SI0788509T1 - Therapeutic peptide derivatives - Google Patents

Therapeutic peptide derivatives

Info

Publication number
SI0788509T1
SI0788509T1 SI9430451T SI9430451T SI0788509T1 SI 0788509 T1 SI0788509 T1 SI 0788509T1 SI 9430451 T SI9430451 T SI 9430451T SI 9430451 T SI9430451 T SI 9430451T SI 0788509 T1 SI0788509 T1 SI 0788509T1
Authority
SI
Slovenia
Prior art keywords
peptide derivatives
therapeutic peptide
peptide
amino
amide
Prior art date
Application number
SI9430451T
Other languages
English (en)
Slovenian (sl)
Inventor
Sun Hyuk Kim
Zhengxin Dong
John E. Taylor
Sylviane Moreau
Susan Riley Apartment 3 KEYES
Original Assignee
Societe De Conseils De Recherches
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Societe De Conseils De Recherches filed Critical Societe De Conseils De Recherches
Publication of SI0788509T1 publication Critical patent/SI0788509T1/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K7/00Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K7/04Linear peptides containing only normal peptide links
    • C07K7/08Linear peptides containing only normal peptide links having 12 to 20 amino acids
    • C07K7/086Bombesin; Related peptides
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/12Antidiarrhoeals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/18Drugs for disorders of the alimentary tract or the digestive system for pancreatic disorders, e.g. pancreatic enzymes
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00Drugs for disorders of the senses
    • A61P27/02Ophthalmic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/14Antivirals for RNA viruses
    • A61P31/18Antivirals for RNA viruses for HIV
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/02Immunomodulators
    • A61P37/04Immunostimulants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00Drugs for disorders of the endocrine system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00Drugs for disorders of the endocrine system
    • A61P5/02Drugs for disorders of the endocrine system of the hypothalamic hormones, e.g. TRH, GnRH, CRH, GRH, somatostatin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00Drugs for disorders of the endocrine system
    • A61P5/02Drugs for disorders of the endocrine system of the hypothalamic hormones, e.g. TRH, GnRH, CRH, GRH, somatostatin
    • A61P5/04Drugs for disorders of the endocrine system of the hypothalamic hormones, e.g. TRH, GnRH, CRH, GRH, somatostatin for decreasing, blocking or antagonising the activity of the hypothalamic hormones
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00Drugs for disorders of the endocrine system
    • A61P5/06Drugs for disorders of the endocrine system of the anterior pituitary hormones, e.g. TSH, ACTH, FSH, LH, PRL, GH
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00Drugs for disorders of the endocrine system
    • A61P5/06Drugs for disorders of the endocrine system of the anterior pituitary hormones, e.g. TSH, ACTH, FSH, LH, PRL, GH
    • A61P5/08Drugs for disorders of the endocrine system of the anterior pituitary hormones, e.g. TSH, ACTH, FSH, LH, PRL, GH for decreasing, blocking or antagonising the activity of the anterior pituitary hormones
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00Drugs for disorders of the endocrine system
    • A61P5/14Drugs for disorders of the endocrine system of the thyroid hormones, e.g. T3, T4
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00Drugs for disorders of the endocrine system
    • A61P5/18Drugs for disorders of the endocrine system of the parathyroid hormones
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00Drugs for disorders of the endocrine system
    • A61P5/38Drugs for disorders of the endocrine system of the suprarenal hormones
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00Drugs for disorders of the endocrine system
    • A61P5/48Drugs for disorders of the endocrine system of the pancreatic hormones
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00Drugs for disorders of the blood or the extracellular fluid
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K14/00Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • C07K14/435Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • C07K14/575Hormones
    • C07K14/655Somatostatins
    • C07K14/6555Somatostatins at least 1 amino acid in D-form
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Diabetes (AREA)
  • Endocrinology (AREA)
  • Molecular Biology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Genetics & Genomics (AREA)
  • Biophysics (AREA)
  • Biochemistry (AREA)
  • Immunology (AREA)
  • Hematology (AREA)
  • Virology (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Zoology (AREA)
  • Toxicology (AREA)
  • Biomedical Technology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Oncology (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Obesity (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Communicable Diseases (AREA)
  • Cardiology (AREA)
  • Vascular Medicine (AREA)
SI9430451T 1993-08-09 1994-08-08 Therapeutic peptide derivatives SI0788509T1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US10419493A 1993-08-09 1993-08-09
PCT/US1994/008875 WO1995004752A1 (en) 1993-08-09 1994-08-08 Therapeutic peptide derivatives

Publications (1)

Publication Number Publication Date
SI0788509T1 true SI0788509T1 (en) 2003-10-31

Family

ID=22299154

Family Applications (2)

Application Number Title Priority Date Filing Date
SI9430451T SI0788509T1 (en) 1993-08-09 1994-08-08 Therapeutic peptide derivatives
SI9420051A SI9420051A (en) 1993-08-09 1994-08-08 Chemical modified peptide derivatives, process for their preparation and their use in human therapy

Family Applications After (1)

Application Number Title Priority Date Filing Date
SI9420051A SI9420051A (en) 1993-08-09 1994-08-08 Chemical modified peptide derivatives, process for their preparation and their use in human therapy

Country Status (30)

Country Link
US (1) US5552520A (fi)
EP (3) EP1288223B1 (fi)
JP (3) JP3618750B2 (fi)
KR (1) KR100325972B1 (fi)
CN (1) CN1055700C (fi)
AT (3) ATE284413T1 (fi)
AU (1) AU689490B2 (fi)
CA (1) CA2168113C (fi)
CZ (3) CZ292586B6 (fi)
DE (3) DE69434181T2 (fi)
DK (3) DK1288224T3 (fi)
ES (3) ES2229045T3 (fi)
FI (1) FI960584A0 (fi)
GE (1) GEP20002146B (fi)
HK (2) HK1053313A1 (fi)
HU (1) HU224350B1 (fi)
LT (1) LT4078B (fi)
LV (1) LV11549B (fi)
MD (1) MD1591B2 (fi)
NZ (1) NZ271238A (fi)
PL (1) PL180612B1 (fi)
PT (2) PT788509E (fi)
RO (1) RO117259B1 (fi)
RU (1) RU2133252C1 (fi)
SG (1) SG75092A1 (fi)
SI (2) SI0788509T1 (fi)
SK (1) SK15096A3 (fi)
UA (1) UA44707C2 (fi)
WO (1) WO1995004752A1 (fi)
ZA (1) ZA945966B (fi)

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Also Published As

Publication number Publication date
ES2196031T3 (es) 2003-12-16
HK1053313A1 (en) 2003-10-17
EP1288223B1 (en) 2004-12-08
DE69434181D1 (de) 2005-01-13
CZ39096A3 (en) 1996-11-13
EP0788509A1 (en) 1997-08-13
EP0788509B1 (en) 2003-05-28
JP3618750B2 (ja) 2005-02-09
ATE399177T1 (de) 2008-07-15
LV11549B (en) 1997-04-20
PT788509E (pt) 2003-10-31
DE69435105D1 (de) 2008-08-07
EP1288224A1 (en) 2003-03-05
ES2229045T3 (es) 2005-04-16
DK1288223T3 (da) 2005-03-29
RO117259B1 (ro) 2001-12-28
CA2168113A1 (en) 1995-02-16
UA44707C2 (uk) 2002-03-15
MD960137A (en) 1999-01-31
KR100325972B1 (ko) 2002-07-27
HU9600281D0 (en) 1996-04-29
GEP20002146B (en) 2000-06-25
US5552520A (en) 1996-09-03
DE69432758T2 (de) 2004-02-19
ATE241643T1 (de) 2003-06-15
CZ289590B6 (cs) 2002-02-13
DE69432758D1 (en) 2003-07-03
ATE284413T1 (de) 2004-12-15
HU224350B1 (hu) 2005-08-29
JP2004339237A (ja) 2004-12-02
SK15096A3 (en) 1996-07-03
SI9420051A (en) 1996-12-31
LV11549A (lv) 1996-10-20
LT4078B (en) 1996-12-27
FI960584A (fi) 1996-02-08
AU7481994A (en) 1995-02-28
PL180612B1 (pl) 2001-03-30
CZ292586B6 (cs) 2003-10-15
PL312989A1 (en) 1996-05-27
CZ289552B6 (cs) 2002-02-13
EP1288223A1 (en) 2003-03-05
HUT73491A (en) 1996-08-28
CN1055700C (zh) 2000-08-23
LT96025A (en) 1996-07-25
WO1995004752A1 (en) 1995-02-16
DK1288224T3 (da) 2008-10-13
JPH09501177A (ja) 1997-02-04
RU2133252C1 (ru) 1999-07-20
CN1133047A (zh) 1996-10-09
JP2005015488A (ja) 2005-01-20
ZA945966B (en) 1995-06-26
CA2168113C (en) 2002-10-01
AU689490B2 (en) 1998-04-02
JP3869439B2 (ja) 2007-01-17
FI960584A0 (fi) 1996-02-08
DK0788509T3 (da) 2003-06-23
PT1288223E (pt) 2005-03-31
ES2309131T3 (es) 2008-12-16
EP0788509A4 (en) 1999-07-14
SG75092A1 (en) 2000-09-19
EP1288224B1 (en) 2008-06-25
DE69434181T2 (de) 2005-12-01
NZ271238A (en) 1997-10-24
HK1053314A1 (en) 2003-10-17
MD1591B2 (ro) 2001-01-31
JP3785179B2 (ja) 2006-06-14

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