NO331689B1 - Oral farmasoytisk sammensetning omfattende rivastigmin, samt anvendelse av rivastigmin - Google Patents
Oral farmasoytisk sammensetning omfattende rivastigmin, samt anvendelse av rivastigmin Download PDFInfo
- Publication number
- NO331689B1 NO331689B1 NO20011471A NO20011471A NO331689B1 NO 331689 B1 NO331689 B1 NO 331689B1 NO 20011471 A NO20011471 A NO 20011471A NO 20011471 A NO20011471 A NO 20011471A NO 331689 B1 NO331689 B1 NO 331689B1
- Authority
- NO
- Norway
- Prior art keywords
- rivastigmine
- composition
- pharmaceutical composition
- cellulose
- water
- Prior art date
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- 239000008203 oral pharmaceutical composition Substances 0.000 title claims description 7
- XSVMFMHYUFZWBK-NSHDSACASA-N Rivastigmine Chemical compound CCN(C)C(=O)OC1=CC=CC([C@H](C)N(C)C)=C1 XSVMFMHYUFZWBK-NSHDSACASA-N 0.000 claims abstract description 53
- 229960004136 rivastigmine Drugs 0.000 claims abstract description 50
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Classifications
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- A—HUMAN NECESSITIES
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- A—HUMAN NECESSITIES
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- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
- A61K9/5084—Mixtures of one or more drugs in different galenical forms, at least one of which being granules, microcapsules or (coated) microparticles according to A61K9/16 or A61K9/50, e.g. for obtaining a specific release pattern or for combining different drugs
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/21—Esters, e.g. nitroglycerine, selenocyanates
- A61K31/27—Esters, e.g. nitroglycerine, selenocyanates of carbamic or thiocarbamic acids, meprobamate, carbachol, neostigmine
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- A—HUMAN NECESSITIES
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- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2072—Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
- A61K9/2077—Tablets comprising drug-containing microparticles in a substantial amount of supporting matrix; Multiparticulate tablets
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
- A61K9/5073—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings
- A61K9/5078—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings with drug-free core
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
- A61K9/2806—Coating materials
- A61K9/2833—Organic macromolecular compounds
- A61K9/286—Polysaccharides, e.g. gums; Cyclodextrin
- A61K9/2866—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
- A61K9/2886—Dragees; Coated pills or tablets, e.g. with film or compression coating having two or more different drug-free coatings; Tablets of the type inert core-drug layer-inactive layer
Applications Claiming Priority (7)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GBGB9821298.8A GB9821298D0 (en) | 1998-10-01 | 1998-10-01 | Organic compoundsq |
| GBGB9821299.6A GB9821299D0 (en) | 1998-10-01 | 1998-10-01 | Organic compounds |
| GBGB9826654.7A GB9826654D0 (en) | 1998-12-03 | 1998-12-03 | Organic compounds |
| GBGB9827624.9A GB9827624D0 (en) | 1998-12-16 | 1998-12-16 | Organic compounds |
| GBGB9907822.2A GB9907822D0 (en) | 1999-04-06 | 1999-04-06 | Organic compounds |
| GBGB9907823.0A GB9907823D0 (en) | 1999-04-06 | 1999-04-06 | Organic compounds |
| PCT/EP1999/007298 WO2000019985A2 (fr) | 1998-10-01 | 1999-10-01 | Nouvelles formulations administrees par voie orale et a liberation prolongee |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| NO20011471L NO20011471L (no) | 2001-03-22 |
| NO20011471D0 NO20011471D0 (no) | 2001-03-22 |
| NO331689B1 true NO331689B1 (no) | 2012-02-27 |
Family
ID=27547321
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| Application Number | Title | Priority Date | Filing Date |
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| NO20011471A NO331689B1 (no) | 1998-10-01 | 2001-03-22 | Oral farmasoytisk sammensetning omfattende rivastigmin, samt anvendelse av rivastigmin |
Country Status (23)
| Country | Link |
|---|---|
| US (5) | US20010033866A1 (fr) |
| EP (1) | EP1121104B1 (fr) |
| JP (1) | JP4012689B2 (fr) |
| KR (1) | KR100603900B1 (fr) |
| CN (1) | CN1406126A (fr) |
| AT (1) | ATE286725T1 (fr) |
| AU (1) | AU764866B2 (fr) |
| BR (1) | BR9914251A (fr) |
| CA (1) | CA2342340C (fr) |
| CZ (1) | CZ302888B6 (fr) |
| DE (1) | DE69923200T2 (fr) |
| ES (1) | ES2237163T3 (fr) |
| HK (1) | HK1052473A1 (fr) |
| HU (1) | HUP0103883A3 (fr) |
| ID (1) | ID27504A (fr) |
| IL (2) | IL141762A0 (fr) |
| NO (1) | NO331689B1 (fr) |
| NZ (1) | NZ510683A (fr) |
| PL (1) | PL196945B1 (fr) |
| PT (1) | PT1121104E (fr) |
| SK (1) | SK285250B6 (fr) |
| TR (1) | TR200100931T2 (fr) |
| WO (1) | WO2000019985A2 (fr) |
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| WO2001013898A2 (fr) * | 1999-08-26 | 2001-03-01 | Elan Corporation, Plc. | Compositions pharmaceutiques |
| GB9923045D0 (en) * | 1999-09-29 | 1999-12-01 | Novartis Ag | New oral formulations |
| NZ524641A (en) * | 2000-09-29 | 2004-09-24 | Solvay Pharmaceuticals B | A pharmaceutical hydrophilic gel forming matrix formulation having prolonged release which is ion strength independent |
| JP5023412B2 (ja) * | 2001-05-09 | 2012-09-12 | 吉澤石灰工業株式会社 | ホルムアルデヒド廃液の処理剤 |
| JP2005525299A (ja) * | 2001-09-14 | 2005-08-25 | スコラー インコーポレイテッド | アミノ酸調節性の長期放出投薬形態 |
| DE60223695T2 (de) * | 2001-09-14 | 2008-10-30 | Scolr, Inc., Redmond | Aminosäure-modulierte dosierform mit verlängerter freisetzung |
| KR100453288B1 (ko) * | 2002-03-12 | 2004-10-21 | 한국화학연구원 | 약물의 제어 방출을 위한 스퀴즈-유형의 삼투성 약물 전달장치 |
| PT1529116E (pt) * | 2002-08-07 | 2009-09-10 | Novartis Ag | Métodos para o tratamento da demência com base no genótipo da apo e |
| AU2003100262B4 (en) * | 2003-04-07 | 2003-09-18 | Jurox Pty Ltd | Stable carprofen composition |
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| ATE454138T1 (de) * | 2003-08-08 | 2010-01-15 | Biovail Lab Int Srl | Tablette mit modifizierter freisetzung von bupropion hydrochlorid |
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| WO2006123357A2 (fr) * | 2005-02-22 | 2006-11-23 | Sun Pharmaceutical Industries Limited | Composition pharmaceutique |
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| GB0525461D0 (en) | 2005-12-15 | 2006-01-25 | Archimedes Dev Ltd | Pharmaceutical compositions |
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| ITMI20071502A1 (it) * | 2007-07-25 | 2009-01-26 | Archimica Srl | Procedimento per la preparazione di formulazioni solide a rilascio controllato contenenti oxcarbazepina e formulazioni ottenibili con tale procedimento |
| WO2009022345A1 (fr) * | 2007-08-14 | 2009-02-19 | Yissum Research Development Company Of The Hebrew University Of Jerusalem | Carbamates de phényle destinés au traitement de la sclérose en plaques |
| LT2187742T (lt) | 2007-08-23 | 2018-01-10 | Theracos Sub, Llc | (2s,3r,4r,5s,6r)-2-(4-chlor-3-benzilfenil)-6-(hidroksimetil)tetrahidro-2h-piran-3,4,5-triolio dariniai, skirti panaudoti diabeto gydymui |
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| BRPI0916769A2 (pt) | 2008-07-15 | 2017-09-26 | Theracos Inc | derivados de benzilbenzeno deuterados e métodos de uso |
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| BR112015009004A8 (pt) | 2012-12-21 | 2021-07-20 | Eisai R&D Man Co Ltd | forma amorfa de derivado de quinolina e método de produção da mesma |
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| CN113398273B (zh) * | 2021-05-14 | 2022-07-19 | 广西壮族自治区中国科学院广西植物研究所 | 木聚糖衍生物作为亲水性缓释材料在制备药物缓释片中的应用 |
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| US4014335A (en) * | 1975-04-21 | 1977-03-29 | Alza Corporation | Ocular drug delivery device |
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| US5472710A (en) * | 1988-04-16 | 1995-12-05 | Schwarz Pharma Ag | Pharmaceutical preparation to be administered orally with controlled release of active substance and method for its manufacture |
| DE3922167A1 (de) * | 1988-04-16 | 1991-01-17 | Sanol Arznei Schwarz Gmbh | Oral zu verabreichende diltiazemhydrochlorid enthaltende pharmazeutische zubereitung zur einmal taeglichen applikation und verfahren zu deren herstellung |
| US5262173A (en) * | 1992-03-02 | 1993-11-16 | American Cyanamid Company | Pulsatile once-a-day delivery systems for minocycline |
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| PT621032E (pt) * | 1993-04-23 | 2001-01-31 | Novartis Ag | Dispositivo de distribuicao de libertacao controlada de farmaco |
| US5698224A (en) * | 1994-06-27 | 1997-12-16 | Alza Corporation | Tacrine therapy |
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| CN1158071C (zh) * | 1997-05-30 | 2004-07-21 | 渗透有限公司 | 多层渗透装置 |
| GB9800526D0 (en) * | 1998-01-12 | 1998-03-11 | Ciba Geigy Ag | Organic compounds |
| IL141762A0 (en) | 1998-10-01 | 2002-03-10 | Novartis Ag | New oral formulations |
| US6534541B1 (en) | 1999-10-19 | 2003-03-18 | Novartis Ag | Treatment of ocular disorders |
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1999
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- 1999-10-01 BR BR9914251-1A patent/BR9914251A/pt not_active Application Discontinuation
- 1999-10-01 WO PCT/EP1999/007298 patent/WO2000019985A2/fr not_active Application Discontinuation
- 1999-10-01 PT PT99950595T patent/PT1121104E/pt unknown
- 1999-10-01 HU HU0103883A patent/HUP0103883A3/hu unknown
- 1999-10-01 ID IDW20010671A patent/ID27504A/id unknown
- 1999-10-01 CA CA002342340A patent/CA2342340C/fr not_active Expired - Fee Related
- 1999-10-01 TR TR2001/00931T patent/TR200100931T2/xx unknown
- 1999-10-01 PL PL348734A patent/PL196945B1/pl not_active IP Right Cessation
- 1999-10-01 DE DE69923200T patent/DE69923200T2/de not_active Expired - Lifetime
- 1999-10-01 EP EP99950595A patent/EP1121104B1/fr not_active Expired - Lifetime
- 1999-10-01 NZ NZ510683A patent/NZ510683A/en not_active IP Right Cessation
- 1999-10-01 CN CN99811633A patent/CN1406126A/zh active Pending
- 1999-10-01 KR KR1020017003384A patent/KR100603900B1/ko not_active IP Right Cessation
- 1999-10-01 ES ES99950595T patent/ES2237163T3/es not_active Expired - Lifetime
- 1999-10-01 AT AT99950595T patent/ATE286725T1/de active
- 1999-10-01 JP JP2000573347A patent/JP4012689B2/ja not_active Expired - Fee Related
- 1999-10-01 CZ CZ20011155A patent/CZ302888B6/cs not_active IP Right Cessation
- 1999-10-01 SK SK439-2001A patent/SK285250B6/sk not_active IP Right Cessation
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2001
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- 2001-03-22 NO NO20011471A patent/NO331689B1/no not_active IP Right Cessation
- 2001-03-27 US US09/818,690 patent/US20010033866A1/en not_active Abandoned
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2002
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2003
- 2003-03-31 US US10/403,146 patent/US20030203025A1/en not_active Abandoned
- 2003-07-09 HK HK03104925.9A patent/HK1052473A1/zh unknown
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2005
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2006
- 2006-11-03 US US11/592,853 patent/US20070053982A1/en not_active Abandoned
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