | WO2007133155A1 (enExample) |
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN112823157A (zh) * | 2018-07-13 | 2021-05-18 | 吉瑞工厂 | 螺色满衍生物 |
Families Citing this family (16)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB0220581D0 (en) | 2002-09-04 | 2002-10-09 | Novartis Ag | Organic Compound |
| PE20060437A1 (es) | 2004-06-18 | 2006-06-08 | Novartis Ag | COMPUESTOS AZA-BICICLONONANOS COMO LIGANDOS COLINERGICOS DE nAChR |
| GB0415746D0 (en) | 2004-07-14 | 2004-08-18 | Novartis Ag | Organic compounds |
| GB0521508D0 (en) | 2005-10-21 | 2005-11-30 | Novartis Ag | Organic compounds |
| GB0525673D0 (en) | 2005-12-16 | 2006-01-25 | Novartis Ag | Organic compounds |
| GB0525672D0 (en) | 2005-12-16 | 2006-01-25 | Novartis Ag | Organic compounds |
| WO2009066107A1 (en) * | 2007-11-21 | 2009-05-28 | Astrazeneca Ab | Use of a nicotinic receptor agonist |
| TWI558398B (zh) | 2009-09-22 | 2016-11-21 | 諾華公司 | 菸鹼乙醯膽鹼受體α７活化劑之用途 |
| BR112013018726A2 (pt) | 2011-01-27 | 2016-10-25 | Novartis Ag | uso de ativadores de alfa 7 do receptor nicotínico de acetilcolina |
| MX2013010698A (es) | 2011-03-18 | 2014-02-17 | Novartis Ag | Combinaciones de activadores del receptor de acetil-colina nicotinico alfa-7 y antagonistas del receptor de glutamato metabotropico 5 (mglur5) para usarse en la discinesia inducida por dopamina en la enfermedad de parkinson. |
| AU2012324458B2 (en) | 2011-10-20 | 2016-05-19 | Novartis Ag | Biomarkers predictive of responsiveness to alpha 7 nicotinic acetylcholine receptor activator treatment |
| JP6114951B2 (ja) | 2012-12-11 | 2017-04-19 | ノバルティス アーゲー | アルファ７ニコチン性アセチルコリン受容体アクチベーターによる処置に対する応答性を予測するバイオマーカー |
| JP2016508159A (ja) | 2013-01-15 | 2016-03-17 | ノバルティス アーゲー | アルファ７ニコチン性アセチルコリン受容体アゴニストの使用 |
| KR101879920B1 (ko) | 2013-01-15 | 2018-07-18 | 노파르티스 아게 | 알파 7 니코틴성 아세틸콜린 수용체 작용물질의 용도 |
| CN105263492B (zh) | 2013-01-15 | 2018-04-10 | 诺华有限公司 | α7烟碱型乙酰胆碱受体激动剂在治疗发作性睡病中的应用 |
| US11209254B2 (en) * | 2016-03-09 | 2021-12-28 | Msato, Llc | Pellet shaped marking round for air rifles and pistols |
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| AR013184A1 (es) * | 1997-07-18 | 2000-12-13 | Astrazeneca Ab | Aminas heterociclicas espiroazobiciclicas, composicion farmaceutica, uso de dichas aminas para preparar medicamentos y metodo de tratamiento o profilaxis |
| DK1397366T3 (da) * | 2001-06-01 | 2007-05-07 | Astrazeneca Ab | Hidtil ukendt ligander for nicotinacetylcholinreceptorer egnede i terapi |
| EP1499618B1 (en) * | 2002-04-18 | 2010-10-13 | AstraZeneca AB | Furyl compounds |
| KR20040099446A (ko) * | 2002-04-18 | 2004-11-26 | 아스트라제네카 아베 | 헤테로시클릭 화합물 |
| CN1325499C (zh) * | 2002-04-18 | 2007-07-11 | 阿斯特拉曾尼卡有限公司 | 噻吩基化合物 |
| EP1668016A1 (en) * | 2003-09-25 | 2006-06-14 | AstraZeneca AB | Ligands |
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2007
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- 2007-05-14 SA SA07280244A patent/SA07280244B1/ar unknown
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- 2007-05-16 JP JP2009510923A patent/JP2009537517A/ja active Pending
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- 2007-05-16 KR KR1020087027857A patent/KR20090007753A/ko not_active Abandoned
- 2007-05-16 CL CL2007001405A patent/CL2007001405A1/es unknown
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- 2007-05-16 AU AU2007250560A patent/AU2007250560B2/en not_active Ceased
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- 2007-05-16 WO PCT/SE2007/000485 patent/WO2007133155A1/en not_active Ceased
- 2007-05-16 CA CA002652610A patent/CA2652610A1/en not_active Abandoned
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2008
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- 2008-12-12 EC EC2008008971A patent/ECSP088971A/es unknown
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2010
- 2010-11-05 US US12/940,449 patent/US20110136804A1/en not_active Abandoned
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN112823157A (zh) * | 2018-07-13 | 2021-05-18 | 吉瑞工厂 | 螺色满衍生物 |
Also Published As
| Publication number | Publication date |
|---|---|
| ES2392997T3 (es) | 2012-12-17 |
| UY30349A1 (es) | 2008-01-02 |
| CA2652610A1 (en) | 2007-11-22 |
| SA07280244B1 (ar) | 2011-06-22 |
| WO2007133155A1 (en) | 2007-11-22 |
| EP2019831B1 (en) | 2012-09-12 |
| AU2007250560B2 (en) | 2011-06-23 |
| RU2441007C2 (ru) | 2012-01-27 |
| US20110136804A1 (en) | 2011-06-09 |
| NO20084915L (no) | 2009-02-13 |
| AU2007250560A1 (en) | 2007-11-22 |
| MX2008014436A (es) | 2008-11-27 |
| US7842803B2 (en) | 2010-11-30 |
| EP2019831A1 (en) | 2009-02-04 |
| EP2019831A4 (en) | 2010-06-09 |
| BRPI0711941A2 (pt) | 2011-12-13 |
| JP2009537517A (ja) | 2009-10-29 |
| AR060914A1 (es) | 2008-07-23 |
| US20080139600A1 (en) | 2008-06-12 |
| CL2007001405A1 (es) | 2008-01-25 |
| KR20090007753A (ko) | 2009-01-20 |
| RU2008143450A (ru) | 2010-06-27 |
| ECSP088971A (es) | 2009-01-30 |
| IL195019A0 (en) | 2009-08-03 |
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