PT2102224E - FORMA CRISTALINA HEMI-HIDRATADA DE 1-(ß-DGLICOPIRANOSIL)- 4-METIL-3-[5-(4-FLUOROFENIL)-2- TIENILMETIL]BENZENO - Google Patents

FORMA CRISTALINA HEMI-HIDRATADA DE 1-(ß-DGLICOPIRANOSIL)- 4-METIL-3-[5-(4-FLUOROFENIL)-2- TIENILMETIL]BENZENO Download PDF

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Publication number
PT2102224E
PT2102224E PT78503067T PT07850306T PT2102224E PT 2102224 E PT2102224 E PT 2102224E PT 78503067 T PT78503067 T PT 78503067T PT 07850306 T PT07850306 T PT 07850306T PT 2102224 E PT2102224 E PT 2102224E
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Portugal
Prior art keywords
thienylmethyl
glucopyranosyl
fluorophenyl
methyl
crystalline form
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PT78503067T
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English (en)
Inventor
Sumihiro Nomura
Eiji Kawanishi
Original Assignee
Mitsubishi Tanabe Pharma Corp
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Application filed by Mitsubishi Tanabe Pharma Corp filed Critical Mitsubishi Tanabe Pharma Corp
Publication of PT2102224E publication Critical patent/PT2102224E/pt

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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H7/00—Compounds containing non-saccharide radicals linked to saccharide radicals by a carbon-to-carbon bond
    • C07H7/04—Carbocyclic radicals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/70—Carbohydrates; Sugars; Derivatives thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/70—Carbohydrates; Sugars; Derivatives thereof
    • A61K31/7028—Compounds having saccharide radicals attached to non-saccharide compounds by glycosidic linkages
    • A61K31/7034—Compounds having saccharide radicals attached to non-saccharide compounds by glycosidic linkages attached to a carbocyclic compound, e.g. phloridzin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/12—Drugs for disorders of the urinary system of the kidneys
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A61P17/02—Drugs for dermatological disorders for treating wounds, ulcers, burns, scars, keloids, or the like
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/06—Antihyperlipidemics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/12—Drugs for disorders of the metabolism for electrolyte homeostasis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/48—Drugs for disorders of the endocrine system of the pancreatic hormones
    • A61P5/50—Drugs for disorders of the endocrine system of the pancreatic hormones for increasing or potentiating the activity of insulin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives
PT78503067T 2006-12-04 2007-12-03 FORMA CRISTALINA HEMI-HIDRATADA DE 1-(ß-DGLICOPIRANOSIL)- 4-METIL-3-[5-(4-FLUOROFENIL)-2- TIENILMETIL]BENZENO PT2102224E (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US86842606P 2006-12-04 2006-12-04
JP2006327019 2006-12-04

Publications (1)

Publication Number Publication Date
PT2102224E true PT2102224E (pt) 2014-04-07

Family

ID=38973167

Family Applications (1)

Application Number Title Priority Date Filing Date
PT78503067T PT2102224E (pt) 2006-12-04 2007-12-03 FORMA CRISTALINA HEMI-HIDRATADA DE 1-(ß-DGLICOPIRANOSIL)- 4-METIL-3-[5-(4-FLUOROFENIL)-2- TIENILMETIL]BENZENO

Country Status (34)

Country Link
US (2) US7943582B2 (pt)
EP (1) EP2102224B2 (pt)
JP (1) JP5159788B2 (pt)
KR (1) KR101146095B1 (pt)
CN (3) CN101573368B (pt)
AR (3) AR064099A1 (pt)
AU (1) AU2007329895C1 (pt)
BR (1) BRPI0718882B8 (pt)
CA (1) CA2671357C (pt)
CL (1) CL2007003487A1 (pt)
CO (1) CO6210719A2 (pt)
CR (1) CR10861A (pt)
DK (1) DK2102224T4 (pt)
EA (1) EA017103B1 (pt)
EC (1) ECSP099489A (pt)
ES (1) ES2456640T5 (pt)
GT (1) GT200900151A (pt)
IL (1) IL199032A (pt)
ME (1) ME01829B (pt)
MX (1) MX2009005857A (pt)
MY (1) MY153702A (pt)
NO (1) NO344354B1 (pt)
NZ (1) NZ577545A (pt)
PA (1) PA8759401A1 (pt)
PE (3) PE20130591A1 (pt)
PL (1) PL2102224T5 (pt)
PT (1) PT2102224E (pt)
RS (1) RS53274B2 (pt)
SI (1) SI2102224T2 (pt)
SV (1) SV2009003285A (pt)
TW (1) TWI403325B (pt)
UY (1) UY30730A1 (pt)
WO (1) WO2008069327A1 (pt)
ZA (1) ZA200903941B (pt)

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