NO328682B1 - Adamtanderivater, fremgangsmate til fremstilling derav, og anvendelse derav i terapi, samt en farmasoytisk blanding inneholdende slike derivater - Google Patents

Adamtanderivater, fremgangsmate til fremstilling derav, og anvendelse derav i terapi, samt en farmasoytisk blanding inneholdende slike derivater Download PDF

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Publication number
NO328682B1
NO328682B1 NO20022856A NO20022856A NO328682B1 NO 328682 B1 NO328682 B1 NO 328682B1 NO 20022856 A NO20022856 A NO 20022856A NO 20022856 A NO20022856 A NO 20022856A NO 328682 B1 NO328682 B1 NO 328682B1
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NO
Norway
Prior art keywords
dec
chloro
ylmethyl
benzamide
tricyclo
Prior art date
Application number
NO20022856A
Other languages
English (en)
Norwegian (no)
Other versions
NO20022856D0 (no
NO20022856L (no
Inventor
Phillip Thorne
Mark Furber
Paul Andrew Willis
Michael Paul Mortimore
Lilian Alcaraz
Timothy Jon Luker
Moya Caffrey
Austen David Pimm
Original Assignee
Astrazeneca Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from SE9904651A external-priority patent/SE9904651D0/xx
Priority claimed from GB0015744A external-priority patent/GB0015744D0/en
Priority claimed from GB0017942A external-priority patent/GB0017942D0/en
Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab
Publication of NO20022856D0 publication Critical patent/NO20022856D0/no
Publication of NO20022856L publication Critical patent/NO20022856L/no
Publication of NO328682B1 publication Critical patent/NO328682B1/no

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    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C235/00—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms
    • C07C235/42—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings and singly-bound oxygen atoms bound to the same carbon skeleton
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C235/00—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms
    • C07C235/42—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings and singly-bound oxygen atoms bound to the same carbon skeleton
    • C07C235/44—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings and singly-bound oxygen atoms bound to the same carbon skeleton with carbon atoms of carboxamide groups and singly-bound oxygen atoms bound to carbon atoms of the same non-condensed six-membered aromatic ring
    • C07C235/46—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms having carbon atoms of carboxamide groups bound to carbon atoms of six-membered aromatic rings and singly-bound oxygen atoms bound to the same carbon skeleton with carbon atoms of carboxamide groups and singly-bound oxygen atoms bound to carbon atoms of the same non-condensed six-membered aromatic ring having the nitrogen atoms of the carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms
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    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C235/00—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms
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    • C07C235/84—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms having carbon atoms of carboxamide groups and doubly-bound oxygen atoms bound to the same carbon skeleton with the carbon atom of at least one of the carboxamide groups bound to a carbon atom of a six-membered aromatic ring
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    • C07C323/23—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and nitrogen atoms, not being part of nitro or nitroso groups, bound to the same carbon skeleton
    • C07C323/24—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and nitrogen atoms, not being part of nitro or nitroso groups, bound to the same carbon skeleton having the sulfur atoms of the thio groups bound to acyclic carbon atoms of the carbon skeleton
    • C07C323/25—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and nitrogen atoms, not being part of nitro or nitroso groups, bound to the same carbon skeleton having the sulfur atoms of the thio groups bound to acyclic carbon atoms of the carbon skeleton the carbon skeleton being acyclic and saturated
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    • C07D233/56—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
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    • C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/56—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
    • C07D233/61—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms with hydrocarbon radicals, substituted by nitrogen atoms not forming part of a nitro radical, attached to ring nitrogen atoms
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    • C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/64—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with substituted hydrocarbon radicals attached to ring carbon atoms, e.g. histidine
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    • C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
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    • C07C2603/74—Adamantanes

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  • Health & Medical Sciences (AREA)
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  • Diabetes (AREA)
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  • Orthopedic Medicine & Surgery (AREA)
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  • Oncology (AREA)
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NO20022856A 1999-12-17 2002-06-14 Adamtanderivater, fremgangsmate til fremstilling derav, og anvendelse derav i terapi, samt en farmasoytisk blanding inneholdende slike derivater NO328682B1 (no)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
SE9904651A SE9904651D0 (sv) 1999-12-17 1999-12-17 Novel compounds
GB0015744A GB0015744D0 (en) 2000-06-27 2000-06-27 Novel compounds
GB0017942A GB0017942D0 (en) 2000-07-22 2000-07-22 Novel compounds
PCT/SE2000/002505 WO2001044170A1 (en) 1999-12-17 2000-12-12 Adamantane derivatives

Publications (3)

Publication Number Publication Date
NO20022856D0 NO20022856D0 (no) 2002-06-14
NO20022856L NO20022856L (no) 2002-08-16
NO328682B1 true NO328682B1 (no) 2010-04-26

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NO20022856A NO328682B1 (no) 1999-12-17 2002-06-14 Adamtanderivater, fremgangsmate til fremstilling derav, og anvendelse derav i terapi, samt en farmasoytisk blanding inneholdende slike derivater

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US (5) US6881754B2 (pl)
EP (5) EP1242364B1 (pl)
JP (2) JP3710418B2 (pl)
KR (2) KR20070012883A (pl)
CN (1) CN1312120C (pl)
AR (1) AR035325A1 (pl)
AT (4) ATE376994T1 (pl)
AU (2) AU780506B2 (pl)
BR (1) BRPI0016395B8 (pl)
CA (1) CA2393352C (pl)
CO (1) CO5251381A1 (pl)
CY (3) CY1106357T1 (pl)
CZ (1) CZ20022093A3 (pl)
DE (4) DE60034155T2 (pl)
DK (4) DK1352897T3 (pl)
EE (1) EE05134B1 (pl)
ES (4) ES2282546T3 (pl)
HK (2) HK1057035A1 (pl)
HU (1) HUP0300616A3 (pl)
IL (2) IL150124A0 (pl)
IS (1) IS2246B (pl)
MX (1) MXPA02005789A (pl)
MY (1) MY125978A (pl)
NO (1) NO328682B1 (pl)
NZ (1) NZ519378A (pl)
PL (1) PL200836B1 (pl)
PT (4) PT1352897E (pl)
SI (1) SI1352895T1 (pl)
SK (1) SK286987B6 (pl)
TR (1) TR200401432T4 (pl)
TW (1) TWI258462B (pl)
WO (1) WO2001044170A1 (pl)

Families Citing this family (43)

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Publication number Priority date Publication date Assignee Title
SE9904505D0 (sv) 1999-12-09 1999-12-09 Astra Pharma Prod Novel compounds
TWI258462B (en) * 1999-12-17 2006-07-21 Astrazeneca Ab Adamantane derivative compounds, process for preparing the same and pharmaceutical composition comprising the same
SE9904738D0 (sv) 1999-12-22 1999-12-22 Astra Pharma Prod Novel compounds
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