PT1513826E - Novos derivados de indolilpiperidina como agentes anti-histaminicos e antialergicos potentes - Google Patents

Novos derivados de indolilpiperidina como agentes anti-histaminicos e antialergicos potentes

Info

Publication number
PT1513826E
PT1513826E PT03755105T PT03755105T PT1513826E PT 1513826 E PT1513826 E PT 1513826E PT 03755105 T PT03755105 T PT 03755105T PT 03755105 T PT03755105 T PT 03755105T PT 1513826 E PT1513826 E PT 1513826E
Authority
PT
Portugal
Prior art keywords
new
agents
indolilpiperidine
antialergic
antihistaminic
Prior art date
Application number
PT03755105T
Other languages
English (en)
Portuguese (pt)
Inventor
Fonquerna Pou Silvia
Pages Santacana Luis Miguel
Original Assignee
Almirall Prodesfarma Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Almirall Prodesfarma Sa filed Critical Almirall Prodesfarma Sa
Publication of PT1513826E publication Critical patent/PT1513826E/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/06—Antiasthmatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00—Drugs for dermatological disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/02—Ophthalmic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/16—Otologicals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/08—Antiallergic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Pulmonology (AREA)
  • Immunology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Dermatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Hydrogenated Pyridines (AREA)
  • Saccharide Compounds (AREA)
PT03755105T 2002-05-29 2003-05-19 Novos derivados de indolilpiperidina como agentes anti-histaminicos e antialergicos potentes PT1513826E (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
ES200201226A ES2201907B1 (es) 2002-05-29 2002-05-29 Nuevos derivados de indolilpiperidina como potentes agentes antihistaminicos y antialergicos.

Publications (1)

Publication Number Publication Date
PT1513826E true PT1513826E (pt) 2006-05-31

Family

ID=29558514

Family Applications (1)

Application Number Title Priority Date Filing Date
PT03755105T PT1513826E (pt) 2002-05-29 2003-05-19 Novos derivados de indolilpiperidina como agentes anti-histaminicos e antialergicos potentes

Country Status (10)

Country Link
US (1) US7560471B2 (enExample)
EP (1) EP1513826B1 (enExample)
JP (1) JP4485353B2 (enExample)
AT (1) ATE316526T1 (enExample)
AU (1) AU2003242544A1 (enExample)
DE (1) DE60303381T2 (enExample)
DK (1) DK1513826T3 (enExample)
ES (2) ES2201907B1 (enExample)
PT (1) PT1513826E (enExample)
WO (1) WO2003099807A1 (enExample)

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JP2013508414A (ja) 2009-10-22 2013-03-07 バーテックス ファーマシューティカルズ インコーポレイテッド 嚢胞性線維症および他の慢性疾患の治療のための組成物
US8247436B2 (en) 2010-03-19 2012-08-21 Novartis Ag Pyridine and pyrazine derivative for the treatment of CF
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WO2012034095A1 (en) 2010-09-09 2012-03-15 Irm Llc Compounds and compositions as trk inhibitors
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TW201605450A (zh) 2013-12-03 2016-02-16 諾華公司 Ｍｄｍ２抑制劑與ＢＲＡＦ抑制劑之組合及其用途
WO2015162558A1 (en) 2014-04-24 2015-10-29 Novartis Ag Autotaxin inhibitors
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BR112016024533A8 (pt) 2014-04-24 2021-03-30 Novartis Ag derivados de amino pirazina como inibidores de fosfatidilinositol 3-cinase ou sal, seu uso, e composição e combinação farmacêuticas
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Also Published As

Publication number Publication date
DE60303381T2 (de) 2006-10-26
US7560471B2 (en) 2009-07-14
JP4485353B2 (ja) 2010-06-23
JP2005527627A (ja) 2005-09-15
AU2003242544A1 (en) 2003-12-12
DE60303381D1 (de) 2006-04-13
DK1513826T3 (da) 2006-06-06
WO2003099807A1 (en) 2003-12-04
EP1513826A1 (en) 2005-03-16
ATE316526T1 (de) 2006-02-15
ES2201907B1 (es) 2005-06-01
ES2201907A1 (es) 2004-03-16
ES2254964T3 (es) 2006-06-16
US20060094879A1 (en) 2006-05-04
EP1513826B1 (en) 2006-01-25

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