AU2007250560B2 - Nicotinic acetylcholine receptor ligands 101 - Google Patents
Nicotinic acetylcholine receptor ligands 101 Download PDFInfo
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- AU2007250560B2 AU2007250560B2 AU2007250560A AU2007250560A AU2007250560B2 AU 2007250560 B2 AU2007250560 B2 AU 2007250560B2 AU 2007250560 A AU2007250560 A AU 2007250560A AU 2007250560 A AU2007250560 A AU 2007250560A AU 2007250560 B2 AU2007250560 B2 AU 2007250560B2
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Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
- C07D491/22—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains four or more hetero rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
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- Hospice & Palliative Care (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Steroid Compounds (AREA)
Applications Claiming Priority (5)
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| US74747606P | 2006-05-17 | 2006-05-17 | |
| US60/747,476 | 2006-05-17 | ||
| US82497506P | 2006-09-08 | 2006-09-08 | |
| US60/824,975 | 2006-09-08 | ||
| PCT/SE2007/000485 WO2007133155A1 (en) | 2006-05-17 | 2007-05-16 | Nicotinic acetylcholine receptor ligands 101 |
Publications (2)
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| AU2007250560A1 AU2007250560A1 (en) | 2007-11-22 |
| AU2007250560B2 true AU2007250560B2 (en) | 2011-06-23 |
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| AU2007250560A Ceased AU2007250560B2 (en) | 2006-05-17 | 2007-05-16 | Nicotinic acetylcholine receptor ligands 101 |
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| EP (1) | EP2019831B1 (enExample) |
| JP (1) | JP2009537517A (enExample) |
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| GB0220581D0 (en) | 2002-09-04 | 2002-10-09 | Novartis Ag | Organic Compound |
| PE20060437A1 (es) | 2004-06-18 | 2006-06-08 | Novartis Ag | COMPUESTOS AZA-BICICLONONANOS COMO LIGANDOS COLINERGICOS DE nAChR |
| GB0415746D0 (en) | 2004-07-14 | 2004-08-18 | Novartis Ag | Organic compounds |
| GB0521508D0 (en) | 2005-10-21 | 2005-11-30 | Novartis Ag | Organic compounds |
| GB0525673D0 (en) | 2005-12-16 | 2006-01-25 | Novartis Ag | Organic compounds |
| GB0525672D0 (en) | 2005-12-16 | 2006-01-25 | Novartis Ag | Organic compounds |
| WO2009066107A1 (en) * | 2007-11-21 | 2009-05-28 | Astrazeneca Ab | Use of a nicotinic receptor agonist |
| TWI558398B (zh) | 2009-09-22 | 2016-11-21 | 諾華公司 | 菸鹼乙醯膽鹼受體α７活化劑之用途 |
| BR112013018726A2 (pt) | 2011-01-27 | 2016-10-25 | Novartis Ag | uso de ativadores de alfa 7 do receptor nicotínico de acetilcolina |
| MX2013010698A (es) | 2011-03-18 | 2014-02-17 | Novartis Ag | Combinaciones de activadores del receptor de acetil-colina nicotinico alfa-7 y antagonistas del receptor de glutamato metabotropico 5 (mglur5) para usarse en la discinesia inducida por dopamina en la enfermedad de parkinson. |
| AU2012324458B2 (en) | 2011-10-20 | 2016-05-19 | Novartis Ag | Biomarkers predictive of responsiveness to alpha 7 nicotinic acetylcholine receptor activator treatment |
| JP6114951B2 (ja) | 2012-12-11 | 2017-04-19 | ノバルティス アーゲー | アルファ７ニコチン性アセチルコリン受容体アクチベーターによる処置に対する応答性を予測するバイオマーカー |
| JP2016508159A (ja) | 2013-01-15 | 2016-03-17 | ノバルティス アーゲー | アルファ７ニコチン性アセチルコリン受容体アゴニストの使用 |
| KR101879920B1 (ko) | 2013-01-15 | 2018-07-18 | 노파르티스 아게 | 알파 7 니코틴성 아세틸콜린 수용체 작용물질의 용도 |
| CN105263492B (zh) | 2013-01-15 | 2018-04-10 | 诺华有限公司 | α7烟碱型乙酰胆碱受体激动剂在治疗发作性睡病中的应用 |
| US11209254B2 (en) * | 2016-03-09 | 2021-12-28 | Msato, Llc | Pellet shaped marking round for air rifles and pistols |
| HU231333B1 (hu) * | 2018-07-13 | 2023-01-28 | Richter Gedeon Nyrt | Spirokromán származékok |
Citations (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO1999003859A1 (en) * | 1997-07-18 | 1999-01-28 | Astra Aktiebolag | Novel spiroazabicyclic heterocyclic compounds |
| WO2002096912A1 (en) * | 2001-06-01 | 2002-12-05 | Astrazeneca Ab | Novel ligand for nicotinic acetylcholine receptors useful in therapy |
| WO2003087103A1 (en) * | 2002-04-18 | 2003-10-23 | Astrazeneca Ab | Thienyl compounds |
| WO2003087102A1 (en) * | 2002-04-18 | 2003-10-23 | Astrazeneca Ab | Furyl compounds |
| WO2003087104A1 (en) * | 2002-04-18 | 2003-10-23 | Astrazeneca Ab | Heterocyclic compounds |
| WO2005030778A1 (en) * | 2003-09-25 | 2005-04-07 | Astrazeneca Ab | Ligands |
-
2007
- 2007-05-10 TW TW096116654A patent/TW200813067A/zh unknown
- 2007-05-14 AR ARP070102066A patent/AR060914A1/es not_active Application Discontinuation
- 2007-05-14 SA SA07280244A patent/SA07280244B1/ar unknown
- 2007-05-15 UY UY30349A patent/UY30349A1/es not_active Application Discontinuation
- 2007-05-16 JP JP2009510923A patent/JP2009537517A/ja active Pending
- 2007-05-16 EP EP07748149A patent/EP2019831B1/en active Active
- 2007-05-16 MX MX2008014436A patent/MX2008014436A/es not_active Application Discontinuation
- 2007-05-16 KR KR1020087027857A patent/KR20090007753A/ko not_active Abandoned
- 2007-05-16 CL CL2007001405A patent/CL2007001405A1/es unknown
- 2007-05-16 RU RU2008143450/04A patent/RU2441007C2/ru not_active IP Right Cessation
- 2007-05-16 AU AU2007250560A patent/AU2007250560B2/en not_active Ceased
- 2007-05-16 ES ES07748149T patent/ES2392997T3/es active Active
- 2007-05-16 WO PCT/SE2007/000485 patent/WO2007133155A1/en not_active Ceased
- 2007-05-16 CA CA002652610A patent/CA2652610A1/en not_active Abandoned
- 2007-05-16 BR BRPI0711941-0A patent/BRPI0711941A2/pt not_active IP Right Cessation
- 2007-05-17 US US11/749,820 patent/US7842803B2/en active Active
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2008
- 2008-10-30 IL IL195019A patent/IL195019A0/en unknown
- 2008-11-21 NO NO20084915A patent/NO20084915L/no not_active Application Discontinuation
- 2008-12-12 EC EC2008008971A patent/ECSP088971A/es unknown
-
2010
- 2010-11-05 US US12/940,449 patent/US20110136804A1/en not_active Abandoned
Patent Citations (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO1999003859A1 (en) * | 1997-07-18 | 1999-01-28 | Astra Aktiebolag | Novel spiroazabicyclic heterocyclic compounds |
| WO2002096912A1 (en) * | 2001-06-01 | 2002-12-05 | Astrazeneca Ab | Novel ligand for nicotinic acetylcholine receptors useful in therapy |
| WO2003087103A1 (en) * | 2002-04-18 | 2003-10-23 | Astrazeneca Ab | Thienyl compounds |
| WO2003087102A1 (en) * | 2002-04-18 | 2003-10-23 | Astrazeneca Ab | Furyl compounds |
| WO2003087104A1 (en) * | 2002-04-18 | 2003-10-23 | Astrazeneca Ab | Heterocyclic compounds |
| WO2005030778A1 (en) * | 2003-09-25 | 2005-04-07 | Astrazeneca Ab | Ligands |
Also Published As
| Publication number | Publication date |
|---|---|
| ES2392997T3 (es) | 2012-12-17 |
| UY30349A1 (es) | 2008-01-02 |
| CA2652610A1 (en) | 2007-11-22 |
| SA07280244B1 (ar) | 2011-06-22 |
| WO2007133155A1 (en) | 2007-11-22 |
| EP2019831B1 (en) | 2012-09-12 |
| RU2441007C2 (ru) | 2012-01-27 |
| US20110136804A1 (en) | 2011-06-09 |
| NO20084915L (no) | 2009-02-13 |
| AU2007250560A1 (en) | 2007-11-22 |
| MX2008014436A (es) | 2008-11-27 |
| US7842803B2 (en) | 2010-11-30 |
| TW200813067A (en) | 2008-03-16 |
| EP2019831A1 (en) | 2009-02-04 |
| EP2019831A4 (en) | 2010-06-09 |
| BRPI0711941A2 (pt) | 2011-12-13 |
| JP2009537517A (ja) | 2009-10-29 |
| AR060914A1 (es) | 2008-07-23 |
| US20080139600A1 (en) | 2008-06-12 |
| CL2007001405A1 (es) | 2008-01-25 |
| KR20090007753A (ko) | 2009-01-20 |
| RU2008143450A (ru) | 2010-06-27 |
| ECSP088971A (es) | 2009-01-30 |
| IL195019A0 (en) | 2009-08-03 |
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