SK283952B6 - Pyrido [2,3-D]pyrimidíny a farmaceutické kompozície na ich báze - Google Patents

Pyrido [2,3-D]pyrimidíny a farmaceutické kompozície na ich báze Download PDF

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Publication number
SK283952B6
SK283952B6 SK1410-97A SK141097A SK283952B6 SK 283952 B6 SK283952 B6 SK 283952B6 SK 141097 A SK141097 A SK 141097A SK 283952 B6 SK283952 B6 SK 283952B6
Authority
SK
Slovakia
Prior art keywords
pyrimidin
pyrido
methyl
dichlorophenyl
phenyl
Prior art date
Application number
SK1410-97A
Other languages
English (en)
Slovak (sk)
Other versions
SK141097A3 (en
Inventor
Clifton John Blankley
Diane Harris Boschelli
Annette Marian Doherty
James Marino Hamby
Sylvester Klutchko
Robert Lee Panek
Original Assignee
Warner-Lambert Company
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US08/433,294 external-priority patent/US5620981A/en
Application filed by Warner-Lambert Company filed Critical Warner-Lambert Company
Publication of SK141097A3 publication Critical patent/SK141097A3/sk
Publication of SK283952B6 publication Critical patent/SK283952B6/sk

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • A61P17/06Antipsoriatics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Urology & Nephrology (AREA)
  • Vascular Medicine (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Dermatology (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
SK1410-97A 1995-05-03 1996-04-26 Pyrido [2,3-D]pyrimidíny a farmaceutické kompozície na ich báze SK283952B6 (sk)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US08/433,294 US5620981A (en) 1995-05-03 1995-05-03 Pyrido [2,3-D]pyrimidines for inhibiting protein tyrosine kinase mediated cellular proliferation
US08/611,279 US5733914A (en) 1995-05-03 1996-04-03 Pyrido 2, 3-d!pyrimidines for inhibiting protein tyrosine kinase mediated cellular proliferation
PCT/US1996/005819 WO1996034867A1 (fr) 1995-05-03 1996-04-26 PYRIDO[2,3-d]PYRIMIDINES DESTINEES A INHIBER LA PROLIFERATION CELLULAIRE INDUITE PAR LES TYROSINES KINASES

Publications (2)

Publication Number Publication Date
SK141097A3 SK141097A3 (en) 1998-07-08
SK283952B6 true SK283952B6 (sk) 2004-06-08

Family

ID=27029804

Family Applications (1)

Application Number Title Priority Date Filing Date
SK1410-97A SK283952B6 (sk) 1995-05-03 1996-04-26 Pyrido [2,3-D]pyrimidíny a farmaceutické kompozície na ich báze

Country Status (21)

Country Link
EP (1) EP0823908B1 (fr)
JP (1) JP3885116B2 (fr)
CN (1) CN1083452C (fr)
AT (1) ATE344263T1 (fr)
AU (1) AU713727B2 (fr)
BG (1) BG62617B1 (fr)
CA (1) CA2214219C (fr)
CZ (1) CZ288160B6 (fr)
DE (1) DE69636671T2 (fr)
EA (1) EA000897B1 (fr)
EE (1) EE03770B1 (fr)
ES (1) ES2274526T3 (fr)
GE (1) GEP20002032B (fr)
HU (1) HUP9801704A3 (fr)
IL (1) IL117923A (fr)
MX (1) MX9706529A (fr)
NO (1) NO310110B1 (fr)
NZ (1) NZ307021A (fr)
PL (1) PL184093B1 (fr)
SK (1) SK283952B6 (fr)
WO (1) WO1996034867A1 (fr)

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GB9508537D0 (en) * 1995-04-27 1995-06-14 Zeneca Ltd Quinazoline derivatives
GB9508565D0 (en) * 1995-04-27 1995-06-14 Zeneca Ltd Quiazoline derivative
US5932574A (en) * 1995-04-27 1999-08-03 Zeneca Limited Quinazoline derivatives
GB9508535D0 (en) * 1995-04-27 1995-06-14 Zeneca Ltd Quinazoline derivative
GB9624482D0 (en) 1995-12-18 1997-01-15 Zeneca Phaema S A Chemical compounds
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GB9603097D0 (en) * 1996-02-14 1996-04-10 Zeneca Ltd Quinazoline compounds
GB9603095D0 (en) * 1996-02-14 1996-04-10 Zeneca Ltd Quinazoline derivatives
NZ331191A (en) 1996-03-05 2000-03-27 Zeneca Ltd 4-anilinoquinazoline derivatives and pharmaceutical compositions thereof
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KR102329720B1 (ko) * 2019-08-30 2021-11-23 한국과학기술연구원 단백질 키나아제 저해 활성을 갖는 신규한 피리미도[4,5-d]피리미딘-2-온 유도체
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Also Published As

Publication number Publication date
CN1083452C (zh) 2002-04-24
BG102003A (en) 1998-12-30
JP3885116B2 (ja) 2007-02-21
SK141097A3 (en) 1998-07-08
AU713727B2 (en) 1999-12-09
IL117923A0 (en) 1996-08-04
HUP9801704A3 (en) 1999-03-01
ES2274526T3 (es) 2007-05-16
NO310110B1 (no) 2001-05-21
AU5576996A (en) 1996-11-21
PL323089A1 (en) 1998-03-02
DE69636671T2 (de) 2007-08-30
MX9706529A (es) 1997-11-29
NO975033D0 (no) 1997-10-31
CA2214219A1 (fr) 1996-11-07
HUP9801704A2 (hu) 1998-11-30
CZ327597A3 (cs) 1998-03-18
GEP20002032B (en) 2000-04-10
EP0823908B1 (fr) 2006-11-02
EA000897B1 (ru) 2000-06-26
CN1183099A (zh) 1998-05-27
NZ307021A (en) 2001-04-27
CA2214219C (fr) 2008-09-30
EE9700274A (et) 1998-06-15
JPH11504922A (ja) 1999-05-11
WO1996034867A1 (fr) 1996-11-07
BG62617B1 (bg) 2000-03-31
NO975033L (no) 1997-10-31
EP0823908A1 (fr) 1998-02-18
ATE344263T1 (de) 2006-11-15
IL117923A (en) 2000-06-01
EE03770B1 (et) 2002-06-17
DE69636671D1 (de) 2006-12-14
CZ288160B6 (en) 2001-05-16
EA199700356A1 (ru) 1998-06-25
PL184093B1 (pl) 2002-08-30

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