FI954616A - Heterosyklisiä johdannaisia verihiutaleiden kasaantumisen inhibiittoreina - Google Patents

Heterosyklisiä johdannaisia verihiutaleiden kasaantumisen inhibiittoreina Download PDF

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Publication number
FI954616A
FI954616A FI954616A FI954616A FI954616A FI 954616 A FI954616 A FI 954616A FI 954616 A FI954616 A FI 954616A FI 954616 A FI954616 A FI 954616A FI 954616 A FI954616 A FI 954616A
Authority
FI
Finland
Prior art keywords
inhibitors
platelet aggregation
heterocyclic derivatives
ylüphenoxybutyric
piperazin
Prior art date
Application number
FI954616A
Other languages
English (en)
Swedish (sv)
Other versions
FI954616A0 (fi
Inventor
Michael Garth Wayne
Michael James Smithers
John Wall Rayner
Alan Wellington Faull
Robert James Pearce
Andrew George Brewster
Richard Eden Shute
Stuart Dennett Mills
Peter William Rodney Caulkett
Original Assignee
Zeneca Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GB939306453A external-priority patent/GB9306453D0/en
Priority claimed from GB939325605A external-priority patent/GB9325605D0/en
Application filed by Zeneca Ltd filed Critical Zeneca Ltd
Publication of FI954616A publication Critical patent/FI954616A/fi
Publication of FI954616A0 publication Critical patent/FI954616A0/fi

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/72—Nitrogen atoms
    • C07D213/74—Amino or imino radicals substituted by hydrocarbon or substituted hydrocarbon radicals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Electrochromic Elements, Electrophoresis, Or Variable Reflection Or Absorption Elements (AREA)
  • Electroluminescent Light Sources (AREA)
  • Emulsifying, Dispersing, Foam-Producing Or Wetting Agents (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pyrrole Compounds (AREA)
  • Peptides Or Proteins (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Pyridine Compounds (AREA)
FI954616A 1993-03-29 1995-09-28 Heterosyklisiä johdannaisia verihiutaleiden kasaantumisen inhibiittoreina FI954616A0 (fi)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GB939306453A GB9306453D0 (en) 1993-03-29 1993-03-29 Heterocyclic derivatives
GB939325605A GB9325605D0 (en) 1993-12-15 1993-12-15 Heterocyclic derivatives
PCT/GB1994/000647 WO1994022834A1 (en) 1993-03-29 1994-03-28 Heterocyclic derivatives as platelet aggregation inhibitors

Publications (2)

Publication Number Publication Date
FI954616A true FI954616A (fi) 1995-09-28
FI954616A0 FI954616A0 (fi) 1995-09-28

Family

ID=26302668

Family Applications (1)

Application Number Title Priority Date Filing Date
FI954616A FI954616A0 (fi) 1993-03-29 1995-09-28 Heterosyklisiä johdannaisia verihiutaleiden kasaantumisen inhibiittoreina

Country Status (26)

Country Link
US (1) US5556977A (fi)
EP (2) EP0825184B1 (fi)
JP (1) JPH08508291A (fi)
KR (1) KR100231089B1 (fi)
CN (1) CN1120334A (fi)
AT (2) ATE202345T1 (fi)
AU (1) AU692438B2 (fi)
BR (1) BR9406613A (fi)
CA (1) CA2156070A1 (fi)
CZ (1) CZ250995A3 (fi)
DE (2) DE69411900T2 (fi)
DK (2) DK0691959T3 (fi)
ES (2) ES2119184T3 (fi)
FI (1) FI954616A0 (fi)
GB (1) GB9406143D0 (fi)
GR (2) GR3027751T3 (fi)
HU (2) HUT72088A (fi)
IL (1) IL109144A (fi)
NO (1) NO305244B1 (fi)
NZ (1) NZ262941A (fi)
PL (1) PL310889A1 (fi)
PT (1) PT825184E (fi)
SK (1) SK120895A3 (fi)
TW (1) TW276254B (fi)
WO (1) WO1994022834A1 (fi)
ZW (1) ZW4294A1 (fi)

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DE202011000090U1 (de) 2011-01-14 2011-04-21 E-LEAD ELECTRONIC CO., LTD., Shengang Shiang Fahrzeug-Audiosystem mit auswechselbarem Plug-In-Computer
WO2019058393A1 (en) 2017-09-22 2019-03-28 Jubilant Biosys Limited HETEROCYCLIC COMPOUNDS AS INHIBITORS OF PAD
SG11202003463XA (en) 2017-10-18 2020-05-28 Jubilant Epipad LLC Imidazo-pyridine compounds as pad inhibitors
CN111386265A (zh) 2017-11-06 2020-07-07 朱比连特普罗德尔有限责任公司 作为pd1/pd-l1活化的抑制剂的嘧啶衍生物
MX2020005363A (es) 2017-11-24 2020-10-01 Jubilant Episcribe Llc Compuestos heterociclicos como inhibidores de prmt5.
EP3765453A1 (en) 2018-03-13 2021-01-20 Jubilant Prodel LLC Bicyclic compounds as inhibitors of pd1/pd-l1 interaction/activation

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Also Published As

Publication number Publication date
GR3027751T3 (en) 1998-11-30
KR100231089B1 (ko) 1999-11-15
ES2119184T3 (es) 1998-10-01
GB9406143D0 (en) 1994-05-18
EP0825184A1 (en) 1998-02-25
DE69427548D1 (de) 2001-07-26
HU9502290D0 (en) 1995-10-30
TW276254B (fi) 1996-05-21
EP0691959B1 (en) 1998-07-22
CA2156070A1 (en) 1994-10-13
GR3036640T3 (en) 2001-12-31
EP0691959A1 (en) 1996-01-17
DE69411900D1 (de) 1998-08-27
HUT72088A (en) 1996-03-28
IL109144A (en) 2000-02-29
CN1120334A (zh) 1996-04-10
DK0691959T3 (da) 1999-04-26
HU211336A9 (en) 1995-11-28
BR9406613A (pt) 1996-02-06
DK0825184T3 (da) 2001-09-10
IL109144A0 (en) 1994-06-24
US5556977A (en) 1996-09-17
ES2159798T3 (es) 2001-10-16
NO305244B1 (no) 1999-04-26
CZ250995A3 (en) 1996-01-17
PT825184E (pt) 2001-11-30
NO953837D0 (no) 1995-09-28
DE69411900T2 (de) 1998-12-10
NZ262941A (en) 1997-07-27
JPH08508291A (ja) 1996-09-03
ATE202345T1 (de) 2001-07-15
DE69427548T2 (de) 2002-04-18
ZW4294A1 (en) 1994-12-21
ATE168678T1 (de) 1998-08-15
EP0825184B1 (en) 2001-06-20
FI954616A0 (fi) 1995-09-28
NO953837L (no) 1995-09-28
AU6288994A (en) 1994-10-24
SK120895A3 (en) 1996-06-05
PL310889A1 (en) 1996-01-08
AU692438B2 (en) 1998-06-11
WO1994022834A1 (en) 1994-10-13

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