RU2014136339A - Замещенные пролины/пиперидины как антагонисты орексиновых рецепторов - Google Patents

Замещенные пролины/пиперидины как антагонисты орексиновых рецепторов Download PDF

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RU2014136339A
RU2014136339A RU2014136339A RU2014136339A RU2014136339A RU 2014136339 A RU2014136339 A RU 2014136339A RU 2014136339 A RU2014136339 A RU 2014136339A RU 2014136339 A RU2014136339 A RU 2014136339A RU 2014136339 A RU2014136339 A RU 2014136339A
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alkyl
mono
independently
compound
substituted
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RU2014136339A
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Russian (ru)
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Теодор КАМЕНЕЦКА
Жун ЦЗЯН
Синьи СУН
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Иолас Терапьютикс, Инк.
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    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
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    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
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    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
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    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems

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RU2014136339A 2012-02-07 2013-02-06 Замещенные пролины/пиперидины как антагонисты орексиновых рецепторов RU2014136339A (ru)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201261596062P 2012-02-07 2012-02-07
US61/596,062 2012-02-07
PCT/US2013/024903 WO2013119639A1 (en) 2012-02-07 2013-02-06 Substituted prolines / piperidines as orexin receptor antagonists

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RU2014136339A true RU2014136339A (ru) 2016-03-27

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US (2) US9499517B2 (https=)
EP (1) EP2811997B1 (https=)
JP (1) JP6346862B2 (https=)
KR (1) KR20140124398A (https=)
CN (1) CN104220065A (https=)
AR (1) AR099466A1 (https=)
AU (1) AU2013217323A1 (https=)
BR (1) BR112014019426A8 (https=)
CA (1) CA2863413A1 (https=)
ES (1) ES2672732T3 (https=)
HK (1) HK1204955A1 (https=)
IL (1) IL234025A0 (https=)
MX (1) MX2014009281A (https=)
NZ (1) NZ628491A (https=)
PH (1) PH12014501784A1 (https=)
RU (1) RU2014136339A (https=)
SG (1) SG11201404738QA (https=)
WO (1) WO2013119639A1 (https=)

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