NO831082L - Nye penamforbindelser som kan anvendes som mellomprodukt for fremstilling av beta-laktamase-hemmende forbindelser - Google Patents

Nye penamforbindelser som kan anvendes som mellomprodukt for fremstilling av beta-laktamase-hemmende forbindelser

Info

Publication number
NO831082L
NO831082L NO831082A NO831082A NO831082L NO 831082 L NO831082 L NO 831082L NO 831082 A NO831082 A NO 831082A NO 831082 A NO831082 A NO 831082A NO 831082 L NO831082 L NO 831082L
Authority
NO
Norway
Prior art keywords
compounds
penamine
lactamase
beta
preparation
Prior art date
Application number
NO831082A
Other languages
English (en)
Other versions
NO160299B (no
NO160299C (no
Inventor
Wayne Ernest Barth
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Publication of NO831082L publication Critical patent/NO831082L/no
Application filed by Pfizer filed Critical Pfizer
Priority to NO83831082A priority Critical patent/NO160299C/no
Publication of NO160299B publication Critical patent/NO160299B/no
Publication of NO160299C publication Critical patent/NO160299C/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D499/21—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring with a nitrogen atom directly attached in position 6 and a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2
    • C07D499/28—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring with a nitrogen atom directly attached in position 6 and a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2 with modified 2-carboxyl group
    • C07D499/32—Esters

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Cephalosporin Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
NO83831082A 1979-09-26 1983-03-25 Nye penamforbindelser som kan anvendes som mellomprodukt for fremstilling av beta-laktamase-hemmende forbindelser. NO160299C (no)

Priority Applications (1)

Application Number Priority Date Filing Date Title
NO83831082A NO160299C (no) 1979-09-26 1983-03-25 Nye penamforbindelser som kan anvendes som mellomprodukt for fremstilling av beta-laktamase-hemmende forbindelser.

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US06/079,127 US4256733A (en) 1979-09-26 1979-09-26 Acetoxymethyl penam compounds as β-lactamase inhibitors
NO802836A NO160370C (no) 1979-09-26 1980-09-25 Analogifremgangsmaate for fremstilling av fysiologisk aktive penam-1,1-dioksyd-forbindelser.
NO83831082A NO160299C (no) 1979-09-26 1983-03-25 Nye penamforbindelser som kan anvendes som mellomprodukt for fremstilling av beta-laktamase-hemmende forbindelser.

Publications (3)

Publication Number Publication Date
NO831082L true NO831082L (no) 1981-03-27
NO160299B NO160299B (no) 1988-12-27
NO160299C NO160299C (no) 1989-04-05

Family

ID=22148609

Family Applications (2)

Application Number Title Priority Date Filing Date
NO802836A NO160370C (no) 1979-09-26 1980-09-25 Analogifremgangsmaate for fremstilling av fysiologisk aktive penam-1,1-dioksyd-forbindelser.
NO83831082A NO160299C (no) 1979-09-26 1983-03-25 Nye penamforbindelser som kan anvendes som mellomprodukt for fremstilling av beta-laktamase-hemmende forbindelser.

Family Applications Before (1)

Application Number Title Priority Date Filing Date
NO802836A NO160370C (no) 1979-09-26 1980-09-25 Analogifremgangsmaate for fremstilling av fysiologisk aktive penam-1,1-dioksyd-forbindelser.

Country Status (36)

Country Link
US (1) US4256733A (no)
JP (1) JPS6016958B2 (no)
KR (1) KR840000796B1 (no)
AR (1) AR224547A1 (no)
AT (1) AT366384B (no)
AU (1) AU517074B2 (no)
BE (1) BE885389A (no)
CA (1) CA1150242A (no)
CH (1) CH645646A5 (no)
CS (1) CS212284B2 (no)
DD (1) DD153123A5 (no)
DE (1) DE3035995C2 (no)
DK (1) DK404980A (no)
EG (1) EG14888A (no)
ES (1) ES8106528A1 (no)
FI (2) FI67552C (no)
FR (1) FR2465736A1 (no)
GB (2) GB2059420B (no)
GR (1) GR70065B (no)
HU (1) HU183212B (no)
IE (2) IE50506B1 (no)
IL (1) IL61117A (no)
IN (1) IN154557B (no)
IT (1) IT1132754B (no)
LU (1) LU82795A1 (no)
MX (1) MX6580E (no)
NL (1) NL185923C (no)
NO (2) NO160370C (no)
NZ (1) NZ195058A (no)
PH (1) PH15697A (no)
PL (1) PL126949B1 (no)
PT (1) PT71837B (no)
SE (2) SE449865B (no)
SU (1) SU959628A3 (no)
YU (1) YU41733B (no)
ZA (1) ZA805132B (no)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4364957A (en) * 1979-09-26 1982-12-21 Pfizer Inc. Bis-esters of alkanediols as antibacterial agents
US4511512A (en) * 1980-05-01 1985-04-16 Leo Pharmaceutical Products Ltd. A/S (Lovens Kemiske Produktionsaktiensel skab) Substantially pure dicyclohexyl ammonium 6-β-bromo-penicillanate
US4474698A (en) * 1980-12-11 1984-10-02 Pfizer Inc. Process for preparing esters of penicillanic acid sulfone
US4361513A (en) * 1980-12-11 1982-11-30 Pfizer Inc. Esters of penicillanic acid sulfone
US4558042A (en) * 1981-05-06 1985-12-10 Farmitalia Carlo Erba S.P.A. β-Lactam-containing antibacterial agents and β-lactamase inhibitors
ZA826687B (en) * 1981-09-14 1983-07-27 Pfizer Beta-lactamase inhibiting 2-beta-substituted-2-alpha-methyl 5(r)penam-3-alpha-carboxylic acid 1,1-dioxides and intermediates therefor
JPS58185589A (ja) * 1982-04-23 1983-10-29 Taiho Yakuhin Kogyo Kk ペニシリン誘導体
JPS62198687A (ja) * 1986-02-27 1987-09-02 Taiho Yakuhin Kogyo Kk ２β−置換チオメチルペニシリン誘導体
US4861768A (en) * 1986-02-27 1989-08-29 Taiho Pharmaceutical Company, Limited 2 β-substituted thiomethylpenicillin derivatives and their preparation and use
DE618979T1 (de) * 1991-12-19 1995-05-18 Novo Nordisk As Verbesserte methode zur herstellung von bestimmten -g(b)-lactam-antibiotika.
CN115385934A (zh) * 2022-10-26 2022-11-25 北京纳百生物科技有限公司 一种舒巴坦半抗原及其合成方法和应用

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IN149747B (no) * 1977-06-07 1982-04-03 Pfizer

Also Published As

Publication number Publication date
AU517074B2 (en) 1981-07-09
GB2125037B (en) 1984-08-01
YU244980A (en) 1983-02-28
ZA805132B (en) 1981-12-30
NO160299B (no) 1988-12-27
LU82795A1 (fr) 1981-04-17
NL185923C (nl) 1990-08-16
GB2059420B (en) 1984-03-14
SU959628A3 (ru) 1982-09-15
DK404980A (da) 1981-03-27
ES495354A0 (es) 1981-08-16
SE461528B (sv) 1990-02-26
PL126949B1 (en) 1983-09-30
GB8319784D0 (en) 1983-08-24
GR70065B (no) 1982-07-26
SE8500965D0 (sv) 1985-02-27
FI840367A0 (fi) 1984-01-30
IE50506B1 (en) 1986-04-30
AT366384B (de) 1982-04-13
KR830003494A (ko) 1983-06-20
NL185923B (nl) 1990-03-16
IT8024920A0 (it) 1980-09-25
GB2125037A (en) 1984-02-29
IL61117A0 (en) 1980-11-30
DE3035995C2 (de) 1985-01-10
NZ195058A (en) 1982-12-07
PT71837A (en) 1980-10-01
KR840000796B1 (ko) 1984-06-12
DD153123A5 (de) 1981-12-23
AU6271380A (en) 1981-04-09
PT71837B (en) 1981-07-09
IE801095L (en) 1981-01-09
MX6580E (es) 1985-07-24
NO802836L (no) 1981-03-27
IN154557B (no) 1984-11-10
HU183212B (en) 1984-04-28
IE50507B1 (en) 1986-04-30
US4256733A (en) 1981-03-17
NO160299C (no) 1989-04-05
SE449865B (sv) 1987-05-25
FR2465736A1 (fr) 1981-03-27
IT1132754B (it) 1986-07-02
FI803028A (fi) 1981-03-27
FI67854B (fi) 1985-02-28
JPS5657788A (en) 1981-05-20
EG14888A (en) 1985-06-30
PH15697A (en) 1983-03-14
PL226868A1 (no) 1981-10-16
NL8005344A (nl) 1981-03-30
BE885389A (fr) 1981-03-25
CA1150242A (en) 1983-07-19
FI67854C (fi) 1985-06-10
NO160370C (no) 1989-04-12
FI67552C (fi) 1985-04-10
FI840367A (fi) 1984-01-30
IL61117A (en) 1983-10-31
JPS6016958B2 (ja) 1985-04-30
CS212284B2 (en) 1982-03-26
IE801998L (en) 1981-03-26
ATA474680A (de) 1981-08-15
GB2059420A (en) 1981-04-23
YU41733B (en) 1987-12-31
ES8106528A1 (es) 1981-08-16
FI67552B (fi) 1984-12-31
FR2465736B1 (no) 1982-04-30
DE3035995A1 (de) 1981-04-02
SE8005714L (sv) 1981-03-27
CH645646A5 (fr) 1984-10-15
AR224547A1 (es) 1981-12-15
NO160370B (no) 1989-01-02

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