SK120895A3 - Pyridine derivatives, process for preparing the same and intermediate products in this process and pharmaceutical compositions containing them - Google Patents

Pyridine derivatives, process for preparing the same and intermediate products in this process and pharmaceutical compositions containing them Download PDF

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Publication number
SK120895A3
SK120895A3 SK1208-95A SK120895A SK120895A3 SK 120895 A3 SK120895 A3 SK 120895A3 SK 120895 A SK120895 A SK 120895A SK 120895 A3 SK120895 A3 SK 120895A3
Authority
SK
Slovakia
Prior art keywords
group
carbon atoms
formula
alkylene
pyridyl
Prior art date
Application number
SK1208-95A
Other languages
English (en)
Slovak (sk)
Inventor
Michael G Wayne
Michael J Smithers
John W Rayner
Alan W Faull
Robert J Pearce
Andrew G Brewster
Richard E Shute
Stuart D Mills
Peter W R Caulkett
Original Assignee
Zeneca Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GB939306453A external-priority patent/GB9306453D0/en
Priority claimed from GB939325605A external-priority patent/GB9325605D0/en
Application filed by Zeneca Ltd filed Critical Zeneca Ltd
Publication of SK120895A3 publication Critical patent/SK120895A3/sk

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/72—Nitrogen atoms
    • C07D213/74—Amino or imino radicals substituted by hydrocarbon or substituted hydrocarbon radicals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Electroluminescent Light Sources (AREA)
  • Emulsifying, Dispersing, Foam-Producing Or Wetting Agents (AREA)
  • Electrochromic Elements, Electrophoresis, Or Variable Reflection Or Absorption Elements (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Peptides Or Proteins (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Pyrrole Compounds (AREA)
  • Pyridine Compounds (AREA)
SK1208-95A 1993-03-29 1994-03-28 Pyridine derivatives, process for preparing the same and intermediate products in this process and pharmaceutical compositions containing them SK120895A3 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GB939306453A GB9306453D0 (en) 1993-03-29 1993-03-29 Heterocyclic derivatives
GB939325605A GB9325605D0 (en) 1993-12-15 1993-12-15 Heterocyclic derivatives
PCT/GB1994/000647 WO1994022834A1 (en) 1993-03-29 1994-03-28 Heterocyclic derivatives as platelet aggregation inhibitors

Publications (1)

Publication Number Publication Date
SK120895A3 true SK120895A3 (en) 1996-06-05

Family

ID=26302668

Family Applications (1)

Application Number Title Priority Date Filing Date
SK1208-95A SK120895A3 (en) 1993-03-29 1994-03-28 Pyridine derivatives, process for preparing the same and intermediate products in this process and pharmaceutical compositions containing them

Country Status (26)

Country Link
US (1) US5556977A (xx)
EP (2) EP0825184B1 (xx)
JP (1) JPH08508291A (xx)
KR (1) KR100231089B1 (xx)
CN (1) CN1120334A (xx)
AT (2) ATE202345T1 (xx)
AU (1) AU692438B2 (xx)
BR (1) BR9406613A (xx)
CA (1) CA2156070A1 (xx)
CZ (1) CZ250995A3 (xx)
DE (2) DE69427548T2 (xx)
DK (2) DK0825184T3 (xx)
ES (2) ES2159798T3 (xx)
FI (1) FI954616A0 (xx)
GB (1) GB9406143D0 (xx)
GR (2) GR3027751T3 (xx)
HU (2) HUT72088A (xx)
IL (1) IL109144A (xx)
NO (1) NO305244B1 (xx)
NZ (1) NZ262941A (xx)
PL (1) PL310889A1 (xx)
PT (1) PT825184E (xx)
SK (1) SK120895A3 (xx)
TW (1) TW276254B (xx)
WO (1) WO1994022834A1 (xx)
ZW (1) ZW4294A1 (xx)

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US6221902B1 (en) 1998-05-12 2001-04-24 American Home Products Corporation Biphenyl sulfonyl aryl carboxylic acids useful in the treatment of insulin resistance and hyperglycemia
US6451827B2 (en) 1998-05-12 2002-09-17 Wyeth 2,3,5-substituted biphenyls useful in the treatment of insulin resistance and hyperglycemia
WO2000006158A1 (en) * 1998-07-31 2000-02-10 Eli Lilly And Company Heterocyclyl sulphonamide derivatives
GB9902989D0 (en) 1999-02-11 1999-03-31 Zeneca Ltd Heterocyclic derivatives
JP2002542224A (ja) * 1999-04-19 2002-12-10 コーエラカント コーポレイション Ｉｉ型糖尿病の治療薬としてのｐｐａｒ−（ガンマ）作用物質
US6310081B1 (en) 1999-05-10 2001-10-30 American Home Products Corporation Biphenyl sulfonyl aryl carboxylic acids useful in the treatment of insulin resistance and hyperglycemia
EP1330444B1 (en) 2000-11-01 2011-03-23 Millennium Pharmaceuticals, Inc. Nitrogenous heterocyclic compounds and process for making them
DE202011000090U1 (de) 2011-01-14 2011-04-21 E-LEAD ELECTRONIC CO., LTD., Shengang Shiang Fahrzeug-Audiosystem mit auswechselbarem Plug-In-Computer
JP7065951B2 (ja) 2017-09-22 2022-05-12 ジュビラント エピパッド エルエルシー Ｐａｄ阻害剤としての複素環式化合物
MX2020003341A (es) 2017-10-18 2020-09-17 Jubilant Epipad LLC Compuestos de imidazo-piridina como inhibidores de pad.
CN111386265A (zh) 2017-11-06 2020-07-07 朱比连特普罗德尔有限责任公司 作为pd1/pd-l1活化的抑制剂的嘧啶衍生物
WO2019102494A1 (en) 2017-11-24 2019-05-31 Jubilant Biosys Limited Heterocyclic compounds as prmt5 inhibitors
MX2020009517A (es) 2018-03-13 2021-01-20 Jubilant Prodel LLC Compuestos biciclicos como inhibidores de la interaccion/activacio n de pdl/pd-l1.

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Also Published As

Publication number Publication date
BR9406613A (pt) 1996-02-06
EP0691959A1 (en) 1996-01-17
ZW4294A1 (en) 1994-12-21
NO305244B1 (no) 1999-04-26
CZ250995A3 (en) 1996-01-17
DE69427548T2 (de) 2002-04-18
NO953837D0 (no) 1995-09-28
DK0825184T3 (da) 2001-09-10
PL310889A1 (en) 1996-01-08
ES2159798T3 (es) 2001-10-16
DE69427548D1 (de) 2001-07-26
EP0825184A1 (en) 1998-02-25
IL109144A (en) 2000-02-29
EP0825184B1 (en) 2001-06-20
DK0691959T3 (da) 1999-04-26
CN1120334A (zh) 1996-04-10
HUT72088A (en) 1996-03-28
GB9406143D0 (en) 1994-05-18
NO953837L (no) 1995-09-28
CA2156070A1 (en) 1994-10-13
DE69411900D1 (de) 1998-08-27
ATE168678T1 (de) 1998-08-15
KR100231089B1 (ko) 1999-11-15
AU6288994A (en) 1994-10-24
IL109144A0 (en) 1994-06-24
ES2119184T3 (es) 1998-10-01
DE69411900T2 (de) 1998-12-10
FI954616A (fi) 1995-09-28
US5556977A (en) 1996-09-17
JPH08508291A (ja) 1996-09-03
PT825184E (pt) 2001-11-30
TW276254B (xx) 1996-05-21
EP0691959B1 (en) 1998-07-22
GR3036640T3 (en) 2001-12-31
GR3027751T3 (en) 1998-11-30
HU211336A9 (en) 1995-11-28
AU692438B2 (en) 1998-06-11
FI954616A0 (fi) 1995-09-28
NZ262941A (en) 1997-07-27
ATE202345T1 (de) 2001-07-15
WO1994022834A1 (en) 1994-10-13
HU9502290D0 (en) 1995-10-30

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