SK1852004A3 - Deriváty piperazínu s účinkami antagonistu receptora CCR1 - Google Patents

Deriváty piperazínu s účinkami antagonistu receptora CCR1 Download PDF

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Publication number
SK1852004A3
SK1852004A3 SK185-2004A SK1852004A SK1852004A3 SK 1852004 A3 SK1852004 A3 SK 1852004A3 SK 1852004 A SK1852004 A SK 1852004A SK 1852004 A3 SK1852004 A3 SK 1852004A3
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Slovakia
Prior art keywords
alkyl
carbon atoms
moiety
group
heteroaryl
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SK185-2004A
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English (en)
Slovak (sk)
Inventor
Laura Cook Blumberg
Matthew Frank Brown
Matthew Merrill Hayward
Christopher Stanley Poss
Gregory Dean Lundquist Jr.
Andrei Shavnya
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Pfizer Products Inc.
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Publication of SK1852004A3 publication Critical patent/SK1852004A3/sk

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    • C07D241/02—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings
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    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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    • C07D213/74—Amino or imino radicals substituted by hydrocarbon or substituted hydrocarbon radicals
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    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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SK185-2004A 2001-10-22 2002-09-26 Deriváty piperazínu s účinkami antagonistu receptora CCR1 SK1852004A3 (sk)

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EP1438298B1 (en) 2010-01-27
OA12670A (en) 2006-06-20
UY27503A1 (es) 2003-06-30
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EA006243B1 (ru) 2005-10-27
CZ2004519A3 (cs) 2004-12-15
JP2005507923A (ja) 2005-03-24
US20040034034A1 (en) 2004-02-19
MXPA04002423A (es) 2004-05-31
CN1575283A (zh) 2005-02-02
EE200400088A (et) 2004-10-15
HUP0401735A2 (hu) 2005-01-28
ES2337241T3 (es) 2010-04-22
ECSP045073A (es) 2004-05-28
PE20030568A1 (es) 2003-07-07
PA8556901A1 (es) 2003-11-12
ATE456559T1 (de) 2010-02-15
BR0213452A (pt) 2004-11-09
CA2463272C (en) 2009-11-17
BG108674A (en) 2005-04-30
IS7180A (is) 2004-03-11
IL160974A0 (en) 2004-08-31
EA200400466A1 (ru) 2004-08-26
AP2004003008A0 (en) 2004-06-30
EP1438298A1 (en) 2004-07-21
HN2002000300A (es) 2003-10-17
HUP0401735A3 (en) 2005-06-28
MA27142A1 (fr) 2005-01-03
DK1438298T3 (da) 2010-04-12
AR037742A1 (es) 2004-12-01
WO2003035627A1 (en) 2003-05-01
TNSN04072A1 (fr) 2006-06-01
US7098212B2 (en) 2006-08-29
ZA200402090B (en) 2005-05-23
HRP20040289A2 (en) 2004-10-31
PL370548A1 (en) 2005-05-30
NO20041631L (no) 2004-05-26
DE60235249D1 (de) 2010-03-18

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