SG10201609188WA - Compounds for treating spinal muscular atrophy - Google Patents

Compounds for treating spinal muscular atrophy

Info

Publication number
SG10201609188WA
SG10201609188WA SG10201609188WA SG10201609188WA SG10201609188WA SG 10201609188W A SG10201609188W A SG 10201609188WA SG 10201609188W A SG10201609188W A SG 10201609188WA SG 10201609188W A SG10201609188W A SG 10201609188WA SG 10201609188W A SG10201609188W A SG 10201609188WA
Authority
SG
Singapore
Prior art keywords
compounds
muscular atrophy
spinal muscular
treating spinal
treating
Prior art date
Application number
SG10201609188WA
Other languages
English (en)
Inventor
Hongyan Qi
Soongyu Choi
Amal Dakka
Gary Mitchell Karp
Jana Narasimhan
Nikolai Naryshkin
Anthony A Turpoff
Marla L Weetall
Ellen Welch
Matthew G Woll
Tianle Yang
Nanjing Zhang
Xiaoyan Zhang
Xin Zhao
Luke Green
Emmanuel Pinard
Hasane Ratni
Original Assignee
Ptc Therapeutics Inc
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=48948163&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=SG10201609188W(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Ptc Therapeutics Inc, Hoffmann La Roche filed Critical Ptc Therapeutics Inc
Publication of SG10201609188WA publication Critical patent/SG10201609188WA/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P21/00Drugs for disorders of the muscular or neuromuscular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D519/00Heterocyclic compounds containing more than one system of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring system not provided for in groups C07D453/00 or C07D455/00

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Neurology (AREA)
  • Epidemiology (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Psychiatry (AREA)
  • Hospice & Palliative Care (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Measuring Or Testing Involving Enzymes Or Micro-Organisms (AREA)
  • Steroid Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pyridine Compounds (AREA)
SG10201609188WA 2012-02-10 2013-02-08 Compounds for treating spinal muscular atrophy SG10201609188WA (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US201261597523P 2012-02-10 2012-02-10

Publications (1)

Publication Number Publication Date
SG10201609188WA true SG10201609188WA (en) 2016-12-29

Family

ID=48948163

Family Applications (2)

Application Number Title Priority Date Filing Date
SG11201404713PA SG11201404713PA (en) 2012-02-10 2013-02-08 Compounds for treating spinal muscular atrophy
SG10201609188WA SG10201609188WA (en) 2012-02-10 2013-02-08 Compounds for treating spinal muscular atrophy

Family Applications Before (1)

Application Number Title Priority Date Filing Date
SG11201404713PA SG11201404713PA (en) 2012-02-10 2013-02-08 Compounds for treating spinal muscular atrophy

Country Status (29)

Country Link
US (6) US9586955B2 (enExample)
EP (2) EP3406252B1 (enExample)
JP (2) JP6092897B2 (enExample)
KR (2) KR102341596B1 (enExample)
CN (3) CN119528903A (enExample)
AR (1) AR092794A1 (enExample)
AU (2) AU2013216870B2 (enExample)
BR (1) BR112014019750B1 (enExample)
CA (1) CA2863874C (enExample)
CL (1) CL2014002100A1 (enExample)
CO (1) CO7061082A2 (enExample)
CR (1) CR20140376A (enExample)
DK (1) DK2812004T3 (enExample)
EA (2) EA037123B1 (enExample)
EC (1) ECSP14017269A (enExample)
ES (1) ES2697174T3 (enExample)
HU (1) HUE039779T2 (enExample)
IL (2) IL233959A (enExample)
MA (1) MA35920B1 (enExample)
MX (2) MX354074B (enExample)
NZ (1) NZ628186A (enExample)
PE (1) PE20142364A1 (enExample)
PH (2) PH12018501711B1 (enExample)
PL (1) PL2812004T3 (enExample)
SG (2) SG11201404713PA (enExample)
TR (1) TR201813877T4 (enExample)
TW (2) TWI585085B (enExample)
UA (1) UA116981C2 (enExample)
WO (1) WO2013119916A2 (enExample)

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