SG11201510637UA - Pyrrolo[3,2-d]pyrimidine derivatives for the treatment of viral infections and other diseases - Google Patents
Pyrrolo[3,2-d]pyrimidine derivatives for the treatment of viral infections and other diseasesInfo
- Publication number
- SG11201510637UA SG11201510637UA SG11201510637UA SG11201510637UA SG11201510637UA SG 11201510637U A SG11201510637U A SG 11201510637UA SG 11201510637U A SG11201510637U A SG 11201510637UA SG 11201510637U A SG11201510637U A SG 11201510637UA SG 11201510637U A SG11201510637U A SG 11201510637UA
- Authority
- SG
- Singapore
- Prior art keywords
- pyrrolo
- diseases
- treatment
- viral infections
- pyrimidine derivatives
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A61P31/14—Antivirals for RNA viruses
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Pharmacology & Pharmacy (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Oncology (AREA)
- Virology (AREA)
- Communicable Diseases (AREA)
- Molecular Biology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP13174108 | 2013-06-27 | ||
| PCT/EP2014/063467 WO2014207082A1 (en) | 2013-06-27 | 2014-06-26 | Pyrrolo[3,2-d]pyrimidine derivatives for the treatment of viral infections and other diseases |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| SG11201510637UA true SG11201510637UA (en) | 2016-01-28 |
Family
ID=48692351
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| SG11201510637UA SG11201510637UA (en) | 2013-06-27 | 2014-06-26 | Pyrrolo[3,2-d]pyrimidine derivatives for the treatment of viral infections and other diseases |
| SG10201803331PA SG10201803331PA (en) | 2013-06-27 | 2014-06-26 | Pyrrolo[3,2-d]pyrimidine derivatives for the treatment of viral infections and other diseases |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| SG10201803331PA SG10201803331PA (en) | 2013-06-27 | 2014-06-26 | Pyrrolo[3,2-d]pyrimidine derivatives for the treatment of viral infections and other diseases |
Country Status (26)
| Country | Link |
|---|---|
| US (2) | US10385054B2 (en) |
| EP (1) | EP3030563B1 (en) |
| JP (2) | JP6763769B2 (en) |
| KR (1) | KR102311234B1 (en) |
| CN (2) | CN105473592B (en) |
| AU (2) | AU2014301089B2 (en) |
| BR (1) | BR112015032546B1 (en) |
| CA (1) | CA2913028C (en) |
| CL (1) | CL2015003686A1 (en) |
| DK (1) | DK3030563T3 (en) |
| EA (2) | EA202090258A3 (en) |
| ES (1) | ES2645950T3 (en) |
| HK (1) | HK1218116A1 (en) |
| HR (1) | HRP20171720T1 (en) |
| HU (1) | HUE037125T2 (en) |
| IL (3) | IL242655B (en) |
| MX (1) | MX361527B (en) |
| MY (1) | MY176142A (en) |
| NO (1) | NO3030563T3 (en) |
| PH (1) | PH12015502780B1 (en) |
| PL (1) | PL3030563T3 (en) |
| PT (1) | PT3030563T (en) |
| SG (2) | SG11201510637UA (en) |
| SI (1) | SI3030563T1 (en) |
| UA (1) | UA117590C2 (en) |
| WO (1) | WO2014207082A1 (en) |
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| JOP20150177B1 (en) | 2014-08-01 | 2021-08-17 | Janssen Pharmaceutica Nv | 6,7-DIHYDROPYRAZOLO[1,5-a]PYRAZIN-4(5H)-ONE COMPOUNDS AND THEIR USE AS NEGATIVE ALLOSTERIC MODULATORS OF MGLUR2 RECEPTORS |
| MA44334A (en) | 2015-10-29 | 2018-09-05 | Novartis Ag | ANTIBODY CONJUGATES INCLUDING A TOLL-TYPE RECEPTOR AGONIST |
| US11045562B2 (en) | 2015-12-18 | 2021-06-29 | Janssen Pharmaceutica Nv | Radiolabelled mGluR2/3 PET ligands |
| SI3389727T1 (en) | 2015-12-18 | 2020-10-30 | Janssen Pharmaceutica Nv | Radiolabelled mglur2/3 pet ligands |
| KR102450287B1 (en) | 2016-09-29 | 2022-09-30 | 얀센 사이언시즈 아일랜드 언리미티드 컴퍼니 | Pyrimidine prodrugs for treatment of viral infections and additional diseases |
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| MX2021009496A (en) | 2019-02-08 | 2021-09-08 | Progeneer Inc | Toll-like receptor 7 or 8 agonist-cholesterol complex, and use of same. |
| JP2023512229A (en) | 2020-01-27 | 2023-03-24 | ブリストル－マイヤーズ スクイブ カンパニー | 1H-pyrazolo[4,3-d]pyrimidine compounds as Toll-like receptor 7 (TLR7) agonists |
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| JP2023512206A (en) | 2020-01-27 | 2023-03-24 | ブリストル－マイヤーズ スクイブ カンパニー | 1H-pyrazolo[4,3-d]pyrimidine compounds as Toll-like receptor 7 (TLR7) agonists |
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| BR112015007366A2 (en) | 2012-10-05 | 2017-07-04 | Janssen Sciences Ireland Uc | acylaminopyrimidine derivatives for the treatment of viral infections and other diseases |
| JP6293765B2 (en) | 2012-10-10 | 2018-03-14 | ヤンセン・サイエンシズ・アイルランド・ユーシー | Pyrrolo [3,2-D] pyrimidine derivatives for the treatment of viral infections and other diseases |
| BR112015011036B1 (en) | 2012-11-16 | 2022-02-01 | Janssen Sciences Ireland Uc | Heterocyclic Substituted 2-Amino-quinazoline Derivatives, Pharmaceutical Composition |
| EA035174B1 (en) | 2013-02-21 | 2020-05-12 | Янссен Сайенсиз Айрлэнд Юси | 2-aminopyrimidine derivatives as modulators of toll-like receptors tlr7 and/or tlr8 |
| SG11201508078XA (en) | 2013-03-29 | 2015-11-27 | Janssen Sciences Ireland Uc | Macrocyclic deaza-purinones for the treatment of viral infections |
| ES2645950T3 (en) * | 2013-06-27 | 2017-12-11 | Janssen Sciences Ireland Uc | Pyrrolo [3,2-d] pyrimidine derivatives for the treatment of viral infections and other diseases |
| JP6401788B2 (en) | 2013-07-30 | 2018-10-10 | ヤンセン・サイエンシズ・アイルランド・ユーシー | Thieno [3,2-d] pyrimidine derivatives for viral infection treatment |
| US9701661B2 (en) | 2014-07-11 | 2017-07-11 | Northwestern University | 2-imidazolyl-pyrimidine scaffolds as potent and selective inhibitors of neuronal nitric oxide synthase |
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