SA07280244B1 - مركبات ترابطية لمستقبل الاسيتيل كولين النيكوتيني - Google Patents
مركبات ترابطية لمستقبل الاسيتيل كولين النيكوتيني Download PDFInfo
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- SA07280244B1 SA07280244B1 SA07280244A SA07280244A SA07280244B1 SA 07280244 B1 SA07280244 B1 SA 07280244B1 SA 07280244 A SA07280244 A SA 07280244A SA 07280244 A SA07280244 A SA 07280244A SA 07280244 B1 SA07280244 B1 SA 07280244B1
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Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
- C07D491/22—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains four or more hetero rings
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- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/439—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom the ring forming part of a bridged ring system, e.g. quinuclidine
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- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
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- A—HUMAN NECESSITIES
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- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
- A61P25/16—Anti-Parkinson drugs
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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- A61P25/20—Hypnotics; Sedatives
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- A—HUMAN NECESSITIES
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- A61P25/00—Drugs for disorders of the nervous system
- A61P25/22—Anxiolytics
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- A—HUMAN NECESSITIES
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- A61P25/00—Drugs for disorders of the nervous system
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- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
- A61P25/34—Tobacco-abuse
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
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- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Neurosurgery (AREA)
- Chemical Kinetics & Catalysis (AREA)
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- Addiction (AREA)
- Pain & Pain Management (AREA)
- Anesthesiology (AREA)
- Psychology (AREA)
- Hospice & Palliative Care (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Steroid Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US74747606P | 2006-05-17 | 2006-05-17 | |
| US82497506P | 2006-09-08 | 2006-09-08 |
Publications (1)
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|---|---|
| SA07280244B1 true SA07280244B1 (ar) | 2011-06-22 |
Family
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Family Applications (1)
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| SA07280244A SA07280244B1 (ar) | 2006-05-17 | 2007-05-14 | مركبات ترابطية لمستقبل الاسيتيل كولين النيكوتيني |
Country Status (19)
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|---|---|
| US (2) | US7842803B2 (enExample) |
| EP (1) | EP2019831B1 (enExample) |
| JP (1) | JP2009537517A (enExample) |
| KR (1) | KR20090007753A (enExample) |
| AR (1) | AR060914A1 (enExample) |
| AU (1) | AU2007250560B2 (enExample) |
| BR (1) | BRPI0711941A2 (enExample) |
| CA (1) | CA2652610A1 (enExample) |
| CL (1) | CL2007001405A1 (enExample) |
| EC (1) | ECSP088971A (enExample) |
| ES (1) | ES2392997T3 (enExample) |
| IL (1) | IL195019A0 (enExample) |
| MX (1) | MX2008014436A (enExample) |
| NO (1) | NO20084915L (enExample) |
| RU (1) | RU2441007C2 (enExample) |
| SA (1) | SA07280244B1 (enExample) |
| TW (1) | TW200813067A (enExample) |
| UY (1) | UY30349A1 (enExample) |
| WO (1) | WO2007133155A1 (enExample) |
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| GB0220581D0 (en) | 2002-09-04 | 2002-10-09 | Novartis Ag | Organic Compound |
| PE20060437A1 (es) | 2004-06-18 | 2006-06-08 | Novartis Ag | COMPUESTOS AZA-BICICLONONANOS COMO LIGANDOS COLINERGICOS DE nAChR |
| GB0415746D0 (en) | 2004-07-14 | 2004-08-18 | Novartis Ag | Organic compounds |
| GB0521508D0 (en) | 2005-10-21 | 2005-11-30 | Novartis Ag | Organic compounds |
| GB0525673D0 (en) | 2005-12-16 | 2006-01-25 | Novartis Ag | Organic compounds |
| GB0525672D0 (en) | 2005-12-16 | 2006-01-25 | Novartis Ag | Organic compounds |
| WO2009066107A1 (en) * | 2007-11-21 | 2009-05-28 | Astrazeneca Ab | Use of a nicotinic receptor agonist |
| JO3250B1 (ar) | 2009-09-22 | 2018-09-16 | Novartis Ag | إستعمال منشطات مستقبل نيكوتينيك أسيتيل كولين ألفا 7 |
| AU2012210652B2 (en) | 2011-01-27 | 2016-04-07 | Novartis Ag | Use of nicotinic acetylcholine receptor alpha 7 activators |
| KR20140018286A (ko) | 2011-03-18 | 2014-02-12 | 노파르티스 아게 | 파킨슨병에서의 도파민 유발 이상운동증에서 사용하기 위한 알파 7 니코틴성 아세틸콜린 수용체 활성화제 및 mGluR5 길항제의 조합물 |
| CA2852268C (en) | 2011-10-20 | 2020-08-25 | Novartis Ag | Biomarkers predictive of responsiveness to alpha 7 nicotinic acetylcholine receptor activator treatment |
| ES2661050T3 (es) | 2012-12-11 | 2018-03-27 | Novartis Ag | Biomarcador predictivo de la capacidad de respuesta a tratamiento con activador del receptor nicotínico de acetilcolina alfa-7 |
| CA2898043C (en) | 2013-01-15 | 2019-08-06 | Novartis Ag | Use of alpha 7 nicotinic receptor agonists for the treatment of narcolepsy |
| CA2898045C (en) | 2013-01-15 | 2018-08-28 | Novartis Ag | Use of alpha 7 nicotinic acetylcholine receptor agonists |
| CN105263495B (zh) | 2013-01-15 | 2019-05-14 | 诺华有限公司 | α7烟碱型乙酰胆碱受体激动剂的应用 |
| WO2017156309A1 (en) * | 2016-03-09 | 2017-09-14 | Msato, Llc | Pellet shaped marking round for air rifles and pistols |
| HU231333B1 (hu) * | 2018-07-13 | 2023-01-28 | Richter Gedeon Nyrt | Spirokromán származékok |
Family Cites Families (6)
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| AR013184A1 (es) * | 1997-07-18 | 2000-12-13 | Astrazeneca Ab | Aminas heterociclicas espiroazobiciclicas, composicion farmaceutica, uso de dichas aminas para preparar medicamentos y metodo de tratamiento o profilaxis |
| SI1397366T1 (sl) * | 2001-06-01 | 2007-06-30 | Astrazeneca Ab | Nov ligand za nikotinske acetilholinske receptorje, koristen v terapiji |
| KR20040099447A (ko) * | 2002-04-18 | 2004-11-26 | 아스트라제네카 아베 | 푸릴 화합물 |
| CN1325501C (zh) * | 2002-04-18 | 2007-07-11 | 阿斯特拉曾尼卡有限公司 | 杂环化合物 |
| AU2003224545B2 (en) * | 2002-04-18 | 2009-08-13 | Astrazeneca Ab | Thienyl compounds |
| EP1668016A1 (en) * | 2003-09-25 | 2006-06-14 | AstraZeneca AB | Ligands |
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2007
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- 2007-05-14 SA SA07280244A patent/SA07280244B1/ar unknown
- 2007-05-14 AR ARP070102066A patent/AR060914A1/es not_active Application Discontinuation
- 2007-05-15 UY UY30349A patent/UY30349A1/es not_active Application Discontinuation
- 2007-05-16 ES ES07748149T patent/ES2392997T3/es active Active
- 2007-05-16 EP EP07748149A patent/EP2019831B1/en active Active
- 2007-05-16 BR BRPI0711941-0A patent/BRPI0711941A2/pt not_active IP Right Cessation
- 2007-05-16 AU AU2007250560A patent/AU2007250560B2/en not_active Ceased
- 2007-05-16 KR KR1020087027857A patent/KR20090007753A/ko not_active Abandoned
- 2007-05-16 CA CA002652610A patent/CA2652610A1/en not_active Abandoned
- 2007-05-16 CL CL2007001405A patent/CL2007001405A1/es unknown
- 2007-05-16 RU RU2008143450/04A patent/RU2441007C2/ru not_active IP Right Cessation
- 2007-05-16 JP JP2009510923A patent/JP2009537517A/ja active Pending
- 2007-05-16 WO PCT/SE2007/000485 patent/WO2007133155A1/en not_active Ceased
- 2007-05-16 MX MX2008014436A patent/MX2008014436A/es not_active Application Discontinuation
- 2007-05-17 US US11/749,820 patent/US7842803B2/en active Active
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2008
- 2008-10-30 IL IL195019A patent/IL195019A0/en unknown
- 2008-11-21 NO NO20084915A patent/NO20084915L/no not_active Application Discontinuation
- 2008-12-12 EC EC2008008971A patent/ECSP088971A/es unknown
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2010
- 2010-11-05 US US12/940,449 patent/US20110136804A1/en not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| CA2652610A1 (en) | 2007-11-22 |
| AU2007250560A1 (en) | 2007-11-22 |
| AR060914A1 (es) | 2008-07-23 |
| US20110136804A1 (en) | 2011-06-09 |
| AU2007250560B2 (en) | 2011-06-23 |
| RU2441007C2 (ru) | 2012-01-27 |
| NO20084915L (no) | 2009-02-13 |
| EP2019831A4 (en) | 2010-06-09 |
| JP2009537517A (ja) | 2009-10-29 |
| BRPI0711941A2 (pt) | 2011-12-13 |
| TW200813067A (en) | 2008-03-16 |
| IL195019A0 (en) | 2009-08-03 |
| KR20090007753A (ko) | 2009-01-20 |
| MX2008014436A (es) | 2008-11-27 |
| US7842803B2 (en) | 2010-11-30 |
| ES2392997T3 (es) | 2012-12-17 |
| US20080139600A1 (en) | 2008-06-12 |
| RU2008143450A (ru) | 2010-06-27 |
| EP2019831A1 (en) | 2009-02-04 |
| EP2019831B1 (en) | 2012-09-12 |
| UY30349A1 (es) | 2008-01-02 |
| WO2007133155A1 (en) | 2007-11-22 |
| CL2007001405A1 (es) | 2008-01-25 |
| ECSP088971A (es) | 2009-01-30 |
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