TR200202287T2 - Sübstitüe edilmiş N6 heterosiklik adenosin türevleri - Google Patents
Sübstitüe edilmiş N6 heterosiklik adenosin türevleriInfo
- Publication number
- TR200202287T2 TR200202287T2 TR2002/02287T TR200202287T TR200202287T2 TR 200202287 T2 TR200202287 T2 TR 200202287T2 TR 2002/02287 T TR2002/02287 T TR 2002/02287T TR 200202287 T TR200202287 T TR 200202287T TR 200202287 T2 TR200202287 T2 TR 200202287T2
- Authority
- TR
- Turkey
- Prior art keywords
- substituted
- heterocyclic
- adenosine derivatives
- formula
- group
- Prior art date
Links
- -1 heterocyclic adenosine derivatives Chemical class 0.000 title 1
- 102000009346 Adenosine receptors Human genes 0.000 abstract 1
- 108050000203 Adenosine receptors Proteins 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- 125000003700 epoxy group Chemical group 0.000 abstract 1
- 125000000623 heterocyclic group Chemical group 0.000 abstract 1
- 125000002950 monocyclic group Chemical group 0.000 abstract 1
- 125000003367 polycyclic group Chemical group 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
- C07H19/02—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
- C07H19/04—Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
- C07H19/16—Purine radicals
- C07H19/167—Purine radicals with ribosyl as the saccharide radical
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
- C07H19/02—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
- C07H19/04—Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
- C07H19/16—Purine radicals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/06—Antiarrhythmics
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- General Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Veterinary Medicine (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Public Health (AREA)
- Biochemistry (AREA)
- Molecular Biology (AREA)
- Genetics & Genomics (AREA)
- Biotechnology (AREA)
- Heart & Thoracic Surgery (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Cardiology (AREA)
- Diabetes (AREA)
- Endocrinology (AREA)
- Hospice & Palliative Care (AREA)
- Psychiatry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Saccharide Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Plural Heterocyclic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Abstract
Bir sübstitüe edilmis N6-oksa, tia, tioksa ve formül (1)' e sahip sübstitüe edilmis azasikloalkil adenosin reseptörü olarak bilesimi kullanmak için bir yöntem. Sözü geçen formülde, R1, en az bir tanesi N, 0 ve S(-O) 0-2 içeren gruptan seçilen 3 ila 15 atom ihtiva eden bir monosiklik ya da polisiklik heterosiklik gruptur, ve burada R1, bir epoksid grup içermemektedir.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US08702234 US5789416B1 (en) | 1996-08-27 | 1996-08-27 | N6 mono heterocyclic substituted adenosine derivatives |
Publications (1)
Publication Number | Publication Date |
---|---|
TR200202287T2 true TR200202287T2 (tr) | 2003-01-21 |
Family
ID=24820367
Family Applications (2)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
TR1999/00377T TR199900377T2 (tr) | 1996-08-27 | 1997-08-20 | Sübstitüe edilmis N6 heterosiklik adenosin türevleri. |
TR2002/02287T TR200202287T2 (tr) | 1996-08-27 | 1997-08-20 | Sübstitüe edilmiş N6 heterosiklik adenosin türevleri |
Family Applications Before (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
TR1999/00377T TR199900377T2 (tr) | 1996-08-27 | 1997-08-20 | Sübstitüe edilmis N6 heterosiklik adenosin türevleri. |
Country Status (25)
Country | Link |
---|---|
US (1) | US5789416B1 (tr) |
EP (3) | EP0992510B1 (tr) |
JP (1) | JP3157842B2 (tr) |
KR (1) | KR100331775B1 (tr) |
CN (1) | CN100363377C (tr) |
AT (2) | ATE202361T1 (tr) |
AU (1) | AU726597B2 (tr) |
BR (1) | BR9711444A (tr) |
CA (1) | CA2264155C (tr) |
CZ (1) | CZ296855B6 (tr) |
DE (2) | DE69719816T2 (tr) |
DK (2) | DK0920438T3 (tr) |
ES (2) | ES2157593T3 (tr) |
GE (1) | GEP20012419B (tr) |
GR (1) | GR3036332T3 (tr) |
HK (1) | HK1020967A1 (tr) |
HU (1) | HU226057B1 (tr) |
IL (2) | IL128652A0 (tr) |
NO (3) | NO312679B1 (tr) |
NZ (3) | NZ505428A (tr) |
PL (1) | PL187635B1 (tr) |
PT (1) | PT920438E (tr) |
TR (2) | TR199900377T2 (tr) |
UA (1) | UA62936C2 (tr) |
WO (1) | WO1998008855A2 (tr) |
Families Citing this family (61)
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JP2018531037A (ja) | 2015-10-19 | 2018-10-25 | アールエックスアイ ファーマシューティカルズ コーポレーション | 長い非コードrnaを標的とする減少したサイズの自己送達型核酸化合物 |
CN105218490B (zh) * | 2015-11-10 | 2017-05-03 | 山东川成医药股份有限公司 | 一种(r)‑3‑氨基四氢呋喃的制备方法 |
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1996
- 1996-08-27 US US08702234 patent/US5789416B1/en not_active Expired - Lifetime
-
1997
- 1997-08-20 DE DE69719816T patent/DE69719816T2/de not_active Expired - Lifetime
- 1997-08-20 ES ES97938502T patent/ES2157593T3/es not_active Expired - Lifetime
- 1997-08-20 KR KR1019997001563A patent/KR100331775B1/ko not_active IP Right Cessation
- 1997-08-20 IL IL12865297A patent/IL128652A0/xx active IP Right Grant
- 1997-08-20 CA CA002264155A patent/CA2264155C/en not_active Expired - Fee Related
- 1997-08-20 DK DK97938502T patent/DK0920438T3/da active
- 1997-08-20 UA UA99021148A patent/UA62936C2/uk unknown
- 1997-08-20 AU AU40809/97A patent/AU726597B2/en not_active Ceased
- 1997-08-20 CZ CZ0061499A patent/CZ296855B6/cs not_active IP Right Cessation
- 1997-08-20 NZ NZ505428A patent/NZ505428A/en unknown
- 1997-08-20 PL PL97331853A patent/PL187635B1/pl not_active IP Right Cessation
- 1997-08-20 WO PCT/US1997/014724 patent/WO1998008855A2/en active IP Right Grant
- 1997-08-20 DE DE69705312T patent/DE69705312T2/de not_active Expired - Lifetime
- 1997-08-20 TR TR1999/00377T patent/TR199900377T2/tr unknown
- 1997-08-20 JP JP51173698A patent/JP3157842B2/ja not_active Expired - Fee Related
- 1997-08-20 DK DK99119389T patent/DK0992510T3/da active
- 1997-08-20 BR BR9711444-8A patent/BR9711444A/pt active Search and Examination
- 1997-08-20 AT AT97938502T patent/ATE202361T1/de active
- 1997-08-20 AT AT99119389T patent/ATE234323T1/de active
- 1997-08-20 NZ NZ334095A patent/NZ334095A/xx not_active IP Right Cessation
- 1997-08-20 EP EP99119389A patent/EP0992510B1/en not_active Expired - Lifetime
- 1997-08-20 GE GEAP19974728A patent/GEP20012419B/en unknown
- 1997-08-20 ES ES99119389T patent/ES2189330T3/es not_active Expired - Lifetime
- 1997-08-20 TR TR2002/02287T patent/TR200202287T2/tr unknown
- 1997-08-20 EP EP97938502A patent/EP0920438B1/en not_active Expired - Lifetime
- 1997-08-20 CN CNB971991790A patent/CN100363377C/zh not_active Expired - Fee Related
- 1997-08-20 HU HU0001640A patent/HU226057B1/hu not_active IP Right Cessation
- 1997-08-20 PT PT97938502T patent/PT920438E/pt unknown
- 1997-08-20 EP EP00123879A patent/EP1081155A3/en not_active Withdrawn
-
1999
- 1999-02-19 NO NO19990787A patent/NO312679B1/no not_active IP Right Cessation
- 1999-02-22 IL IL128652A patent/IL128652A/en not_active IP Right Cessation
- 1999-12-30 HK HK99106191A patent/HK1020967A1/xx not_active IP Right Cessation
-
2001
- 2001-06-08 NZ NZ512242A patent/NZ512242A/xx not_active IP Right Cessation
- 2001-08-06 GR GR20010401184T patent/GR3036332T3/el unknown
-
2002
- 2002-02-15 NO NO20020759A patent/NO20020759D0/no not_active Application Discontinuation
- 2002-02-15 NO NO20020758A patent/NO322459B1/no not_active IP Right Cessation
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