PT101654B - Processo para a obtencao de 3-<<2-{4-(6-fluoro-benzo-{d}-isoxazol-3-il)piperidin-1-il}-etil>>-2-metil-6,7,8,9-tetra-hidro-4h-pirido-{1,2-a}pirimidin-4-ona - Google Patents
Processo para a obtencao de 3-<<2-{4-(6-fluoro-benzo-{d}-isoxazol-3-il)piperidin-1-il}-etil>>-2-metil-6,7,8,9-tetra-hidro-4h-pirido-{1,2-a}pirimidin-4-ona Download PDFInfo
- Publication number
- PT101654B PT101654B PT101654A PT10165495A PT101654B PT 101654 B PT101654 B PT 101654B PT 101654 A PT101654 A PT 101654A PT 10165495 A PT10165495 A PT 10165495A PT 101654 B PT101654 B PT 101654B
- Authority
- PT
- Portugal
- Prior art keywords
- tetrahydro
- pyrimidin
- pyrido
- methyl
- fluoro
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
ES09400252A ES2074966B1 (es) | 1994-02-11 | 1994-02-11 | Procedimiento para la obtencion de 3-(2-(4-(6-fluoro-benzo(d)isoxazol-3-il)piperidin-1-il)-etil)-2-metil-6,7,8,9-tetrahidro-4h-pirido-(1,2-a)pirimidin-4-ona. |
Publications (2)
Publication Number | Publication Date |
---|---|
PT101654A PT101654A (pt) | 1995-09-12 |
PT101654B true PT101654B (pt) | 2002-01-30 |
Family
ID=8285178
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
PT101654A PT101654B (pt) | 1994-02-11 | 1995-02-09 | Processo para a obtencao de 3-<<2-{4-(6-fluoro-benzo-{d}-isoxazol-3-il)piperidin-1-il}-etil>>-2-metil-6,7,8,9-tetra-hidro-4h-pirido-{1,2-a}pirimidin-4-ona |
Country Status (14)
Country | Link |
---|---|
KR (1) | KR100221108B1 (de) |
AT (1) | AT405401B (de) |
CZ (1) | CZ286398B6 (de) |
EG (1) | EG20877A (de) |
ES (1) | ES2074966B1 (de) |
FI (1) | FI110000B (de) |
GR (1) | GR1002344B (de) |
HU (1) | HU222110B1 (de) |
IS (1) | IS1766B (de) |
NO (1) | NO306022B1 (de) |
PL (1) | PL181420B1 (de) |
PT (1) | PT101654B (de) |
RU (1) | RU2123004C1 (de) |
SK (1) | SK281752B6 (de) |
Families Citing this family (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
ES2101646B1 (es) * | 1995-04-12 | 1998-04-01 | Ferrer Int | Nuevo compuesto derivado del cromeno. |
ES2144355B1 (es) * | 1997-12-30 | 2001-01-01 | Ferrer Int | Compuestos derivados del cromeno. |
DE60009959T2 (de) * | 2000-05-05 | 2005-03-31 | Rpg Life Sciences Limited | Verfahren zur herstellung von antipsychotischem 3-[2-[4-(6-fluoro-1,2-benzisoxazol-3-yl)-1-piperidinyl]ethyl]-6,7,8,9-tetrahydro-2-methyl-4h-pyrido[1,2-a]pyrimidin-4-on |
HUP0302874A2 (hu) | 2000-08-14 | 2003-12-29 | Teva Pharmaceutical Industries Ltd. | Eljárás risperidon előállítására |
KR20040034996A (ko) | 2002-10-18 | 2004-04-29 | 한미약품 주식회사 | 리스페리돈의 개선된 제조방법 |
WO2004043923A1 (en) | 2002-11-13 | 2004-05-27 | Synthon B.V. | Process for making risperidone and intermediates therefor |
JP5315336B2 (ja) * | 2007-04-19 | 2013-10-16 | 又欣 李 | 精神疾患治療用の新規化合物とその調剤及び使用 |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4352811A (en) * | 1981-11-12 | 1982-10-05 | Hoechst-Roussel Pharmaceuticals Inc. | 3-(1-Substituted-4-piperidyl)-1,2-benzisoxazoles |
US4804663A (en) * | 1985-03-27 | 1989-02-14 | Janssen Pharmaceutica N.V. | 3-piperidinyl-substituted 1,2-benzisoxazoles and 1,2-benzisothiazoles |
US4980365A (en) * | 1987-07-13 | 1990-12-25 | Hoechst-Roussel Pharmaceuticals Inc. | N-substituted-5,6-dimethoxy-1,2-benzisoxazole-3-propanamine and related compounds as analgesic and hypotensive agents |
-
1994
- 1994-02-11 ES ES09400252A patent/ES2074966B1/es not_active Expired - Fee Related
-
1995
- 1995-02-01 GR GR950100035A patent/GR1002344B/el not_active IP Right Cessation
- 1995-02-07 SK SK156-95A patent/SK281752B6/sk not_active IP Right Cessation
- 1995-02-08 IS IS4259A patent/IS1766B/is unknown
- 1995-02-08 CZ CZ1995329A patent/CZ286398B6/cs not_active IP Right Cessation
- 1995-02-09 PT PT101654A patent/PT101654B/pt active IP Right Grant
- 1995-02-09 EG EG11595A patent/EG20877A/xx active
- 1995-02-09 NO NO950501A patent/NO306022B1/no not_active IP Right Cessation
- 1995-02-10 PL PL95307200A patent/PL181420B1/pl not_active IP Right Cessation
- 1995-02-10 AT AT0024995A patent/AT405401B/de not_active IP Right Cessation
- 1995-02-10 HU HU9500418A patent/HU222110B1/hu not_active IP Right Cessation
- 1995-02-10 RU RU95101859/04A patent/RU2123004C1/ru not_active IP Right Cessation
- 1995-02-10 FI FI950579A patent/FI110000B/fi not_active IP Right Cessation
- 1995-02-11 KR KR1019950002516A patent/KR100221108B1/ko not_active IP Right Cessation
Also Published As
Publication number | Publication date |
---|---|
ATA24995A (de) | 1998-12-15 |
HU222110B1 (hu) | 2003-04-28 |
SK281752B6 (sk) | 2001-07-10 |
RU95101859A (ru) | 1997-03-20 |
NO950501D0 (no) | 1995-02-09 |
IS4259A (is) | 1995-08-12 |
HUT70169A (en) | 1995-09-28 |
PL307200A1 (en) | 1995-08-21 |
EG20877A (en) | 2000-05-31 |
HU9500418D0 (en) | 1995-03-28 |
ES2074966B1 (es) | 1996-06-16 |
AT405401B (de) | 1999-08-25 |
FI110000B (fi) | 2002-11-15 |
IS1766B (is) | 2001-03-15 |
ES2074966A1 (es) | 1995-09-16 |
KR950032196A (ko) | 1995-12-20 |
FI950579A (fi) | 1995-08-12 |
RU2123004C1 (ru) | 1998-12-10 |
CZ32995A3 (en) | 1995-09-13 |
SK15695A3 (en) | 1995-10-11 |
FI950579A0 (fi) | 1995-02-10 |
GR1002344B (el) | 1996-05-24 |
PL181420B1 (pl) | 2001-07-31 |
NO306022B1 (no) | 1999-09-06 |
CZ286398B6 (en) | 2000-04-12 |
NO950501L (no) | 1995-08-14 |
KR100221108B1 (ko) | 1999-09-15 |
PT101654A (pt) | 1995-09-12 |
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Legal Events
Date | Code | Title | Description |
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FG3A | Patent granted, date of granting |
Effective date: 20011031 |
|
PC3A | Transfer or assignment |
Free format text: LABORATORIOS VITA, S.A. ES Effective date: 20030718 |
|
PC3A | Transfer or assignment |
Free format text: VITA CIENTIFICA ES Effective date: 20050107 |
|
PC4A | Transfer of assignment |
Owner name: INKE, S. A., ES Effective date: 20071203 |