SI3030563T1 - Derivati pirolo (3,2-d) pirimidina za zdravljenje virusnih okužb in drugih bolezni - Google Patents

Derivati pirolo (3,2-d) pirimidina za zdravljenje virusnih okužb in drugih bolezni

Info

Publication number
SI3030563T1
SI3030563T1 SI201430476T SI201430476T SI3030563T1 SI 3030563 T1 SI3030563 T1 SI 3030563T1 SI 201430476 T SI201430476 T SI 201430476T SI 201430476 T SI201430476 T SI 201430476T SI 3030563 T1 SI3030563 T1 SI 3030563T1
Authority
SI
Slovenia
Prior art keywords
pyrrolo
diseases
treatment
viral infections
pyrimidine derivatives
Prior art date
Application number
SI201430476T
Other languages
English (en)
Inventor
Gowan David Craig Mc
Serge Maria Aloysius Pieters
Stefaan Julien Last
Werner EMBRECHTS
Tim Hugo Maria Jonckers
Pierre Jean-Marie Bernard Raboisson
Original Assignee
Janssen Sciences Ireland Uc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Janssen Sciences Ireland Uc filed Critical Janssen Sciences Ireland Uc
Publication of SI3030563T1 publication Critical patent/SI3030563T1/sl

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/14—Antivirals for RNA viruses
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Oncology (AREA)
  • Virology (AREA)
  • Communicable Diseases (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Molecular Biology (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
SI201430476T 2013-06-27 2014-06-26 Derivati pirolo (3,2-d) pirimidina za zdravljenje virusnih okužb in drugih bolezni SI3030563T1 (sl)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP13174108 2013-06-27
EP14738751.8A EP3030563B1 (en) 2013-06-27 2014-06-26 Pyrrolo [3,2-d] pyrimidine derivatives for the treatment of viral infections and other diseases
PCT/EP2014/063467 WO2014207082A1 (en) 2013-06-27 2014-06-26 Pyrrolo[3,2-d]pyrimidine derivatives for the treatment of viral infections and other diseases

Publications (1)

Publication Number Publication Date
SI3030563T1 true SI3030563T1 (sl) 2017-12-29

Family

ID=48692351

Family Applications (1)

Application Number Title Priority Date Filing Date
SI201430476T SI3030563T1 (sl) 2013-06-27 2014-06-26 Derivati pirolo (3,2-d) pirimidina za zdravljenje virusnih okužb in drugih bolezni

Country Status (26)

Country Link
US (2) US10385054B2 (sl)
EP (1) EP3030563B1 (sl)
JP (2) JP6763769B2 (sl)
KR (1) KR102311234B1 (sl)
CN (2) CN105473592B (sl)
AU (2) AU2014301089B2 (sl)
BR (1) BR112015032546B1 (sl)
CA (1) CA2913028C (sl)
CL (1) CL2015003686A1 (sl)
DK (1) DK3030563T3 (sl)
EA (2) EA202090258A3 (sl)
ES (1) ES2645950T3 (sl)
HK (1) HK1218116A1 (sl)
HR (1) HRP20171720T1 (sl)
HU (1) HUE037125T2 (sl)
IL (3) IL242655B (sl)
MX (1) MX361527B (sl)
MY (1) MY176142A (sl)
NO (1) NO3030563T3 (sl)
PH (1) PH12015502780A1 (sl)
PL (1) PL3030563T3 (sl)
PT (1) PT3030563T (sl)
SG (2) SG11201510637UA (sl)
SI (1) SI3030563T1 (sl)
UA (1) UA117590C2 (sl)
WO (1) WO2014207082A1 (sl)

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KR20220132594A (ko) 2020-01-27 2022-09-30 브리스톨-마이어스 스큅 컴퍼니 톨-유사 수용체 7 (TLR7) 효능제로서의 1H-피라졸로[4,3-d]피리미딘 화합물
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