SV2016005318A - Pirazolopiridinas y pirazolopirimidinas - Google Patents

Pirazolopiridinas y pirazolopirimidinas

Info

Publication number
SV2016005318A
SV2016005318A SV2016005318A SV2016005318A SV2016005318A SV 2016005318 A SV2016005318 A SV 2016005318A SV 2016005318 A SV2016005318 A SV 2016005318A SV 2016005318 A SV2016005318 A SV 2016005318A SV 2016005318 A SV2016005318 A SV 2016005318A
Authority
SV
El Salvador
Prior art keywords
rent
phenyl
independently
replaced
naftilo
Prior art date
Application number
SV2016005318A
Other languages
English (en)
Spanish (es)
Inventor
Jotham Wadsworth Coe
Christoph Martin Dehnhardt
Peter Jones
Yogesh Anil Sabnis
Joseph Walter Strohbach
Florian Michel Wakenhut
Gavin Alistair Whitlock
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=53264695&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=SV2016005318(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Pfizer filed Critical Pfizer
Publication of SV2016005318A publication Critical patent/SV2016005318A/es

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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
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    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/415—1,2-Diazoles
    • A61K31/4162—1,2-Diazoles condensed with heterocyclic ring systems
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
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    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
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    • C07D—HETEROCYCLIC COMPOUNDS
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    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Epidemiology (AREA)
  • Immunology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Diabetes (AREA)
  • Cardiology (AREA)
  • Hematology (AREA)
  • Pulmonology (AREA)
  • Rheumatology (AREA)
  • Neurology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Pain & Pain Management (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Ophthalmology & Optometry (AREA)
  • Endocrinology (AREA)
  • Obesity (AREA)
  • Oncology (AREA)
  • Reproductive Health (AREA)
  • Hospice & Palliative Care (AREA)
  • Communicable Diseases (AREA)
  • Urology & Nephrology (AREA)
  • Dermatology (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Gynecology & Obstetrics (AREA)
SV2016005318A 2014-05-14 2016-11-11 Pirazolopiridinas y pirazolopirimidinas SV2016005318A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201461993138P 2014-05-14 2014-05-14
PCT/IB2015/053174 WO2015173683A1 (en) 2014-05-14 2015-04-30 Pyrazolopyridines and pyrazolopyrimidines

Publications (1)

Publication Number Publication Date
SV2016005318A true SV2016005318A (es) 2017-03-06

Family

ID=53264695

Family Applications (1)

Application Number Title Priority Date Filing Date
SV2016005318A SV2016005318A (es) 2014-05-14 2016-11-11 Pirazolopiridinas y pirazolopirimidinas

Country Status (29)

Country Link
US (2) US9518052B2 (cg-RX-API-DMAC7.html)
EP (1) EP3143021B1 (cg-RX-API-DMAC7.html)
JP (1) JP6663857B2 (cg-RX-API-DMAC7.html)
KR (1) KR20170002623A (cg-RX-API-DMAC7.html)
CN (1) CN106459048A (cg-RX-API-DMAC7.html)
AP (1) AP2016009562A0 (cg-RX-API-DMAC7.html)
AR (1) AR100438A1 (cg-RX-API-DMAC7.html)
AU (1) AU2015260905A1 (cg-RX-API-DMAC7.html)
CA (1) CA2948587C (cg-RX-API-DMAC7.html)
CL (1) CL2016002888A1 (cg-RX-API-DMAC7.html)
CR (1) CR20160525A (cg-RX-API-DMAC7.html)
CU (1) CU20160167A7 (cg-RX-API-DMAC7.html)
DO (1) DOP2016000298A (cg-RX-API-DMAC7.html)
EA (1) EA201650029A1 (cg-RX-API-DMAC7.html)
EC (1) ECSP16087271A (cg-RX-API-DMAC7.html)
ES (1) ES2737696T3 (cg-RX-API-DMAC7.html)
GE (1) GEP20186921B (cg-RX-API-DMAC7.html)
IL (1) IL248970A0 (cg-RX-API-DMAC7.html)
MD (1) MD20160121A2 (cg-RX-API-DMAC7.html)
MX (1) MX2016014878A (cg-RX-API-DMAC7.html)
NI (1) NI201600170A (cg-RX-API-DMAC7.html)
PE (1) PE20161475A1 (cg-RX-API-DMAC7.html)
PH (1) PH12016502228A1 (cg-RX-API-DMAC7.html)
SG (1) SG11201609139WA (cg-RX-API-DMAC7.html)
SV (1) SV2016005318A (cg-RX-API-DMAC7.html)
TN (1) TN2016000503A1 (cg-RX-API-DMAC7.html)
TW (1) TWI591067B (cg-RX-API-DMAC7.html)
UY (1) UY36121A (cg-RX-API-DMAC7.html)
WO (1) WO2015173683A1 (cg-RX-API-DMAC7.html)

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JP6663857B2 (ja) 2014-05-14 2020-03-13 ファイザー・インク ピラゾロピリジンおよびピラゾロピリミジン
US9403810B2 (en) 2014-05-14 2016-08-02 Novartis Ag Carboxamide derivatives
PL3371185T3 (pl) 2015-11-03 2021-04-06 Topivert Pharma Limited Pochodne 4,5,6,7-tetrahydro-1h-imidazo[4,5-c]pirydyny i 1,4,5,6,7,8-heksahydroimidazo[4,5-d]azepiny jako inhibitory kinaz janusowych
EP3865481A1 (en) 2015-11-03 2021-08-18 Topivert Pharma Limited 4,5,6,7-tetrahydro-1h-imidazo[4,5-c]pyridine and 1,4,5,6,7,8-hexahydroimidazo[4,5-d]azepine derivatives as janus kinase inhibitors
HK1252685A1 (zh) 2015-11-03 2019-05-31 Theravance Biopharma R&D Ip, Llc 用於治疗呼吸疾病的jak激酶抑制剂化合物
EP3592743A1 (en) 2017-03-09 2020-01-15 Theravance Biopharma R&D IP, LLC Fused imidazo-piperidine jak inhibitors
AR111495A1 (es) 2017-05-01 2019-07-17 Theravance Biopharma R&D Ip Llc Compuestos de imidazo-piperidina fusionada como inhibidores de jak
CN110603255B (zh) 2017-05-01 2023-02-10 施万生物制药研发Ip有限责任公司 Jak抑制剂化合物的结晶型式
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