PT100409A - Utilizacao de inibidores de aromatase, por exemplo derivados de imidazopiridina, para a anticoncepcao em primatas femeas sem afectar o ciclo menstrual - Google Patents

Utilizacao de inibidores de aromatase, por exemplo derivados de imidazopiridina, para a anticoncepcao em primatas femeas sem afectar o ciclo menstrual

Info

Publication number
PT100409A
PT100409A PT100409A PT10040992A PT100409A PT 100409 A PT100409 A PT 100409A PT 100409 A PT100409 A PT 100409A PT 10040992 A PT10040992 A PT 10040992A PT 100409 A PT100409 A PT 100409A
Authority
PT
Portugal
Prior art keywords
female
primatas
anticonception
affecting
aromatase inhibitors
Prior art date
Application number
PT100409A
Other languages
English (en)
Other versions
PT100409B (pt
Inventor
Ajay Bhatnagar
Original Assignee
Ciba Geigy Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ciba Geigy Ag filed Critical Ciba Geigy Ag
Publication of PT100409A publication Critical patent/PT100409A/pt
Publication of PT100409B publication Critical patent/PT100409B/pt

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4151,2-Diazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • A61P15/18Feminine contraceptives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
PT100409A 1991-04-24 1992-04-22 Utilizacao de inibidores de aromatase, por exemplo derivados de imidazopiridina, para a anticoncepcao em primatas femeas sem afectar o ciclo menstrual PT100409B (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
CH1227/91A CH683151A5 (de) 1991-04-24 1991-04-24 Antikonzeption bei weiblichen Primaten ohne Beeinflussung des menstruellen Zyklus.

Publications (2)

Publication Number Publication Date
PT100409A true PT100409A (pt) 1993-08-31
PT100409B PT100409B (pt) 1999-10-29

Family

ID=4205470

Family Applications (1)

Application Number Title Priority Date Filing Date
PT100409A PT100409B (pt) 1991-04-24 1992-04-22 Utilizacao de inibidores de aromatase, por exemplo derivados de imidazopiridina, para a anticoncepcao em primatas femeas sem afectar o ciclo menstrual

Country Status (25)

Country Link
US (1) US5583128A (pt)
JP (1) JP3710830B2 (pt)
KR (1) KR100219017B1 (pt)
AT (1) AT401873B (pt)
AU (1) AU654540B2 (pt)
BE (1) BE1005781A3 (pt)
CA (1) CA2066807C (pt)
CH (1) CH683151A5 (pt)
DE (1) DE4213005B4 (pt)
DK (1) DK176332B1 (pt)
FR (1) FR2675693B1 (pt)
GB (1) GB2256137B (pt)
IE (1) IE64875B1 (pt)
IL (1) IL101688A (pt)
IT (1) IT1257474B (pt)
LU (1) LU88106A1 (pt)
MX (1) MX9201908A (pt)
NL (1) NL9200755A (pt)
NO (1) NO300156B1 (pt)
NZ (1) NZ242443A (pt)
PH (1) PH30495A (pt)
PT (1) PT100409B (pt)
SE (1) SE512618C2 (pt)
TW (1) TW201267B (pt)
ZA (1) ZA922931B (pt)

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ZA9510926B (en) 1994-12-23 1996-07-03 Schering Ag Compounds with progesterone-antagonistic and antiestrogenic action to be used together for female contraception
IT1286866B1 (it) * 1996-10-28 1998-07-17 Menarini Farma Ind Composti furano-eterociclici,loro preparazione ed uso come inibitori di aromatasi
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US6624197B1 (en) 1998-05-08 2003-09-23 Calyx Therapeutics, Inc. Diphenylethylene compounds
US6245814B1 (en) 1998-05-08 2001-06-12 Calyx Therapeutics, Inc. Diphenylethylene compounds
US7105552B2 (en) 1998-05-08 2006-09-12 Theracos, Inc. Heterocyclic analogs of diphenylethylene compounds
US6331633B1 (en) 1998-05-08 2001-12-18 Calyx Therapeutics Inc. Heterocyclic analogs of diphenylethylene compounds
US6485972B1 (en) 1998-10-15 2002-11-26 President And Fellows Of Harvard College WNT signalling in reproductive organs
US7407978B2 (en) * 1999-04-06 2008-08-05 Theracos, Inc. Heterocyclic analogs of diphenylethylene compounds
US6525093B1 (en) * 1999-11-08 2003-02-25 Calyx Therapeutics Inc. Compounds to treat diabetes and associated conditions
US7323496B2 (en) * 1999-11-08 2008-01-29 Theracos, Inc. Compounds for treatment of inflammation, diabetes and related disorders
US20020002200A1 (en) * 2000-02-04 2002-01-03 Bishwagit Nag Novel diphenylethylene compounds
US20080108825A1 (en) * 1999-11-08 2008-05-08 Theracos, Inc. Compounds for treatment of inflammation, diabetes and related disorders
US20080103302A1 (en) * 2000-02-04 2008-05-01 Theracos, Inc. Compounds for treatment of inflammation, diabetes and related disorders
JP2005515207A (ja) * 2001-12-11 2005-05-26 エモリー ユニバーシティ 乳癌の予防において使用するためのビス(シアノフェニル)メチル−トリアゾール
US8685950B2 (en) * 2004-10-04 2014-04-01 Wayne State University Use of aromatase inhibitors for treatment of ectopic pregnancy
CA2619503A1 (en) * 2005-06-28 2007-01-04 Robert F. Casper Aromatase inhibitors for emergency contraception
GT200600381A (es) 2005-08-25 2007-03-28 Compuestos organicos
WO2008019048A1 (en) * 2006-08-04 2008-02-14 Meditrina Pharmaceuticals Use of aromatase inhibitors for thining the endometrium or treating menorrhagia
US20100292150A1 (en) * 2007-12-10 2010-11-18 Meditrina Pharmaceuticals, Inc. Treatment of Menorrhagia with Aromatase Inhibitor
GB0914767D0 (en) 2009-08-24 2009-09-30 Sterix Ltd Compound

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Also Published As

Publication number Publication date
GB2256137B (en) 1995-01-11
PT100409B (pt) 1999-10-29
AU1509292A (en) 1992-10-29
JPH05112467A (ja) 1993-05-07
ITRM920310A1 (it) 1993-10-24
CH683151A5 (de) 1994-01-31
US5583128A (en) 1996-12-10
IL101688A (en) 1997-01-10
AU654540B2 (en) 1994-11-10
DK53392D0 (da) 1992-04-24
ZA922931B (en) 1993-04-28
IT1257474B (it) 1996-01-25
SE9201249D0 (sv) 1992-04-21
NO921575D0 (no) 1992-04-23
DK176332B1 (da) 2007-08-20
NO300156B1 (no) 1997-04-21
IE64875B1 (en) 1995-09-20
DK53392A (da) 1992-10-25
SE9201249L (sv) 1992-10-25
SE512618C2 (sv) 2000-04-10
NL9200755A (nl) 1992-11-16
CA2066807A1 (en) 1992-10-25
DE4213005A1 (de) 1992-10-29
JP3710830B2 (ja) 2005-10-26
PH30495A (en) 1997-05-28
CA2066807C (en) 2003-09-23
IE921318A1 (en) 1992-11-04
KR920019351A (ko) 1992-11-19
IL101688A0 (en) 1992-12-30
BE1005781A3 (fr) 1994-01-25
FR2675693B1 (fr) 1995-06-30
AT401873B (de) 1996-12-27
DE4213005B4 (de) 2005-12-08
GB2256137A (en) 1992-12-02
KR100219017B1 (ko) 1999-09-01
NZ242443A (en) 1996-10-28
TW201267B (pt) 1993-03-01
MX9201908A (es) 1992-11-01
ATA83692A (de) 1996-05-15
LU88106A1 (de) 1993-12-06
NO921575L (no) 1992-10-26
GB9208718D0 (en) 1992-06-10
FR2675693A1 (fr) 1992-10-30
ITRM920310A0 (it) 1992-04-24

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