IT1286866B1 - Composti furano-eterociclici,loro preparazione ed uso come inibitori di aromatasi - Google Patents

Composti furano-eterociclici,loro preparazione ed uso come inibitori di aromatasi

Info

Publication number
IT1286866B1
IT1286866B1 ITFI960253A IT1286866B1 IT 1286866 B1 IT1286866 B1 IT 1286866B1 IT FI960253 A ITFI960253 A IT FI960253A IT 1286866 B1 IT1286866 B1 IT 1286866B1
Authority
IT
Italy
Prior art keywords
furano
preparation
heterocyclic compounds
aromatase inhibitors
aromatase
Prior art date
Application number
Other languages
English (en)
Inventor
Paolo Lombardi
Pietro Giovanna Di
Original Assignee
Menarini Farma Ind
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Menarini Farma Ind filed Critical Menarini Farma Ind
Priority to ITFI960253 priority Critical patent/IT1286866B1/it
Priority to AU49491/97A priority patent/AU4949197A/en
Priority to PCT/EP1997/005854 priority patent/WO1998018791A1/en
Publication of ITFI960253A1 publication Critical patent/ITFI960253A1/it
Application granted granted Critical
Publication of IT1286866B1 publication Critical patent/IT1286866B1/it

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D405/00Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/06Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
ITFI960253 1996-10-28 1996-10-28 Composti furano-eterociclici,loro preparazione ed uso come inibitori di aromatasi IT1286866B1 (it)

Priority Applications (3)

Application Number Priority Date Filing Date Title
ITFI960253 IT1286866B1 (it) 1996-10-28 1996-10-28 Composti furano-eterociclici,loro preparazione ed uso come inibitori di aromatasi
AU49491/97A AU4949197A (en) 1996-10-28 1997-10-23 Heterocyclic furan compounds, their preparation and use as aromatase inhibitors
PCT/EP1997/005854 WO1998018791A1 (en) 1996-10-28 1997-10-23 Heterocyclic furan compounds, their preparation and use as aromatase inhibitors

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
ITFI960253 IT1286866B1 (it) 1996-10-28 1996-10-28 Composti furano-eterociclici,loro preparazione ed uso come inibitori di aromatasi

Publications (2)

Publication Number Publication Date
ITFI960253A1 ITFI960253A1 (it) 1998-04-28
IT1286866B1 true IT1286866B1 (it) 1998-07-17

Family

ID=11351840

Family Applications (1)

Application Number Title Priority Date Filing Date
ITFI960253 IT1286866B1 (it) 1996-10-28 1996-10-28 Composti furano-eterociclici,loro preparazione ed uso come inibitori di aromatasi

Country Status (3)

Country Link
AU (1) AU4949197A (it)
IT (1) IT1286866B1 (it)
WO (1) WO1998018791A1 (it)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB0223915D0 (en) * 2002-10-15 2002-11-20 Univ Cardiff Benzofuran derivatives formulations and uses thereof
EP1756054B1 (en) * 2004-06-01 2010-03-31 F.Hoffmann-La Roche Ag 3-amino-1-arylpropyl indoles as monoamine reuptake inhibitor

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4766140A (en) * 1984-06-18 1988-08-23 Eli Lilly And Company Method of inhibiting aromatase
IT1216256B (it) * 1986-08-13 1990-02-22 Menarini Sas (benzofuran-2-il) imidazoli, con attivita' farmacologica,loro sali e procedimenti di fabbricazione relativi.
NZ221729A (en) * 1986-09-15 1989-07-27 Janssen Pharmaceutica Nv Imidazolyl methyl-substituted benzimidazole derivatives and pharmaceutical compositions
NZ224714A (en) * 1987-06-01 1990-03-27 Janssen Pharmaceutica Nv Substituted benzotriazole derivatives and pharmaceutical compositions
DE3811574A1 (de) * 1988-03-31 1989-10-19 Schering Ag N-substituierte imidazole, verfahren zu ihrer herstellung sowie ihre verwendung in arzneimitteln
DE59010171D1 (de) * 1989-07-14 1996-04-11 Ciba Geigy Ag Substituierte Benzonitrile
AU7124691A (en) * 1990-02-27 1991-08-29 Ciba-Geigy Ag Benzofurans
TW210334B (it) * 1990-12-12 1993-08-01 Ciba Geigy Ag
CH683151A5 (de) * 1991-04-24 1994-01-31 Ciba Geigy Ag Antikonzeption bei weiblichen Primaten ohne Beeinflussung des menstruellen Zyklus.

Also Published As

Publication number Publication date
AU4949197A (en) 1998-05-22
ITFI960253A1 (it) 1998-04-28
WO1998018791A1 (en) 1998-05-07

Similar Documents

Publication Publication Date Title
AT503376A3 (de) Synergistische spot-on-formulierung
EE9900147A (et) Oksadiasoolid, nende saamismeetodid ja kasutamine ravimitena
EE200100185A (et) Asendatud fenüülderivaadid, nende valmistamine jakasutamine
DE69822124D1 (de) Axiallüfter
ID28698A (id) Formulasi antiparasit
EE04721B1 (et) Fenüülksantiini derivaadid, nende valmistamismeetodid ja kasutamine
EE200000621A (et) Pikornaviirusevastased ühendid, nende valmistamine ja kasutamine
BR9711191A (pt) Composto e uso do mesmo
FI103704B1 (fi) Mikrobinvastainen koostumus, sen valmistusmenetelmä ja sen käyttö
ID23083A (id) Popok sekali pakai
DE69921931D1 (de) Axiallüfter
BR9506594A (pt) Composição apropriada para uso tópico
BR9707808A (pt) Composto composição farmacêutica e uso do composto
ID27655A (id) Formulasi mikrokapsul
ID17561A (id) Komposisi untuk pemakaian luar
IT1297886B1 (it) Nifedipina per uso topico
BR9402143A (pt) Composto, composição e uso
EE04346B1 (et) Asoolid, nende valmistamismeetod, kasutamine ja farmatseutiline kompositsioon
BR9612413A (pt) Composto uso do mesmo e composição farmacêutica
ITMI941112A0 (it) Alcaloidi da mappia foetida, loro uso e formulazioni che li contengono
IT1286866B1 (it) Composti furano-eterociclici,loro preparazione ed uso come inibitori di aromatasi
ITFI950221A1 (it) Composti furano-eterociclici, loro preparazione ed uso come inibitori di aromatasi
EE200000179A (et) 1-oxa, aza ja tianaftaleen-2-1 biseetrid fosfolambaani inhibiitoritena
IT243826Y1 (it) Struttura amovibile ad uso igienico-sanitario
ITMI941135A0 (it) Estratti di piliostigma thonningii, loro uso e formulazioni che li contengono

Legal Events

Date Code Title Description
0001 Granted