MX2008014436A - Ligandos receptores de acetilcolina nicotinica 101. - Google Patents
Ligandos receptores de acetilcolina nicotinica 101.Info
- Publication number
- MX2008014436A MX2008014436A MX2008014436A MX2008014436A MX2008014436A MX 2008014436 A MX2008014436 A MX 2008014436A MX 2008014436 A MX2008014436 A MX 2008014436A MX 2008014436 A MX2008014436 A MX 2008014436A MX 2008014436 A MX2008014436 A MX 2008014436A
- Authority
- MX
- Mexico
- Prior art keywords
- pyridine
- azabicyclo
- spiro
- octane
- furyl
- Prior art date
Links
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
- C07D491/22—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains four or more hetero rings
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- A—HUMAN NECESSITIES
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/439—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom the ring forming part of a bridged ring system, e.g. quinuclidine
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- A—HUMAN NECESSITIES
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- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
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- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
- A61P25/16—Anti-Parkinson drugs
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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- A61P25/20—Hypnotics; Sedatives
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- A61P25/22—Anxiolytics
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- A—HUMAN NECESSITIES
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
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- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
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- Anesthesiology (AREA)
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- Hospice & Palliative Care (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Steroid Compounds (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US74747606P | 2006-05-17 | 2006-05-17 | |
| US82497506P | 2006-09-08 | 2006-09-08 | |
| PCT/SE2007/000485 WO2007133155A1 (en) | 2006-05-17 | 2007-05-16 | Nicotinic acetylcholine receptor ligands 101 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| MX2008014436A true MX2008014436A (es) | 2008-11-27 |
Family
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Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| MX2008014436A MX2008014436A (es) | 2006-05-17 | 2007-05-16 | Ligandos receptores de acetilcolina nicotinica 101. |
Country Status (19)
| Country | Link |
|---|---|
| US (2) | US7842803B2 (enExample) |
| EP (1) | EP2019831B1 (enExample) |
| JP (1) | JP2009537517A (enExample) |
| KR (1) | KR20090007753A (enExample) |
| AR (1) | AR060914A1 (enExample) |
| AU (1) | AU2007250560B2 (enExample) |
| BR (1) | BRPI0711941A2 (enExample) |
| CA (1) | CA2652610A1 (enExample) |
| CL (1) | CL2007001405A1 (enExample) |
| EC (1) | ECSP088971A (enExample) |
| ES (1) | ES2392997T3 (enExample) |
| IL (1) | IL195019A0 (enExample) |
| MX (1) | MX2008014436A (enExample) |
| NO (1) | NO20084915L (enExample) |
| RU (1) | RU2441007C2 (enExample) |
| SA (1) | SA07280244B1 (enExample) |
| TW (1) | TW200813067A (enExample) |
| UY (1) | UY30349A1 (enExample) |
| WO (1) | WO2007133155A1 (enExample) |
Families Citing this family (17)
| Publication number | Priority date | Publication date | Assignee | Title |
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| GB0220581D0 (en) | 2002-09-04 | 2002-10-09 | Novartis Ag | Organic Compound |
| PE20060437A1 (es) | 2004-06-18 | 2006-06-08 | Novartis Ag | COMPUESTOS AZA-BICICLONONANOS COMO LIGANDOS COLINERGICOS DE nAChR |
| GB0415746D0 (en) | 2004-07-14 | 2004-08-18 | Novartis Ag | Organic compounds |
| GB0521508D0 (en) | 2005-10-21 | 2005-11-30 | Novartis Ag | Organic compounds |
| GB0525673D0 (en) | 2005-12-16 | 2006-01-25 | Novartis Ag | Organic compounds |
| GB0525672D0 (en) | 2005-12-16 | 2006-01-25 | Novartis Ag | Organic compounds |
| WO2009066107A1 (en) * | 2007-11-21 | 2009-05-28 | Astrazeneca Ab | Use of a nicotinic receptor agonist |
| TWI558398B (zh) | 2009-09-22 | 2016-11-21 | 諾華公司 | 菸鹼乙醯膽鹼受體α７活化劑之用途 |
| BR112013018726A2 (pt) | 2011-01-27 | 2016-10-25 | Novartis Ag | uso de ativadores de alfa 7 do receptor nicotínico de acetilcolina |
| MX2013010698A (es) | 2011-03-18 | 2014-02-17 | Novartis Ag | Combinaciones de activadores del receptor de acetil-colina nicotinico alfa-7 y antagonistas del receptor de glutamato metabotropico 5 (mglur5) para usarse en la discinesia inducida por dopamina en la enfermedad de parkinson. |
| AU2012324458B2 (en) | 2011-10-20 | 2016-05-19 | Novartis Ag | Biomarkers predictive of responsiveness to alpha 7 nicotinic acetylcholine receptor activator treatment |
| JP6114951B2 (ja) | 2012-12-11 | 2017-04-19 | ノバルティス アーゲー | アルファ７ニコチン性アセチルコリン受容体アクチベーターによる処置に対する応答性を予測するバイオマーカー |
| JP2016508159A (ja) | 2013-01-15 | 2016-03-17 | ノバルティス アーゲー | アルファ７ニコチン性アセチルコリン受容体アゴニストの使用 |
| KR101879920B1 (ko) | 2013-01-15 | 2018-07-18 | 노파르티스 아게 | 알파 7 니코틴성 아세틸콜린 수용체 작용물질의 용도 |
| CN105263492B (zh) | 2013-01-15 | 2018-04-10 | 诺华有限公司 | α7烟碱型乙酰胆碱受体激动剂在治疗发作性睡病中的应用 |
| US11209254B2 (en) * | 2016-03-09 | 2021-12-28 | Msato, Llc | Pellet shaped marking round for air rifles and pistols |
| HU231333B1 (hu) * | 2018-07-13 | 2023-01-28 | Richter Gedeon Nyrt | Spirokromán származékok |
Family Cites Families (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AR013184A1 (es) * | 1997-07-18 | 2000-12-13 | Astrazeneca Ab | Aminas heterociclicas espiroazobiciclicas, composicion farmaceutica, uso de dichas aminas para preparar medicamentos y metodo de tratamiento o profilaxis |
| DK1397366T3 (da) * | 2001-06-01 | 2007-05-07 | Astrazeneca Ab | Hidtil ukendt ligander for nicotinacetylcholinreceptorer egnede i terapi |
| EP1499618B1 (en) * | 2002-04-18 | 2010-10-13 | AstraZeneca AB | Furyl compounds |
| KR20040099446A (ko) * | 2002-04-18 | 2004-11-26 | 아스트라제네카 아베 | 헤테로시클릭 화합물 |
| CN1325499C (zh) * | 2002-04-18 | 2007-07-11 | 阿斯特拉曾尼卡有限公司 | 噻吩基化合物 |
| EP1668016A1 (en) * | 2003-09-25 | 2006-06-14 | AstraZeneca AB | Ligands |
-
2007
- 2007-05-10 TW TW096116654A patent/TW200813067A/zh unknown
- 2007-05-14 AR ARP070102066A patent/AR060914A1/es not_active Application Discontinuation
- 2007-05-14 SA SA07280244A patent/SA07280244B1/ar unknown
- 2007-05-15 UY UY30349A patent/UY30349A1/es not_active Application Discontinuation
- 2007-05-16 JP JP2009510923A patent/JP2009537517A/ja active Pending
- 2007-05-16 EP EP07748149A patent/EP2019831B1/en active Active
- 2007-05-16 MX MX2008014436A patent/MX2008014436A/es not_active Application Discontinuation
- 2007-05-16 KR KR1020087027857A patent/KR20090007753A/ko not_active Abandoned
- 2007-05-16 CL CL2007001405A patent/CL2007001405A1/es unknown
- 2007-05-16 RU RU2008143450/04A patent/RU2441007C2/ru not_active IP Right Cessation
- 2007-05-16 AU AU2007250560A patent/AU2007250560B2/en not_active Ceased
- 2007-05-16 ES ES07748149T patent/ES2392997T3/es active Active
- 2007-05-16 WO PCT/SE2007/000485 patent/WO2007133155A1/en not_active Ceased
- 2007-05-16 CA CA002652610A patent/CA2652610A1/en not_active Abandoned
- 2007-05-16 BR BRPI0711941-0A patent/BRPI0711941A2/pt not_active IP Right Cessation
- 2007-05-17 US US11/749,820 patent/US7842803B2/en active Active
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2008
- 2008-10-30 IL IL195019A patent/IL195019A0/en unknown
- 2008-11-21 NO NO20084915A patent/NO20084915L/no not_active Application Discontinuation
- 2008-12-12 EC EC2008008971A patent/ECSP088971A/es unknown
-
2010
- 2010-11-05 US US12/940,449 patent/US20110136804A1/en not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| ES2392997T3 (es) | 2012-12-17 |
| UY30349A1 (es) | 2008-01-02 |
| CA2652610A1 (en) | 2007-11-22 |
| SA07280244B1 (ar) | 2011-06-22 |
| WO2007133155A1 (en) | 2007-11-22 |
| EP2019831B1 (en) | 2012-09-12 |
| AU2007250560B2 (en) | 2011-06-23 |
| RU2441007C2 (ru) | 2012-01-27 |
| US20110136804A1 (en) | 2011-06-09 |
| NO20084915L (no) | 2009-02-13 |
| AU2007250560A1 (en) | 2007-11-22 |
| US7842803B2 (en) | 2010-11-30 |
| TW200813067A (en) | 2008-03-16 |
| EP2019831A1 (en) | 2009-02-04 |
| EP2019831A4 (en) | 2010-06-09 |
| BRPI0711941A2 (pt) | 2011-12-13 |
| JP2009537517A (ja) | 2009-10-29 |
| AR060914A1 (es) | 2008-07-23 |
| US20080139600A1 (en) | 2008-06-12 |
| CL2007001405A1 (es) | 2008-01-25 |
| KR20090007753A (ko) | 2009-01-20 |
| RU2008143450A (ru) | 2010-06-27 |
| ECSP088971A (es) | 2009-01-30 |
| IL195019A0 (en) | 2009-08-03 |
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Legal Events
| Date | Code | Title | Description |
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| FA | Abandonment or withdrawal |