SG162722A1 - N,n-substituted 3-aminopyrrolidine compounds useful as monoamines reuptake inhibitors - Google Patents
N,n-substituted 3-aminopyrrolidine compounds useful as monoamines reuptake inhibitorsInfo
- Publication number
- SG162722A1 SG162722A1 SG201003432-0A SG2010034320A SG162722A1 SG 162722 A1 SG162722 A1 SG 162722A1 SG 2010034320 A SG2010034320 A SG 2010034320A SG 162722 A1 SG162722 A1 SG 162722A1
- Authority
- SG
- Singapore
- Prior art keywords
- substituted
- compounds useful
- reuptake inhibitors
- salt
- halogen atoms
- Prior art date
Links
- 239000003112 inhibitor Substances 0.000 title 1
- NGXSWUFDCSEIOO-UHFFFAOYSA-N pyrrolidin-3-amine Chemical class NC1CCNC1 NGXSWUFDCSEIOO-UHFFFAOYSA-N 0.000 title 1
- RWRDLPDLKQPQOW-UHFFFAOYSA-N tetrahydropyrrole Natural products C1CCNC1 RWRDLPDLKQPQOW-UHFFFAOYSA-N 0.000 abstract 4
- 125000005843 halogen group Chemical group 0.000 abstract 2
- 125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 abstract 2
- 125000004076 pyridyl group Chemical group 0.000 abstract 2
- -1 pyrrolidine compound Chemical class 0.000 abstract 2
- 150000003839 salts Chemical class 0.000 abstract 2
- 230000001225 therapeutic effect Effects 0.000 abstract 2
- 125000000217 alkyl group Chemical group 0.000 abstract 1
- 230000001747 exhibiting effect Effects 0.000 abstract 1
- 239000000825 pharmaceutical preparation Substances 0.000 abstract 1
- 238000001228 spectrum Methods 0.000 abstract 1
- 125000001424 substituent group Chemical group 0.000 abstract 1
Classifications
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- C07D205/02—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings
- C07D205/04—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
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- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
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- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Biomedical Technology (AREA)
- Diabetes (AREA)
- Addiction (AREA)
- Psychiatry (AREA)
- Endocrinology (AREA)
- Pain & Pain Management (AREA)
- Reproductive Health (AREA)
- Hematology (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Gynecology & Obstetrics (AREA)
- Obesity (AREA)
- Psychology (AREA)
- Emergency Medicine (AREA)
- Child & Adolescent Psychology (AREA)
- Pregnancy & Childbirth (AREA)
- Hospice & Palliative Care (AREA)
- Dermatology (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Physical Education & Sports Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP2005141230 | 2005-05-13 |
Publications (1)
Publication Number | Publication Date |
---|---|
SG162722A1 true SG162722A1 (en) | 2010-07-29 |
Family
ID=36693623
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
SG201003432-0A SG162722A1 (en) | 2005-05-13 | 2006-05-12 | N,n-substituted 3-aminopyrrolidine compounds useful as monoamines reuptake inhibitors |
Country Status (25)
Country | Link |
---|---|
US (6) | US8084442B2 (ru) |
EP (2) | EP2407451B1 (ru) |
JP (1) | JP4776631B2 (ru) |
KR (2) | KR20100038453A (ru) |
CN (3) | CN103613527B (ru) |
AR (1) | AR054191A1 (ru) |
AU (2) | AU2006244851B2 (ru) |
BR (1) | BRPI0610279A2 (ru) |
CA (1) | CA2608184C (ru) |
CY (1) | CY1114767T1 (ru) |
DK (1) | DK2407451T3 (ru) |
ES (2) | ES2451523T3 (ru) |
HK (1) | HK1193094A1 (ru) |
IL (1) | IL187311A (ru) |
IN (1) | IN2012DN00758A (ru) |
MX (1) | MX2007014252A (ru) |
MY (1) | MY148653A (ru) |
PL (1) | PL2407451T3 (ru) |
PT (1) | PT2407451E (ru) |
RU (1) | RU2414454C2 (ru) |
SG (1) | SG162722A1 (ru) |
SI (1) | SI2407451T1 (ru) |
TW (3) | TWI439452B (ru) |
WO (1) | WO2006121218A1 (ru) |
ZA (1) | ZA200709691B (ru) |
Families Citing this family (16)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EA010027B1 (ru) | 2002-11-27 | 2008-06-30 | Инсайт Корпорейшн | Производные 3-аминопирролидина в качестве модуляторов рецепторов хемокинов |
TWI439452B (zh) | 2005-05-13 | 2014-06-01 | Otsuka Pharma Co Ltd | 吡咯烷化合物(二) |
JP2009518313A (ja) * | 2005-11-30 | 2009-05-07 | スミスクライン・ビーチャム・コーポレイション | ピロリジンアニリン |
EP1960355A1 (en) * | 2005-11-30 | 2008-08-27 | F.Hoffmann-La Roche Ag | 3-amino-1-arylpropyl indoles and aza-substituted indoles |
JP5219465B2 (ja) * | 2006-11-10 | 2013-06-26 | 大塚製薬株式会社 | 医薬 |
CA2718736A1 (en) * | 2008-03-20 | 2009-09-24 | F. Hoffmann-La Roche Ag | Pyrrolidinyl derivatives and uses thereof |
US8987301B2 (en) | 2009-11-07 | 2015-03-24 | Merck Patent Gmbh | Heteroarylaminoquinolines as TGF-beta receptor kinase inhibitors |
EP2560953B1 (en) * | 2010-04-21 | 2016-01-06 | Probiodrug AG | Inhibitors of glutaminyl cyclase |
CN102766079B (zh) * | 2011-05-06 | 2015-04-08 | 上海医药工业研究院 | 一类吡咯烷衍生物、其制备方法及应用 |
US9353078B2 (en) | 2013-10-01 | 2016-05-31 | New York University | Amino, amido and heterocyclic compounds as modulators of rage activity and uses thereof |
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RU2698400C1 (ru) * | 2018-12-17 | 2019-08-26 | Георгий Сергеевич Немов | Способ лечения депрессии у собак и кошек |
CN113024517A (zh) * | 2019-12-09 | 2021-06-25 | 武汉九州钰民医药科技有限公司 | 一种制备厄达替尼的方法 |
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