PL307200A1 - Method of obtaining 3-[2-[4-(6-fluoro-benzo[d]isoxazol-3-yl)piperidin-1-yl]ethyl]-2-methyl-6,7,8,9-tetrahydro-4h-pyridil[1,2-a]pyrimidin-4-one and intermediate compounds - Google Patents

Method of obtaining 3-[2-[4-(6-fluoro-benzo[d]isoxazol-3-yl)piperidin-1-yl]ethyl]-2-methyl-6,7,8,9-tetrahydro-4h-pyridil[1,2-a]pyrimidin-4-one and intermediate compounds

Info

Publication number
PL307200A1
PL307200A1 PL95307200A PL30720095A PL307200A1 PL 307200 A1 PL307200 A1 PL 307200A1 PL 95307200 A PL95307200 A PL 95307200A PL 30720095 A PL30720095 A PL 30720095A PL 307200 A1 PL307200 A1 PL 307200A1
Authority
PL
Poland
Prior art keywords
pyridil
isoxazol
pyrimidin
piperidin
benzo
Prior art date
Application number
PL95307200A
Other versions
PL181420B1 (en
Inventor
Pere Dalmases Barjoan
Francisco Marquillas Olondriz
Joan Huguet Clotet
Ana Bosch Rovira
Castillo Nieto Juan Carlos Del
Jose Maria Caldero Ges
Original Assignee
Vita Invest Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Vita Invest Sa filed Critical Vita Invest Sa
Publication of PL307200A1 publication Critical patent/PL307200A1/en
Publication of PL181420B1 publication Critical patent/PL181420B1/en

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
PL95307200A 1994-02-11 1995-02-10 Method of obtaining 3-[2-[4-(6-fluoro-benzo[d]isoxazol-3-yl)piperidin-1-yl]ethyl]-2-methyl-6,7,8,9-tetrahydro-4h-pyridil[1,2-a]pyrimidin-4-one and intermediate compounds PL181420B1 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
ES09400252A ES2074966B1 (en) 1994-02-11 1994-02-11 PROCEDURE FOR OBTAINING 3- (2- (4- (6-FLUORO-BENZO (D) ISOXAZOL-3-IL) PIPERIDIN-1-IL) -ETIL) -2-METHYL-6,7,8,9- TETRAHIDRO-4H-PIRIDO- (1,2-A) PIRIMIDIN-4-ONA.

Publications (2)

Publication Number Publication Date
PL307200A1 true PL307200A1 (en) 1995-08-21
PL181420B1 PL181420B1 (en) 2001-07-31

Family

ID=8285178

Family Applications (1)

Application Number Title Priority Date Filing Date
PL95307200A PL181420B1 (en) 1994-02-11 1995-02-10 Method of obtaining 3-[2-[4-(6-fluoro-benzo[d]isoxazol-3-yl)piperidin-1-yl]ethyl]-2-methyl-6,7,8,9-tetrahydro-4h-pyridil[1,2-a]pyrimidin-4-one and intermediate compounds

Country Status (14)

Country Link
KR (1) KR100221108B1 (en)
AT (1) AT405401B (en)
CZ (1) CZ286398B6 (en)
EG (1) EG20877A (en)
ES (1) ES2074966B1 (en)
FI (1) FI110000B (en)
GR (1) GR1002344B (en)
HU (1) HU222110B1 (en)
IS (1) IS1766B (en)
NO (1) NO306022B1 (en)
PL (1) PL181420B1 (en)
PT (1) PT101654B (en)
RU (1) RU2123004C1 (en)
SK (1) SK281752B6 (en)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2101646B1 (en) * 1995-04-12 1998-04-01 Ferrer Int NEW COMPOUND DERIVED FROM CHROMENE.
ES2144355B1 (en) * 1997-12-30 2001-01-01 Ferrer Int COMPOUNDS DERIVED FROM THE CHROME.
DE60009959T2 (en) * 2000-05-05 2005-03-31 Rpg Life Sciences Limited PROCESS FOR PREPARING ANTIPSYCHOTIC 3- [2- [4- (6-FLUORO-1,2-BENZOXOXOZOL-3-YL) -1-PIPERIDINYL] ETHYL] -6,7,8,9-TETRAHYDRO-2-METHYL- 4H-pyrido [1,2-A] PYRIMIDIN-4-ON
CZ2003668A3 (en) 2000-08-14 2004-04-14 Teva Pharmaceutical Industries Ltd. Preparation of risperidone
KR20040034996A (en) 2002-10-18 2004-04-29 한미약품 주식회사 Improved method for the preparation of risperidone
AU2003288017A1 (en) 2002-11-13 2004-06-03 Synthon B.V. Process for making risperidone and intermediates therefor
EP2154138B1 (en) * 2007-04-19 2015-08-19 Youxin Li Novel compounds for treatment of psychotic disorders, preparation methods and uses thereof

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4352811A (en) * 1981-11-12 1982-10-05 Hoechst-Roussel Pharmaceuticals Inc. 3-(1-Substituted-4-piperidyl)-1,2-benzisoxazoles
US4804663A (en) * 1985-03-27 1989-02-14 Janssen Pharmaceutica N.V. 3-piperidinyl-substituted 1,2-benzisoxazoles and 1,2-benzisothiazoles
US4980365A (en) * 1987-07-13 1990-12-25 Hoechst-Roussel Pharmaceuticals Inc. N-substituted-5,6-dimethoxy-1,2-benzisoxazole-3-propanamine and related compounds as analgesic and hypotensive agents

Also Published As

Publication number Publication date
PT101654B (en) 2002-01-30
CZ32995A3 (en) 1995-09-13
HU222110B1 (en) 2003-04-28
PT101654A (en) 1995-09-12
NO950501D0 (en) 1995-02-09
ES2074966B1 (en) 1996-06-16
FI950579A0 (en) 1995-02-10
SK15695A3 (en) 1995-10-11
RU95101859A (en) 1997-03-20
FI950579A (en) 1995-08-12
SK281752B6 (en) 2001-07-10
ES2074966A1 (en) 1995-09-16
RU2123004C1 (en) 1998-12-10
KR950032196A (en) 1995-12-20
IS1766B (en) 2001-03-15
IS4259A (en) 1995-08-12
ATA24995A (en) 1998-12-15
AT405401B (en) 1999-08-25
CZ286398B6 (en) 2000-04-12
EG20877A (en) 2000-05-31
HU9500418D0 (en) 1995-03-28
HUT70169A (en) 1995-09-28
NO306022B1 (en) 1999-09-06
FI110000B (en) 2002-11-15
NO950501L (en) 1995-08-14
KR100221108B1 (en) 1999-09-15
GR1002344B (en) 1996-05-24
PL181420B1 (en) 2001-07-31

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Effective date: 20110210