FI840367A0 - Vid framstaellning av som mellanprodukter vid terapeutiskt anvaendbara 2 -acetoximetyl-2 -metyl-(5r)-penam-3 -karboxyksyra-1,1-dioxidderivat anvaenbara 2 -acetoxymetyl-2 -metyl-(5r)-penam-3 -karboxylsyraderivat - Google Patents

Vid framstaellning av som mellanprodukter vid terapeutiskt anvaendbara 2 -acetoximetyl-2 -metyl-(5r)-penam-3 -karboxyksyra-1,1-dioxidderivat anvaenbara 2 -acetoxymetyl-2 -metyl-(5r)-penam-3 -karboxylsyraderivat

Info

Publication number
FI840367A0
FI840367A0 FI840367A FI840367A FI840367A0 FI 840367 A0 FI840367 A0 FI 840367A0 FI 840367 A FI840367 A FI 840367A FI 840367 A FI840367 A FI 840367A FI 840367 A0 FI840367 A0 FI 840367A0
Authority
FI
Finland
Prior art keywords
methyl
vid
dioxidderivat
carboxyxyra
anvaenbara
Prior art date
Application number
FI840367A
Other languages
English (en)
Other versions
FI67854C (fi
FI67854B (fi
FI840367A (fi
Inventor
Wayne Ernest Barth
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of FI840367A0 publication Critical patent/FI840367A0/fi
Publication of FI840367A publication Critical patent/FI840367A/fi
Application granted granted Critical
Publication of FI67854B publication Critical patent/FI67854B/fi
Publication of FI67854C publication Critical patent/FI67854C/fi

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D499/21—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring with a nitrogen atom directly attached in position 6 and a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2
    • C07D499/28—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring with a nitrogen atom directly attached in position 6 and a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2 with modified 2-carboxyl group
    • C07D499/32—Esters

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Cephalosporin Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Saccharide Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
FI840367A 1979-09-26 1984-01-30 Som mellanprodukter vid framstaellningen av terapeutiskt anvaendbara 2beta-acetoximetyl-2alfa-metyl-(5r)-penam-3alfa-karboxylsyra-1,1-dioxidderivat anvaendbara 2beta-acetoximetyl-2alfa-metyl-(5r)-penam-3alfa-karboxylsyraderivat FI67854C (fi)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US06/079,127 US4256733A (en) 1979-09-26 1979-09-26 Acetoxymethyl penam compounds as β-lactamase inhibitors
US7912779 1979-09-26
FI803028A FI67552C (fi) 1979-09-26 1980-09-25 Foerfarande foer framstaellning av en ny som beta-laktamas-inhibitor anvaendbar 2beta-acetoxymetyl-2alfa-metyl-(5r)-penam-3alfa-karboxylsyra-1,1-dioxid
FI803028 1980-09-25

Publications (4)

Publication Number Publication Date
FI840367A0 true FI840367A0 (fi) 1984-01-30
FI840367A FI840367A (fi) 1984-01-30
FI67854B FI67854B (fi) 1985-02-28
FI67854C FI67854C (fi) 1985-06-10

Family

ID=22148609

Family Applications (2)

Application Number Title Priority Date Filing Date
FI803028A FI67552C (fi) 1979-09-26 1980-09-25 Foerfarande foer framstaellning av en ny som beta-laktamas-inhibitor anvaendbar 2beta-acetoxymetyl-2alfa-metyl-(5r)-penam-3alfa-karboxylsyra-1,1-dioxid
FI840367A FI67854C (fi) 1979-09-26 1984-01-30 Som mellanprodukter vid framstaellningen av terapeutiskt anvaendbara 2beta-acetoximetyl-2alfa-metyl-(5r)-penam-3alfa-karboxylsyra-1,1-dioxidderivat anvaendbara 2beta-acetoximetyl-2alfa-metyl-(5r)-penam-3alfa-karboxylsyraderivat

Family Applications Before (1)

Application Number Title Priority Date Filing Date
FI803028A FI67552C (fi) 1979-09-26 1980-09-25 Foerfarande foer framstaellning av en ny som beta-laktamas-inhibitor anvaendbar 2beta-acetoxymetyl-2alfa-metyl-(5r)-penam-3alfa-karboxylsyra-1,1-dioxid

Country Status (36)

Country Link
US (1) US4256733A (fi)
JP (1) JPS6016958B2 (fi)
KR (1) KR840000796B1 (fi)
AR (1) AR224547A1 (fi)
AT (1) AT366384B (fi)
AU (1) AU517074B2 (fi)
BE (1) BE885389A (fi)
CA (1) CA1150242A (fi)
CH (1) CH645646A5 (fi)
CS (1) CS212284B2 (fi)
DD (1) DD153123A5 (fi)
DE (1) DE3035995C2 (fi)
DK (1) DK404980A (fi)
EG (1) EG14888A (fi)
ES (1) ES8106528A1 (fi)
FI (2) FI67552C (fi)
FR (1) FR2465736A1 (fi)
GB (2) GB2059420B (fi)
GR (1) GR70065B (fi)
HU (1) HU183212B (fi)
IE (2) IE50506B1 (fi)
IL (1) IL61117A (fi)
IN (1) IN154557B (fi)
IT (1) IT1132754B (fi)
LU (1) LU82795A1 (fi)
MX (1) MX6580E (fi)
NL (1) NL185923C (fi)
NO (2) NO160370C (fi)
NZ (1) NZ195058A (fi)
PH (1) PH15697A (fi)
PL (1) PL126949B1 (fi)
PT (1) PT71837B (fi)
SE (2) SE449865B (fi)
SU (1) SU959628A3 (fi)
YU (1) YU41733B (fi)
ZA (1) ZA805132B (fi)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4364957A (en) * 1979-09-26 1982-12-21 Pfizer Inc. Bis-esters of alkanediols as antibacterial agents
US4511512A (en) * 1980-05-01 1985-04-16 Leo Pharmaceutical Products Ltd. A/S (Lovens Kemiske Produktionsaktiensel skab) Substantially pure dicyclohexyl ammonium 6-β-bromo-penicillanate
US4361513A (en) * 1980-12-11 1982-11-30 Pfizer Inc. Esters of penicillanic acid sulfone
US4474698A (en) * 1980-12-11 1984-10-02 Pfizer Inc. Process for preparing esters of penicillanic acid sulfone
US4558042A (en) * 1981-05-06 1985-12-10 Farmitalia Carlo Erba S.P.A. β-Lactam-containing antibacterial agents and β-lactamase inhibitors
ZA826687B (en) * 1981-09-14 1983-07-27 Pfizer Beta-lactamase inhibiting 2-beta-substituted-2-alpha-methyl 5(r)penam-3-alpha-carboxylic acid 1,1-dioxides and intermediates therefor
JPS58185589A (ja) * 1982-04-23 1983-10-29 Taiho Yakuhin Kogyo Kk ペニシリン誘導体
JPS62198687A (ja) * 1986-02-27 1987-09-02 Taiho Yakuhin Kogyo Kk ２β−置換チオメチルペニシリン誘導体
US4861768A (en) * 1986-02-27 1989-08-29 Taiho Pharmaceutical Company, Limited 2 β-substituted thiomethylpenicillin derivatives and their preparation and use
ES2059285T1 (es) * 1991-12-19 1994-11-16 Novo Nordisk As Un metodo mejorado para la preparacion de ciertos antibioticos beta-lactamicos.
CN115385934A (zh) * 2022-10-26 2022-11-25 北京纳百生物科技有限公司 一种舒巴坦半抗原及其合成方法和应用

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IN149747B (fi) * 1977-06-07 1982-04-03 Pfizer

Also Published As

Publication number Publication date
CA1150242A (en) 1983-07-19
NO160370B (no) 1989-01-02
SE8500965D0 (sv) 1985-02-27
ATA474680A (de) 1981-08-15
SE8005714L (sv) 1981-03-27
HU183212B (en) 1984-04-28
DE3035995C2 (de) 1985-01-10
GR70065B (fi) 1982-07-26
PT71837A (en) 1980-10-01
IE801095L (en) 1981-01-09
ZA805132B (en) 1981-12-30
LU82795A1 (fr) 1981-04-17
IE50506B1 (en) 1986-04-30
SE449865B (sv) 1987-05-25
IT8024920A0 (it) 1980-09-25
IL61117A (en) 1983-10-31
FI803028A (fi) 1981-03-27
DD153123A5 (de) 1981-12-23
FI67854C (fi) 1985-06-10
US4256733A (en) 1981-03-17
BE885389A (fr) 1981-03-25
NL185923B (nl) 1990-03-16
SE461528B (sv) 1990-02-26
NO831082L (no) 1981-03-27
FI67552B (fi) 1984-12-31
DE3035995A1 (de) 1981-04-02
GB2125037A (en) 1984-02-29
CH645646A5 (fr) 1984-10-15
ES495354A0 (es) 1981-08-16
AT366384B (de) 1982-04-13
NO802836L (no) 1981-03-27
PH15697A (en) 1983-03-14
ES8106528A1 (es) 1981-08-16
GB2059420A (en) 1981-04-23
IE50507B1 (en) 1986-04-30
KR830003494A (ko) 1983-06-20
PL126949B1 (en) 1983-09-30
FI67854B (fi) 1985-02-28
NL185923C (nl) 1990-08-16
NO160299B (no) 1988-12-27
JPS6016958B2 (ja) 1985-04-30
PT71837B (en) 1981-07-09
NZ195058A (en) 1982-12-07
SU959628A3 (ru) 1982-09-15
YU41733B (en) 1987-12-31
JPS5657788A (en) 1981-05-20
YU244980A (en) 1983-02-28
PL226868A1 (fi) 1981-10-16
NO160370C (no) 1989-04-12
AU6271380A (en) 1981-04-09
GB2125037B (en) 1984-08-01
EG14888A (en) 1985-06-30
FR2465736B1 (fi) 1982-04-30
AR224547A1 (es) 1981-12-15
NO160299C (no) 1989-04-05
IE801998L (en) 1981-03-26
AU517074B2 (en) 1981-07-09
FR2465736A1 (fr) 1981-03-27
IT1132754B (it) 1986-07-02
CS212284B2 (en) 1982-03-26
IL61117A0 (en) 1980-11-30
DK404980A (da) 1981-03-27
FI840367A (fi) 1984-01-30
KR840000796B1 (ko) 1984-06-12
GB8319784D0 (en) 1983-08-24
IN154557B (fi) 1984-11-10
FI67552C (fi) 1985-04-10
GB2059420B (en) 1984-03-14
NL8005344A (nl) 1981-03-30
MX6580E (es) 1985-07-24

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Legal Events

Date Code Title Description
MM Patent lapsed

Owner name: PFIZER INC.