NO996264L - Behandling av diabetes med tiazolidindion og sulfonylurea - Google Patents

Behandling av diabetes med tiazolidindion og sulfonylurea

Info

Publication number
NO996264L
NO996264L NO996264A NO996264A NO996264L NO 996264 L NO996264 L NO 996264L NO 996264 A NO996264 A NO 996264A NO 996264 A NO996264 A NO 996264A NO 996264 L NO996264 L NO 996264L
Authority
NO
Norway
Prior art keywords
thiazolidinedione
sulfonylurea
diabetes
treatment
Prior art date
Application number
NO996264A
Other languages
English (en)
Other versions
NO326263B1 (no
NO996264D0 (no
Inventor
Stephen Alistair Smith
Original Assignee
Smithkline Beecham Plc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=26311744&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=NO996264(L) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Priority claimed from GBGB9712854.0A external-priority patent/GB9712854D0/en
Priority claimed from GBGB9806710.1A external-priority patent/GB9806710D0/en
Application filed by Smithkline Beecham Plc filed Critical Smithkline Beecham Plc
Publication of NO996264D0 publication Critical patent/NO996264D0/no
Publication of NO996264L publication Critical patent/NO996264L/no
Publication of NO326263B1 publication Critical patent/NO326263B1/no

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/13Amines
    • A61K31/145Amines having sulfur, e.g. thiurams (>N—C(S)—S—C(S)—N< and >N—C(S)—S—S—C(S)—N<), Sulfinylamines (—N=SO), Sulfonylamines (—N=SO2)
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425Thiazoles
    • A61K31/4261,3-Thiazoles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425Thiazoles
    • A61K31/427Thiazoles not condensed and containing further heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/4439Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/64Sulfonylureas, e.g. glibenclamide, tolbutamide, chlorpropamide
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/08Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00Drugs for disorders of the endocrine system
    • A61P5/48Drugs for disorders of the endocrine system of the pancreatic hormones
    • A61P5/50Drugs for disorders of the endocrine system of the pancreatic hormones for increasing or potentiating the activity of insulin

Landscapes

  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Epidemiology (AREA)
  • Diabetes (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Endocrinology (AREA)
  • Emergency Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
NO19996264A 1997-06-18 1999-12-17 Kombinasjon omfattende tiazolidindion og sulfonylurea, anvendelse derav, samt farmasoytisk sammensetning NO326263B1 (no)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GBGB9712854.0A GB9712854D0 (en) 1997-06-18 1997-06-18 Novel method of treatment
GBGB9806710.1A GB9806710D0 (en) 1998-03-27 1998-03-27 Novel method
PCT/EP1998/003688 WO1998057649A1 (en) 1997-06-18 1998-06-15 Treatment of diabetes with thiazolidinedione and sulphonylurea

Publications (3)

Publication Number Publication Date
NO996264D0 NO996264D0 (no) 1999-12-17
NO996264L true NO996264L (no) 2000-02-17
NO326263B1 NO326263B1 (no) 2008-10-27

Family

ID=26311744

Family Applications (3)

Application Number Title Priority Date Filing Date
NO19996264A NO326263B1 (no) 1997-06-18 1999-12-17 Kombinasjon omfattende tiazolidindion og sulfonylurea, anvendelse derav, samt farmasoytisk sammensetning
NO20083276A NO20083276L (no) 1997-06-18 2008-07-24 Behandling av diabetes med tiazolidindion og sulfonylurea
NO2009002C NO2009002I1 (no) 1997-06-18 2009-02-13 5-{4-[2-(N-metyl-N-(2-pyridyl)amino)etoksy]benzyl}tiazolidin-2,4-dionmaleat(salter/solvater)+glimepirid

Family Applications After (2)

Application Number Title Priority Date Filing Date
NO20083276A NO20083276L (no) 1997-06-18 2008-07-24 Behandling av diabetes med tiazolidindion og sulfonylurea
NO2009002C NO2009002I1 (no) 1997-06-18 2009-02-13 5-{4-[2-(N-metyl-N-(2-pyridyl)amino)etoksy]benzyl}tiazolidin-2,4-dionmaleat(salter/solvater)+glimepirid

Country Status (33)

Country Link
EP (3) EP0999845B1 (no)
JP (1) JP2001523270A (no)
KR (3) KR20070011651A (no)
CN (1) CN1168451C (no)
AP (1) AP1600A (no)
AR (2) AR012996A1 (no)
AT (1) ATE353654T1 (no)
AU (1) AU8539298A (no)
BG (2) BG64817B1 (no)
BR (1) BR9810142A (no)
CA (1) CA2294385C (no)
CO (1) CO4940457A1 (no)
CZ (1) CZ299310B6 (no)
DE (1) DE69837089T2 (no)
DZ (1) DZ2522A1 (no)
EA (1) EA003025B1 (no)
ES (1) ES2283064T3 (no)
ID (1) ID24065A (no)
IL (1) IL133137A (no)
IN (1) IN189319B (no)
MA (1) MA24571A1 (no)
MY (1) MY125855A (no)
NO (3) NO326263B1 (no)
NZ (1) NZ501163A (no)
OA (1) OA11510A (no)
PE (1) PE108199A1 (no)
PL (2) PL337510A1 (no)
SK (1) SK286028B6 (no)
TR (1) TR199903096T2 (no)
TW (1) TW542717B (no)
UA (1) UA67743C2 (no)
UY (1) UY25048A1 (no)
WO (1) WO1998057649A1 (no)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9715295D0 (en) * 1997-07-18 1997-09-24 Smithkline Beecham Plc Novel method of treatment
US7045519B2 (en) 1998-06-19 2006-05-16 Chiron Corporation Inhibitors of glycogen synthase kinase 3
DE60037602T2 (de) 1999-04-23 2009-01-08 Smithkline Beecham P.L.C., Brentford Herstellung einer polymorphen Form eines Thiazolidindionderivates
EP1227818A2 (en) 1999-11-01 2002-08-07 Wisconsin Alumni Research Foundation Abc1 modulation for the modulation of cholesterol transport
CA2725833A1 (en) 2001-01-12 2002-07-18 Sun Pharmaceutical Industries Limited Spaced drug delivery system
KR100698595B1 (ko) * 2003-09-29 2007-03-21 보령제약 주식회사 무정형 또는 준결정형 글리메피리드, 이의 제조방법 및 무정형 또는 준결정형 글리메피리드를 포함하는 약학적조성물
AU2004285354B2 (en) 2003-10-31 2009-09-17 Takeda Pharmaceutical Company Limited Solid preparation comprising an insulin sensitizer, an insulin secretagogue and a polyoxyethylene sorbitan fatty acid ester
RU2426530C2 (ru) 2005-12-22 2011-08-20 Такеда Фармасьютикал Компани Лимитед Твердый препарат
CN104158867B (zh) * 2014-08-06 2017-05-17 电子科技大学 一种基于wave协议的信息多跳转发方法

Family Cites Families (32)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS5522636A (en) 1978-08-04 1980-02-18 Takeda Chem Ind Ltd Thiazoliding derivative
JPS5697277A (en) 1980-01-07 1981-08-05 Takeda Chem Ind Ltd Thiazolidine derivative
JPS6051189A (ja) 1983-08-30 1985-03-22 Sankyo Co Ltd チアゾリジン誘導体およびその製造法
US4582839A (en) 1984-03-21 1986-04-15 Takeda Chemical Industries, Ltd. 2,4-thiazolidinediones
CN1003445B (zh) 1984-10-03 1989-03-01 武田药品工业株式会社 噻唑烷二酮衍生物,其制备方法和用途
DK173350B1 (da) 1985-02-26 2000-08-07 Sankyo Co Thiazolidinderivater, deres fremstilling og farmaceutisk paæparat indeholdende dem
JPH06779B2 (ja) 1985-06-10 1994-01-05 武田薬品工業株式会社 チアゾリジオン誘導体およびそれを含んでなる医薬組成物
US4812570A (en) 1986-07-24 1989-03-14 Takeda Chemical Industries, Ltd. Method for producing thiazolidinedione derivatives
EP0842925A1 (en) * 1987-09-04 1998-05-20 Beecham Group Plc Substituted thiazolidinedione derivatives
US4791125A (en) 1987-12-02 1988-12-13 Pfizer Inc. Thiazolidinediones as hypoglycemic and anti-atherosclerosis agents
MX15171A (es) 1988-03-08 1993-05-01 Pfizer Derivados de tiazolidinodiona hipoglicemicos
US5061717A (en) 1988-03-08 1991-10-29 Pfizer Inc. Thiazolidinedione hypoglycemic agents
WO1991007107A1 (en) 1989-11-13 1991-05-30 Pfizer Inc. Oxazolidinedione hypoglycemic agents
US5089514A (en) 1990-06-14 1992-02-18 Pfizer Inc. 3-coxazolyl [phenyl, chromanyl or benzofuranyl]-2-hydroxypropionic acid derivatives and analogs as hypoglycemic agents
WO1992000967A1 (en) 1990-07-03 1992-01-23 Yamanouchi Pharmaceutical Co., Ltd. Bisheterocyclic compound
CA2087437A1 (en) 1990-08-23 1992-02-24 Steven W. Goldstein Hypoglycemic hydroxyurea derivatives
JPH04210683A (ja) 1990-12-06 1992-07-31 Terumo Corp チアゾリジン−2,4−ジオン誘導体およびこれを含有する糖尿病合併症治療薬
US5183823A (en) 1991-04-11 1993-02-02 Takeda Chemical Industries, Ltd. Pyridine n-oxide compounds which are useful as hypoglycemic and hypolipidemic agents
EP0579733B1 (en) 1991-04-11 2001-06-20 PHARMACIA &amp; UPJOHN COMPANY Thiazolidinedione derivatives, production and use thereof
TW222626B (no) 1991-07-22 1994-04-21 Pfizer
FR2680512B1 (fr) 1991-08-20 1995-01-20 Adir Nouveaux derives de 2,4-thiazolidinedione, leur procede de preparation et les compositions pharmaceutiques qui les contiennent.
DE69219136T2 (de) * 1991-08-26 1997-08-28 Pharmacia & Upjohn Co., Kalamazoo, Mich. Flüssiges nahrungsmittel, das 3-guanidinopropionsäure enthält
JPH05271204A (ja) 1992-03-26 1993-10-19 Japan Tobacco Inc 新規なトリアジン誘導体
US5264451A (en) 1992-04-07 1993-11-23 American Home Products Corporation Process for treating hyperglycemia using trifluoromethyl substituted 3H-pyrazol-3-ones
WO1993021166A1 (en) 1992-04-10 1993-10-28 Smithkline Beecham Plc Heterocyclic compounds and their use in the treatment of type ii-diabetes
WO1993022445A1 (en) 1992-05-05 1993-11-11 The Upjohn Company A process for producing pioglitazone metabolite
EP0648212B1 (en) 1992-07-03 2001-10-24 Smithkline Beecham Plc Benzoxazole and benzothiazole derivatives as pharmaceutical
US5232945A (en) 1992-07-20 1993-08-03 Pfizer Inc. 3-aryl-2-hydroxypropionic acid derivatives and analogs as antihypertensives
GB9218830D0 (en) * 1992-09-05 1992-10-21 Smithkline Beecham Plc Novel compounds
US5478852C1 (en) 1993-09-15 2001-03-13 Sankyo Co Use of thiazolidinedione derivatives and related antihyperglycemic agents in the treatment of impaired glucose tolerance in order to prevent or delay the onset of noninsulin-dependent diabetes mellitus
TWI238064B (en) * 1995-06-20 2005-08-21 Takeda Chemical Industries Ltd A pharmaceutical composition for prophylaxis and treatment of diabetes
US5859037A (en) * 1997-02-19 1999-01-12 Warner-Lambert Company Sulfonylurea-glitazone combinations for diabetes

Also Published As

Publication number Publication date
TW542717B (en) 2003-07-21
AU8539298A (en) 1999-01-04
EP1671637A3 (en) 2007-12-19
AP9901717A0 (en) 1999-12-31
IL133137A0 (en) 2001-03-19
BG64817B1 (bg) 2006-05-31
EA200000039A1 (ru) 2000-08-28
DZ2522A1 (fr) 2003-02-01
EA003025B1 (ru) 2002-12-26
BG109397A (bg) 2006-05-31
BG104058A (en) 2000-10-31
KR20080011356A (ko) 2008-02-01
CA2294385A1 (en) 1998-12-23
CZ9904577A3 (en) 2001-05-16
DE69837089D1 (de) 2007-03-29
CN1260719A (zh) 2000-07-19
NZ501163A (en) 2002-02-01
CN1168451C (zh) 2004-09-29
EP1671637A2 (en) 2006-06-21
KR20070011651A (ko) 2007-01-24
AP1600A (en) 2006-04-28
JP2001523270A (ja) 2001-11-20
CO4940457A1 (es) 2000-07-24
AR008025A1 (es) 1999-12-09
IL133137A (en) 2004-02-08
MA24571A1 (fr) 1998-12-31
PE108199A1 (es) 2000-01-14
NO2009002I1 (no) 2009-03-02
NO20083276L (no) 2000-02-17
WO1998057649A1 (en) 1998-12-23
NO326263B1 (no) 2008-10-27
DE69837089T2 (de) 2007-06-21
MY125855A (en) 2006-08-30
EP0999845B1 (en) 2007-02-14
SK286028B6 (sk) 2008-01-07
ID24065A (id) 2000-07-06
AR012996A1 (es) 2000-11-22
ES2283064T3 (es) 2007-10-16
CA2294385C (en) 2007-06-05
NO996264D0 (no) 1999-12-17
KR20010013840A (ko) 2001-02-26
SK179199A3 (en) 2000-11-07
IN189319B (no) 2003-02-08
EP0999845A1 (en) 2000-05-17
HK1028200A1 (en) 2001-02-09
BR9810142A (pt) 2000-08-08
PL198018B1 (pl) 2008-05-30
CZ299310B6 (cs) 2008-06-18
PL337510A1 (en) 2000-08-28
OA11510A (en) 2004-02-03
UY25048A1 (es) 2000-09-29
TR199903096T2 (xx) 2000-08-21
EP2266576A1 (en) 2010-12-29
ATE353654T1 (de) 2007-03-15
UA67743C2 (uk) 2004-07-15

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Legal Events

Date Code Title Description
SPCF Filing of supplementary protection certificate

Free format text: PRODUCT NAME: AVAGLIM - ROSIGLITAZON/GLIMEPIRID; NAT. REG. NO/DATE: EU106349001-008NO 20060713; FIRST REG. NO/DATE: EU , EU106349001-008 20060627

Spc suppl protection certif: 2009002

Filing date: 20090213

MM1K Lapsed by not paying the annual fees