BR0112756A - Composto, composição farmacêutica, métodos para o tratamento de doenças mediadas por prostaglandina, de congestão nasal, asma alérgica, e rinite alérgica, e, uso de um composto - Google Patents
Composto, composição farmacêutica, métodos para o tratamento de doenças mediadas por prostaglandina, de congestão nasal, asma alérgica, e rinite alérgica, e, uso de um compostoInfo
- Publication number
- BR0112756A BR0112756A BR0112756-0A BR0112756A BR0112756A BR 0112756 A BR0112756 A BR 0112756A BR 0112756 A BR0112756 A BR 0112756A BR 0112756 A BR0112756 A BR 0112756A
- Authority
- BR
- Brazil
- Prior art keywords
- compound
- allergic
- methods
- pharmaceutical composition
- mediated diseases
- Prior art date
Links
- 150000001875 compounds Chemical class 0.000 title abstract 4
- 201000010099 disease Diseases 0.000 title abstract 3
- 208000037265 diseases, disorders, signs and symptoms Diseases 0.000 title abstract 3
- 206010028735 Nasal congestion Diseases 0.000 title abstract 2
- 201000009961 allergic asthma Diseases 0.000 title abstract 2
- 208000006673 asthma Diseases 0.000 title abstract 2
- 230000001404 mediated effect Effects 0.000 title abstract 2
- 238000000034 method Methods 0.000 title abstract 2
- 239000008194 pharmaceutical composition Substances 0.000 title abstract 2
- 150000003180 prostaglandins Chemical class 0.000 title abstract 2
- 206010039085 Rhinitis allergic Diseases 0.000 title 1
- 201000010105 allergic rhinitis Diseases 0.000 title 1
- GTIUBIOUTIDMOU-UHFFFAOYSA-N N1C=CC2=CC=CC=C12.C1CCCC1 Chemical class N1C=CC2=CC=CC=C12.C1CCCC1 GTIUBIOUTIDMOU-UHFFFAOYSA-N 0.000 abstract 1
- 230000000172 allergic effect Effects 0.000 abstract 1
- 208000010668 atopic eczema Diseases 0.000 abstract 1
- 239000002089 prostaglandin antagonist Substances 0.000 abstract 1
Classifications
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- H—ELECTRICITY
- H04—ELECTRIC COMMUNICATION TECHNIQUE
- H04W—WIRELESS COMMUNICATION NETWORKS
- H04W52/00—Power management, e.g. TPC [Transmission Power Control], power saving or power classes
- H04W52/04—TPC
- H04W52/38—TPC being performed in particular situations
- H04W52/46—TPC being performed in particular situations in multi hop networks, e.g. wireless relay networks
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/56—Ring systems containing three or more rings
- C07D209/80—[b, c]- or [b, d]-condensed
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/02—Nasal agents, e.g. decongestants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/06—Antiasthmatics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/16—Otologicals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/56—Ring systems containing three or more rings
- C07D209/80—[b, c]- or [b, d]-condensed
- C07D209/94—[b, c]- or [b, d]-condensed containing carbocyclic rings other than six-membered
-
- H—ELECTRICITY
- H04—ELECTRIC COMMUNICATION TECHNIQUE
- H04B—TRANSMISSION
- H04B17/00—Monitoring; Testing
- H04B17/30—Monitoring; Testing of propagation channels
- H04B17/309—Measuring or estimating channel quality parameters
- H04B17/318—Received signal strength
-
- H—ELECTRICITY
- H04—ELECTRIC COMMUNICATION TECHNIQUE
- H04W—WIRELESS COMMUNICATION NETWORKS
- H04W48/00—Access restriction; Network selection; Access point selection
- H04W48/02—Access restriction performed under specific conditions
- H04W48/04—Access restriction performed under specific conditions based on user or terminal location or mobility data, e.g. moving direction, speed
-
- H—ELECTRICITY
- H04—ELECTRIC COMMUNICATION TECHNIQUE
- H04W—WIRELESS COMMUNICATION NETWORKS
- H04W52/00—Power management, e.g. TPC [Transmission Power Control], power saving or power classes
- H04W52/04—TPC
- H04W52/06—TPC algorithms
- H04W52/14—Separate analysis of uplink or downlink
- H04W52/146—Uplink power control
-
- H—ELECTRICITY
- H04—ELECTRIC COMMUNICATION TECHNIQUE
- H04W—WIRELESS COMMUNICATION NETWORKS
- H04W52/00—Power management, e.g. TPC [Transmission Power Control], power saving or power classes
- H04W52/04—TPC
- H04W52/18—TPC being performed according to specific parameters
- H04W52/24—TPC being performed according to specific parameters using SIR [Signal to Interference Ratio] or other wireless path parameters
-
- H—ELECTRICITY
- H04—ELECTRIC COMMUNICATION TECHNIQUE
- H04W—WIRELESS COMMUNICATION NETWORKS
- H04W52/00—Power management, e.g. TPC [Transmission Power Control], power saving or power classes
- H04W52/04—TPC
- H04W52/18—TPC being performed according to specific parameters
- H04W52/28—TPC being performed according to specific parameters using user profile, e.g. mobile speed, priority or network state, e.g. standby, idle or non transmission
- H04W52/288—TPC being performed according to specific parameters using user profile, e.g. mobile speed, priority or network state, e.g. standby, idle or non transmission taking into account the usage mode, e.g. hands-free, data transmission, telephone
-
- H—ELECTRICITY
- H04—ELECTRIC COMMUNICATION TECHNIQUE
- H04W—WIRELESS COMMUNICATION NETWORKS
- H04W48/00—Access restriction; Network selection; Access point selection
- H04W48/20—Selecting an access point
-
- H—ELECTRICITY
- H04—ELECTRIC COMMUNICATION TECHNIQUE
- H04W—WIRELESS COMMUNICATION NETWORKS
- H04W52/00—Power management, e.g. TPC [Transmission Power Control], power saving or power classes
- H04W52/04—TPC
-
- H—ELECTRICITY
- H04—ELECTRIC COMMUNICATION TECHNIQUE
- H04W—WIRELESS COMMUNICATION NETWORKS
- H04W52/00—Power management, e.g. TPC [Transmission Power Control], power saving or power classes
- H04W52/04—TPC
- H04W52/18—TPC being performed according to specific parameters
- H04W52/24—TPC being performed according to specific parameters using SIR [Signal to Interference Ratio] or other wireless path parameters
- H04W52/245—TPC being performed according to specific parameters using SIR [Signal to Interference Ratio] or other wireless path parameters taking into account received signal strength
-
- H—ELECTRICITY
- H04—ELECTRIC COMMUNICATION TECHNIQUE
- H04W—WIRELESS COMMUNICATION NETWORKS
- H04W52/00—Power management, e.g. TPC [Transmission Power Control], power saving or power classes
- H04W52/04—TPC
- H04W52/18—TPC being performed according to specific parameters
- H04W52/24—TPC being performed according to specific parameters using SIR [Signal to Interference Ratio] or other wireless path parameters
- H04W52/247—TPC being performed according to specific parameters using SIR [Signal to Interference Ratio] or other wireless path parameters where the output power of a terminal is based on a path parameter sent by another terminal
Abstract
"COMPOSTO, COMPOSIçãO FARMACêUTICA, MéTODOS PARA O TRATAMENTO DE DOENçAS MEDIADAS POR PROSTAGLANDINA, DE CONGESTãO NASAL, ASMA ALéRGICA, E RINITE ALéRGICA, E, USO DE UM COMPOSTO". Derivados de ciclo-pentano-indol substituído são antagonistas de prostaglandinas, e como tais são úteis para o tratamento de doenças mediadas por prostaglandina.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US22068300P | 2000-07-25 | 2000-07-25 | |
PCT/CA2001/001069 WO2002008186A2 (en) | 2000-07-25 | 2001-07-23 | Cyclopentanoindoles, compositions containing such compounds and methods of treatment |
Publications (1)
Publication Number | Publication Date |
---|---|
BR0112756A true BR0112756A (pt) | 2003-06-24 |
Family
ID=22824535
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BR0112756-0A BR0112756A (pt) | 2000-07-25 | 2001-07-23 | Composto, composição farmacêutica, métodos para o tratamento de doenças mediadas por prostaglandina, de congestão nasal, asma alérgica, e rinite alérgica, e, uso de um composto |
Country Status (34)
Country | Link |
---|---|
US (1) | US6410583B1 (pt) |
EP (1) | EP1305286B1 (pt) |
JP (1) | JP4119745B2 (pt) |
KR (1) | KR100746814B1 (pt) |
CN (1) | CN1214007C (pt) |
AT (1) | ATE284388T1 (pt) |
AU (2) | AU7743001A (pt) |
BG (1) | BG66084B1 (pt) |
BR (1) | BR0112756A (pt) |
CA (1) | CA2416867C (pt) |
CZ (1) | CZ2003236A3 (pt) |
DE (1) | DE60107687T2 (pt) |
DK (1) | DK1305286T3 (pt) |
DZ (1) | DZ3402A1 (pt) |
EA (1) | EA006765B1 (pt) |
EC (1) | ECSP034428A (pt) |
EE (1) | EE05287B1 (pt) |
ES (1) | ES2231526T3 (pt) |
GE (1) | GEP20053595B (pt) |
HK (1) | HK1058934A1 (pt) |
HR (1) | HRP20021039B1 (pt) |
HU (1) | HUP0301745A3 (pt) |
IL (2) | IL153406A0 (pt) |
IS (1) | IS2170B (pt) |
MX (1) | MXPA03000710A (pt) |
NO (1) | NO325011B1 (pt) |
NZ (1) | NZ523106A (pt) |
PL (1) | PL207342B1 (pt) |
PT (1) | PT1305286E (pt) |
RS (1) | RS50491B (pt) |
SK (1) | SK287507B6 (pt) |
UA (1) | UA73787C2 (pt) |
WO (1) | WO2002008186A2 (pt) |
ZA (1) | ZA200300554B (pt) |
Families Citing this family (50)
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US7273883B2 (en) * | 2000-09-14 | 2007-09-25 | Allergan, Inc. | Prostaglandin EP4 antagonist |
US7217725B2 (en) * | 2000-09-14 | 2007-05-15 | Allergan, Inc. | Prostaglandin D2 antagonist |
US6777407B2 (en) | 2000-11-03 | 2004-08-17 | Wyeth | Cyclopenta[b][1,4]diazepino[6,7,1-hi]indoles and derivatives |
US7141563B2 (en) | 2000-11-03 | 2006-11-28 | Wyeth | Process for the preparation of 1, 2, 3, 4, 8, 9, 10, 10a-octahydro-7bH-cyclopenta[b] [1, 4]diazepino[6, 7, 1-hi] indole derivatives |
AR031200A1 (es) | 2000-11-03 | 2003-09-10 | Wyeth Corp | Cicloocta [b] [1,4] diazepino [6,7,1-hi] indoles y derivados |
US6916922B2 (en) | 2000-11-03 | 2005-07-12 | Wyeth | Process for the preparation of 1,2,3,4,8,9,10,10a-octahydro-7bH-cyclopenta [B] [1,4] diazepino- [6,7,1-hi] indole derivatives |
EP1330457B1 (en) * | 2000-11-03 | 2004-10-20 | Wyeth | Cyclopenta[b][1,4] diazepino[6,7,1-hi]indoles as 5ht2c antagonists |
US6784172B2 (en) | 2000-11-03 | 2004-08-31 | Wyeth | Processes for preparation of cyclopenta[b][1,4]diazepino[6,7,1-hi]indoles and derivatives |
US6858604B2 (en) | 2000-11-03 | 2005-02-22 | Wyeth | Cyclohepta[b][1,4]diazepino[6,7,1-hi]indoles and derivatives |
AR038136A1 (es) * | 2002-01-24 | 2004-12-29 | Merck Frosst Canada Inc | Cicloalcanindoles con sustitucion con fluor composiciones que contienen estos compuestos y metodos de tratamiento |
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TW200307540A (en) | 2002-04-25 | 2003-12-16 | Wyeth Corp | [1, 4]Diazocino[7, 8, 1-hi] indole derivatives as antipsychotic and antiobesity agents |
TW200307682A (en) | 2002-04-25 | 2003-12-16 | Wyeth Corp | 1,2,3,4,7,8-Hexahydro-6H-[1,4]diazepino[6,7,1-ij]quinoline derivatives as antipsychotic and antiobesity agents |
TW200400963A (en) | 2002-05-21 | 2004-01-16 | Wyeth Corp | R-enantiomers of pyranoindole derivatives and the use thereof for the treatment of hepatitis C virus infection or disease |
TW200400818A (en) | 2002-05-21 | 2004-01-16 | Wyeth Corp | Method for the use of pyranoindole derivatives to treat infection with hepatitis C virus |
AR041089A1 (es) * | 2003-05-15 | 2005-05-04 | Merck & Co Inc | Procedimiento y composiciones farmaceutiicas para tratar aterosclerosis, dislipidemias y afecciones relacionadas |
AU2004240705A1 (en) * | 2003-05-20 | 2004-12-02 | Merck Frosst Canada & Co. | Fluoro-methanesulfonyl-substituted cycloalkanoindoles and their use as prostaglandin D2 antagonists |
CA2527773A1 (en) * | 2003-06-12 | 2004-12-23 | Merck Frosst Canada Ltd. | Cycloalkanepyrrolopyridines as dp receptor antagonists |
US20080153817A1 (en) * | 2003-08-07 | 2008-06-26 | Dirk Beher | Treatment for Alzheimer's Disease and Related Conditions |
US20050107350A1 (en) * | 2003-08-22 | 2005-05-19 | Pharmacia Corporation | Method for the treatment or prevention of bone disorders with a cyclooxygenase-2 inhibitor alone and in combination with a bone disorder treatment agent and compositions therewith |
PE20050483A1 (es) | 2003-10-31 | 2005-08-25 | Arena Pharm Inc | Derivados de tetrazol de formula (i), sus composiciones farmaceuticas y procesos para producir composiciones farmaceuticas |
US7019022B2 (en) * | 2003-12-15 | 2006-03-28 | Merck Frosst Canada & Co. | Substituted tetrahydrocarbazole and cyclopentanoindole derivatives |
KR20070033033A (ko) | 2004-07-16 | 2007-03-23 | 프로테오시스 악티엔게젤샤프트 | 염증성 질환 치료제로서 parp 및 sir 조절 활성을갖는 무스카린 길항제 |
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CN101160125A (zh) * | 2005-04-13 | 2008-04-09 | 默克公司 | 烟酸受体激动剂、含有这样化合物的组合物和治疗方法 |
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US20100260841A1 (en) * | 2007-02-08 | 2010-10-14 | Paolini John F | Method of Treating Atherosclerosis, Dyslipidemias and Related Conditions |
KR20190004843A (ko) * | 2008-07-23 | 2019-01-14 | 아레나 파마슈티칼스, 인크. | 자가면역성 및 염증성의 장애의 치료에 유용한 치환된 1,2,3,4-테트라히드로시클로펜타[b]인돌-3-일)아세트산 유도체 |
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US20180021302A1 (en) * | 2015-02-13 | 2018-01-25 | Institut National De La Sante Et De La Recherche Medicale (Inserm) | Ptgdr-1 and/or ptgdr-2 antagonists for preventing and/or treating systemic lupus erythematosus |
PL3310760T3 (pl) | 2015-06-22 | 2023-03-06 | Arena Pharmaceuticals, Inc. | Krystaliczna sól L-argininy kwasu (R)-2-(7-(4-cyklopentylo-3-(trifluorometylo)benzyloksy)- 1,2,3,4-tetrahydrocyklo-penta[b]indol-3-ilo)octowego do zastosowania w zaburzeniach związanych z receptorem S1P1 |
CN110545848A (zh) | 2017-02-16 | 2019-12-06 | 艾尼纳制药公司 | 用于治疗具有肠外表现的炎症性肠病的化合物和方法 |
CN110520124A (zh) | 2017-02-16 | 2019-11-29 | 艾尼纳制药公司 | 用于治疗原发性胆汁性胆管炎的化合物和方法 |
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-
2001
- 2001-07-20 US US09/909,636 patent/US6410583B1/en not_active Expired - Lifetime
- 2001-07-23 ES ES01955162T patent/ES2231526T3/es not_active Expired - Lifetime
- 2001-07-23 MX MXPA03000710A patent/MXPA03000710A/es active IP Right Grant
- 2001-07-23 SK SK93-2003A patent/SK287507B6/sk not_active IP Right Cessation
- 2001-07-23 PT PT01955162T patent/PT1305286E/pt unknown
- 2001-07-23 AU AU7743001A patent/AU7743001A/xx active Pending
- 2001-07-23 RS YUP-979/02A patent/RS50491B/sr unknown
- 2001-07-23 DE DE60107687T patent/DE60107687T2/de not_active Expired - Lifetime
- 2001-07-23 EP EP01955162A patent/EP1305286B1/en not_active Expired - Lifetime
- 2001-07-23 CZ CZ2003236A patent/CZ2003236A3/cs unknown
- 2001-07-23 EA EA200300171A patent/EA006765B1/ru not_active IP Right Cessation
- 2001-07-23 UA UA2003021565A patent/UA73787C2/uk unknown
- 2001-07-23 DK DK01955162T patent/DK1305286T3/da active
- 2001-07-23 PL PL363168A patent/PL207342B1/pl not_active IP Right Cessation
- 2001-07-23 DZ DZ013402A patent/DZ3402A1/fr active
- 2001-07-23 CA CA002416867A patent/CA2416867C/en not_active Expired - Fee Related
- 2001-07-23 NZ NZ523106A patent/NZ523106A/en not_active IP Right Cessation
- 2001-07-23 BR BR0112756-0A patent/BR0112756A/pt active Search and Examination
- 2001-07-23 AT AT01955162T patent/ATE284388T1/de active
- 2001-07-23 KR KR1020037001117A patent/KR100746814B1/ko active IP Right Grant
- 2001-07-23 WO PCT/CA2001/001069 patent/WO2002008186A2/en active IP Right Grant
- 2001-07-23 JP JP2002514093A patent/JP4119745B2/ja not_active Expired - Fee Related
- 2001-07-23 IL IL15340601A patent/IL153406A0/xx active IP Right Grant
- 2001-07-23 GE GE5105A patent/GEP20053595B/en unknown
- 2001-07-23 HU HU0301745A patent/HUP0301745A3/hu unknown
- 2001-07-23 EE EEP200300033A patent/EE05287B1/xx not_active IP Right Cessation
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2002
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2003
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