AR224547A1 - Compuestos de 2-beta-acetoximetil-2-alfa-metil(5r)penam desprovistos de actividad terapeutica,y utiles,como intermediarios para la preparacion de inhibidores de beta-lactamasa,y procedimiento para preparar a dichos inhibidores partiendo del citado intermediario - Google Patents
Compuestos de 2-beta-acetoximetil-2-alfa-metil(5r)penam desprovistos de actividad terapeutica,y utiles,como intermediarios para la preparacion de inhibidores de beta-lactamasa,y procedimiento para preparar a dichos inhibidores partiendo del citado intermediarioInfo
- Publication number
- AR224547A1 AR224547A1 AR282629A AR28262980A AR224547A1 AR 224547 A1 AR224547 A1 AR 224547A1 AR 282629 A AR282629 A AR 282629A AR 28262980 A AR28262980 A AR 28262980A AR 224547 A1 AR224547 A1 AR 224547A1
- Authority
- AR
- Argentina
- Prior art keywords
- beta
- inhidents
- inhidated
- acetoximetil
- penam
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
- C07D499/21—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring with a nitrogen atom directly attached in position 6 and a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2
- C07D499/28—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring with a nitrogen atom directly attached in position 6 and a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2 with modified 2-carboxyl group
- C07D499/32—Esters
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Communicable Diseases (AREA)
- Oncology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Cephalosporin Compounds (AREA)
- Preparation Of Compounds By Using Micro-Organisms (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Saccharide Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US06/079,127 US4256733A (en) | 1979-09-26 | 1979-09-26 | Acetoxymethyl penam compounds as β-lactamase inhibitors |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| AR224547A1 true AR224547A1 (es) | 1981-12-15 |
Family
ID=22148609
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AR282629A AR224547A1 (es) | 1979-09-26 | 1980-09-24 | Compuestos de 2-beta-acetoximetil-2-alfa-metil(5r)penam desprovistos de actividad terapeutica,y utiles,como intermediarios para la preparacion de inhibidores de beta-lactamasa,y procedimiento para preparar a dichos inhibidores partiendo del citado intermediario |
Country Status (36)
| Country | Link |
|---|---|
| US (1) | US4256733A (es) |
| JP (1) | JPS6016958B2 (es) |
| KR (1) | KR840000796B1 (es) |
| AR (1) | AR224547A1 (es) |
| AT (1) | AT366384B (es) |
| AU (1) | AU517074B2 (es) |
| BE (1) | BE885389A (es) |
| CA (1) | CA1150242A (es) |
| CH (1) | CH645646A5 (es) |
| CS (1) | CS212284B2 (es) |
| DD (1) | DD153123A5 (es) |
| DE (1) | DE3035995C2 (es) |
| DK (1) | DK404980A (es) |
| EG (1) | EG14888A (es) |
| ES (1) | ES8106528A1 (es) |
| FI (2) | FI67552C (es) |
| FR (1) | FR2465736A1 (es) |
| GB (2) | GB2059420B (es) |
| GR (1) | GR70065B (es) |
| HU (1) | HU183212B (es) |
| IE (2) | IE50507B1 (es) |
| IL (1) | IL61117A (es) |
| IN (1) | IN154557B (es) |
| IT (1) | IT1132754B (es) |
| LU (1) | LU82795A1 (es) |
| MX (1) | MX6580E (es) |
| NL (1) | NL185923C (es) |
| NO (2) | NO160370C (es) |
| NZ (1) | NZ195058A (es) |
| PH (1) | PH15697A (es) |
| PL (1) | PL126949B1 (es) |
| PT (1) | PT71837B (es) |
| SE (2) | SE449865B (es) |
| SU (1) | SU959628A3 (es) |
| YU (1) | YU41733B (es) |
| ZA (1) | ZA805132B (es) |
Families Citing this family (11)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4364957A (en) * | 1979-09-26 | 1982-12-21 | Pfizer Inc. | Bis-esters of alkanediols as antibacterial agents |
| US4511512A (en) * | 1980-05-01 | 1985-04-16 | Leo Pharmaceutical Products Ltd. A/S (Lovens Kemiske Produktionsaktiensel skab) | Substantially pure dicyclohexyl ammonium 6-β-bromo-penicillanate |
| US4361513A (en) * | 1980-12-11 | 1982-11-30 | Pfizer Inc. | Esters of penicillanic acid sulfone |
| US4474698A (en) * | 1980-12-11 | 1984-10-02 | Pfizer Inc. | Process for preparing esters of penicillanic acid sulfone |
| US4558042A (en) * | 1981-05-06 | 1985-12-10 | Farmitalia Carlo Erba S.P.A. | β-Lactam-containing antibacterial agents and β-lactamase inhibitors |
| ZA826687B (en) * | 1981-09-14 | 1983-07-27 | Pfizer | Beta-lactamase inhibiting 2-beta-substituted-2-alpha-methyl 5(r)penam-3-alpha-carboxylic acid 1,1-dioxides and intermediates therefor |
| JPS58185589A (ja) * | 1982-04-23 | 1983-10-29 | Taiho Yakuhin Kogyo Kk | ペニシリン誘導体 |
| JPS62198687A (ja) * | 1986-02-27 | 1987-09-02 | Taiho Yakuhin Kogyo Kk | ２β−置換チオメチルペニシリン誘導体 |
| US4861768A (en) * | 1986-02-27 | 1989-08-29 | Taiho Pharmaceutical Company, Limited | 2 β-substituted thiomethylpenicillin derivatives and their preparation and use |
| SK63894A3 (en) * | 1991-12-19 | 1995-03-08 | Novo Nordisk As | Method of preparation of beta-lactam antibiotic |
| CN115385934A (zh) * | 2022-10-26 | 2022-11-25 | 北京纳百生物科技有限公司 | 一种舒巴坦半抗原及其合成方法和应用 |
Family Cites Families (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| IN149747B (es) * | 1977-06-07 | 1982-04-03 | Pfizer |
-
1979
- 1979-09-26 US US06/079,127 patent/US4256733A/en not_active Expired - Lifetime
-
1980
- 1980-08-13 SE SE8005714A patent/SE449865B/sv not_active IP Right Cessation
- 1980-08-20 ZA ZA00805132A patent/ZA805132B/xx unknown
- 1980-08-20 IN IN607/DEL/80A patent/IN154557B/en unknown
- 1980-09-19 SU SU802983144A patent/SU959628A3/ru active
- 1980-09-19 HU HU802310A patent/HU183212B/hu unknown
- 1980-09-22 PL PL1980226868A patent/PL126949B1/pl unknown
- 1980-09-22 CS CS806403A patent/CS212284B2/cs unknown
- 1980-09-23 AT AT0474680A patent/AT366384B/de not_active IP Right Cessation
- 1980-09-23 GB GB8030639A patent/GB2059420B/en not_active Expired
- 1980-09-23 EG EG584/80A patent/EG14888A/xx active
- 1980-09-23 GR GR62939A patent/GR70065B/el unknown
- 1980-09-23 CA CA000360886A patent/CA1150242A/en not_active Expired
- 1980-09-23 IL IL61117A patent/IL61117A/xx unknown
- 1980-09-24 PH PH24617A patent/PH15697A/en unknown
- 1980-09-24 LU LU82795A patent/LU82795A1/fr unknown
- 1980-09-24 DE DE3035995A patent/DE3035995C2/de not_active Expired
- 1980-09-24 KR KR1019800003721A patent/KR840000796B1/ko active
- 1980-09-24 AR AR282629A patent/AR224547A1/es active
- 1980-09-24 MX MX809044U patent/MX6580E/es unknown
- 1980-09-25 IT IT24920/80A patent/IT1132754B/it active
- 1980-09-25 FI FI803028A patent/FI67552C/fi not_active IP Right Cessation
- 1980-09-25 NO NO802836A patent/NO160370C/no unknown
- 1980-09-25 IE IE1095/85A patent/IE50507B1/en unknown
- 1980-09-25 NZ NZ195058A patent/NZ195058A/xx unknown
- 1980-09-25 PT PT71837A patent/PT71837B/pt unknown
- 1980-09-25 ES ES495354A patent/ES8106528A1/es not_active Expired
- 1980-09-25 FR FR8020618A patent/FR2465736A1/fr active Granted
- 1980-09-25 CH CH719980A patent/CH645646A5/fr not_active IP Right Cessation
- 1980-09-25 DD DD80224128A patent/DD153123A5/de unknown
- 1980-09-25 AU AU62713/80A patent/AU517074B2/en not_active Ceased
- 1980-09-25 BE BE0/202222A patent/BE885389A/fr not_active IP Right Cessation
- 1980-09-25 YU YU2449/80A patent/YU41733B/xx unknown
- 1980-09-25 IE IE1998/80A patent/IE50506B1/en not_active IP Right Cessation
- 1980-09-25 JP JP55133639A patent/JPS6016958B2/ja not_active Expired
- 1980-09-25 NL NLAANVRAGE8005344,A patent/NL185923C/xx not_active IP Right Cessation
- 1980-09-25 DK DK404980A patent/DK404980A/da not_active Application Discontinuation
-
1983
- 1983-03-25 NO NO83831082A patent/NO160299C/no unknown
- 1983-07-22 GB GB08319784A patent/GB2125037B/en not_active Expired
-
1984
- 1984-01-30 FI FI840367A patent/FI67854C/fi not_active IP Right Cessation
-
1985
- 1985-02-27 SE SE8500965A patent/SE461528B/sv not_active IP Right Cessation
Also Published As
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| IT7820811A0 (it) | Fenossi-benzil-ossicarbonil-derivati sostituiti, procedimento per laloro preparazione e loro impiegocome insetticidi e come acaricidi. | |
| IT7820169A0 (it) | Procedimento per la fabbricazione di etilbenzene. | |
| IT7825315A0 (it) | Fenossi-benzil-ossicarbonilderivati sostituiti, procedimento per la loro preparazione e loro impiego come insetticidi e come acaricidi. | |
| NL190554C (nl) | Cefalosporinederivaat, en farmaceutisch of veterinair preparaat met antibacteriële werking, dat dit cefalosporinederivaat bevat. | |
| NL183358C (nl) | Farmaceutisch preparaat, en daarin te gebruiken penicillaanzuur-derivaat met beta-lactamase-remmende werking. | |
| NO156787C (no) | Analogifremgangsmaate for fremstilling av terapeutisk aktive kinolonderivater. | |
| IT7828141A0 (it) | Triazolil-o,n-acetali diastereomeri, procedimento per laloro preparazione ed il loro impiego come fungicidi. | |
| NO162561C (no) | Fremgangsmaate for fremstilling av oksazolinforbindelser egnet for fremstilling av antibakterielt virksomme 1-oksa-detiacefalosporiner. | |
| AR224547A1 (es) | Compuestos de 2-beta-acetoximetil-2-alfa-metil(5r)penam desprovistos de actividad terapeutica,y utiles,como intermediarios para la preparacion de inhibidores de beta-lactamasa,y procedimiento para preparar a dichos inhibidores partiendo del citado intermediario | |
| NO820290L (no) | Mellomprodukter for fremstilling av terapeutisk aktive antrakinon-derivater. | |
| NO155548C (no) | Fremgangsmaate til fremstilling av optisk aktive cefalosporin-analoger. | |
| ES513111A0 (es) | Procedimiento para la obtencion de benzoil-(tio)ureas sustituidas, de efecto pesticida. | |
| IT8022944A0 (it) | Composti della cefalosporina, procedimenti per la loro preparazione, e farmaci antibatterici contenenti glistessi. | |
| ES508222A0 (es) | "procedimiento, para preparar deca-, undeca- y tridecapeptidos con actividad timica". | |
| IT7819009A0 (it) | Fenil-carbammoil-2-pirazoline sostituite, procedimento per laloro preparazione e loro impiegocome insetticidi. | |
| NO157505C (no) | Analogifremgangsmaate for fremstilling av organiske selenforbindelser med antineoplastisk aktivitet. | |
| TR19208A (tr) | 1-azolil-4-hidroksi-butan tuerevleri,bunlarin hazirlanisina ait usul ve bunlarin fungisidler ve bakteriler olarak kullanilmalari | |
| ES500038A0 (es) | Un procedimiento para la preparacion de un derivado de 3-o- desmetilsannamicina c o del antibiotico ax-127b-1. | |
| NO152843C (no) | Analogifremgangsmaate for fremstilling av terapeutisk aktive pyrimidopyrimidiner. | |
| RO75739A (ro) | Procedeu pentru prepararea unor carbamoil triazolil-o,n-acetali | |
| NO147108C (no) | Analogifremgangsmaate for fremstilling av terapeutisk virksomme 1-amino-lavere-alkyl-3,4-difenyl-1h-pyrazoler | |
| NO154131C (no) | Analogifremgangsmaate for fremstilling av terapeutisk aktive karbostyrilderivater. | |
| IT8019609A0 (it) | Procedimento per la preparazione di composti beta-lattamici. | |
| NO154635C (no) | Fremgangsmaate for fremstilling av terapeutisk aktive ergotalkaloider. | |
| IT7825712A0 (it) | Composti di b-lattami, procedimento per la loro preparazione e loro impiego. |