NO323608B1 - Aryl-fusjonerte azapolysykliske forbindelser, anvendelse derav og farmasoytisk sammensetning. - Google Patents
Aryl-fusjonerte azapolysykliske forbindelser, anvendelse derav og farmasoytisk sammensetning. Download PDFInfo
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- NO323608B1 NO323608B1 NO20024042A NO20024042A NO323608B1 NO 323608 B1 NO323608 B1 NO 323608B1 NO 20024042 A NO20024042 A NO 20024042A NO 20024042 A NO20024042 A NO 20024042A NO 323608 B1 NO323608 B1 NO 323608B1
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- dodeca
- triene
- aza
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- C07D221/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00
- C07D221/02—Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00 condensed with carbocyclic rings or ring systems
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- C07D221/02—Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00 condensed with carbocyclic rings or ring systems
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- C07D221/24—Camphidines
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- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
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- C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
- C07D233/56—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
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- C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
- C07D249/08—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
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- C—CHEMISTRY; METALLURGY
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- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
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- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
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Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US09/514,002 US6605610B1 (en) | 1997-12-31 | 2000-02-25 | Aryl fused azapolycyclic compounds |
PCT/IB2001/000153 WO2001062736A1 (en) | 2000-02-25 | 2001-02-08 | Aryl fused azapolycyclic compounds |
Publications (3)
Publication Number | Publication Date |
---|---|
NO20024042D0 NO20024042D0 (no) | 2002-08-23 |
NO20024042L NO20024042L (no) | 2002-10-17 |
NO323608B1 true NO323608B1 (no) | 2007-06-18 |
Family
ID=24045406
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
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NO20024042A NO323608B1 (no) | 2000-02-25 | 2002-08-23 | Aryl-fusjonerte azapolysykliske forbindelser, anvendelse derav og farmasoytisk sammensetning. |
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Country | Link |
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US (3) | US6605610B1 (ja) |
EP (2) | EP1619192B1 (ja) |
JP (1) | JP2003524002A (ja) |
KR (1) | KR100537976B1 (ja) |
CN (1) | CN1263745C (ja) |
AP (1) | AP1860A (ja) |
AT (2) | ATE453643T1 (ja) |
AU (2) | AU784081B2 (ja) |
BG (1) | BG65891B1 (ja) |
BR (1) | BR0108610A (ja) |
CA (1) | CA2401229C (ja) |
CR (1) | CR6726A (ja) |
CU (1) | CU23148A3 (ja) |
CY (1) | CY1105301T1 (ja) |
CZ (1) | CZ303203B6 (ja) |
DE (2) | DE60120366T2 (ja) |
DK (2) | DK1259489T3 (ja) |
DZ (1) | DZ3328A1 (ja) |
EA (1) | EA005316B1 (ja) |
EE (1) | EE200200475A (ja) |
ES (2) | ES2336800T3 (ja) |
GE (1) | GEP20053454B (ja) |
HK (1) | HK1050894A1 (ja) |
HR (1) | HRP20020700A2 (ja) |
HU (1) | HU229482B1 (ja) |
IL (2) | IL150639A0 (ja) |
IS (1) | IS2293B (ja) |
MA (1) | MA26875A1 (ja) |
MX (1) | MXPA02008311A (ja) |
NO (1) | NO323608B1 (ja) |
NZ (1) | NZ519973A (ja) |
OA (1) | OA12181A (ja) |
PL (1) | PL365163A1 (ja) |
PT (1) | PT1259489E (ja) |
RS (1) | RS51123B (ja) |
SI (1) | SI1259489T1 (ja) |
SK (1) | SK12042002A3 (ja) |
UA (1) | UA74813C2 (ja) |
WO (1) | WO2001062736A1 (ja) |
ZA (1) | ZA200206768B (ja) |
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AU2002365314A1 (en) * | 2001-11-30 | 2003-06-10 | Pfizer Products Inc. | Aryl fused azapolycyclic compounds |
BR0312297A (pt) | 2002-07-18 | 2005-04-12 | Cytos Biotechnology Ag | Conjugados veìculos de hapteno e seu uso |
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RU2284319C2 (ru) * | 2002-11-25 | 2006-09-27 | Пфайзер Продактс Инк. | Усовершенствованный способ получения 1,3-замещенных инденов |
MXPA05007565A (es) * | 2003-01-15 | 2005-09-21 | Pfizer Prod Inc | Procedimiento mejorado de preparacion de lactamas policiclicas fusionadas con arilos. |
BRPI0410219A (pt) * | 2003-05-20 | 2006-05-09 | Pfizer Prod Inc | composições farmacêuticas de vareniclina |
PL378491A1 (pl) * | 2003-06-04 | 2006-05-02 | Pfizer Products Inc. | Sposób wytwarzania podstawionych chinoksalin z dianiliny i z 2,3-dihydroksy-1,4-dioksanu |
WO2005007630A2 (en) * | 2003-07-21 | 2005-01-27 | Pfizer Products Inc. | Aryl fused azapolycyclic compounds |
US8580842B2 (en) * | 2003-09-30 | 2013-11-12 | Abbott Gmbh & Co. Kg | Heteroaryl-substituted 1,3-dihydroindol-2-one derivatives and medicaments containing them |
JP4308263B2 (ja) | 2003-10-14 | 2009-08-05 | ゼノポート,インコーポレイティド | γ−アミノ酪酸アナログの結晶形 |
JP2007516275A (ja) * | 2003-12-23 | 2007-06-21 | ファイザー・プロダクツ・インク | 認知増強および精神病性障害のための治療的組合せ |
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EP1866308B1 (en) * | 2005-02-24 | 2008-10-22 | Pfizer Products Incorporated | Preparation of a high purity substituted quinoxaline |
RU2403016C2 (ru) * | 2006-04-24 | 2010-11-10 | Пфайзер Продактс Инк. | Асимметричные мембраны для устройств доставки лекарственного препарата |
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US8486979B2 (en) * | 2006-12-12 | 2013-07-16 | Abbvie Inc. | 1,2,4 oxadiazole compounds and methods of use thereof |
US20080167286A1 (en) | 2006-12-12 | 2008-07-10 | Abbott Laboratories | Pharmaceutical compositions and their methods of use |
UY30846A1 (es) * | 2006-12-30 | 2008-07-31 | Abbott Gmbh & Amp | Derivados de oxindol sustituidos, medicamentos que los comprenden y uso de los mismos |
US20090062257A1 (en) * | 2007-08-29 | 2009-03-05 | Protia, Llc | Deuterium-enriched varenicline |
WO2009034431A2 (en) | 2007-09-10 | 2009-03-19 | Pfizer Inc. | Controlled-release dosage forms for varenicline |
WO2009065872A2 (en) * | 2007-11-20 | 2009-05-28 | Medichem, S.A. | Improved processes for the synthesis of varenicline l-tartrate |
US8703774B2 (en) * | 2007-12-07 | 2014-04-22 | AbbVie Deutschland GmbH & Co. KG | Carbamate-substituted oxindole derivatives and use thereof for the treatment of vasopressin-dependent diseases |
CN101952276B (zh) * | 2007-12-07 | 2014-10-22 | Abbvie德国有限责任两合公司 | 5-卤素取代的羟吲哚衍生物和其用于治疗加压素依赖性疾病的用途 |
JP5645217B2 (ja) | 2007-12-07 | 2014-12-24 | アッヴィ・ドイチュラント・ゲー・エム・ベー・ハー・ウント・コー・カー・ゲー | 5,6−二置換オキシンドール誘導体およびバソプレッシン依存性疾患を治療するためのこれらの使用 |
JP5701607B2 (ja) * | 2007-12-07 | 2015-04-15 | アッヴィ・ドイチュラント・ゲー・エム・ベー・ハー・ウント・コー・カー・ゲー | アミドメチル置換オキシインドール誘導体およびバソプレッシン依存性疾患の治療へのこれらの使用 |
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JP2011516489A (ja) | 2008-03-31 | 2011-05-26 | ユニバーシティ・オブ・サウス・フロリダ | 疾患誘発性運動失調症および非運動失調性平衡異常の治療法 |
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CN110381919A (zh) | 2017-03-03 | 2019-10-25 | 西梯茜生命工学股份有限公司 | 含有伐尼克兰或其药学上可接受的盐的包合复合物的口服施用制剂 |
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2000
- 2000-02-25 US US09/514,002 patent/US6605610B1/en not_active Expired - Fee Related
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- 2001-02-08 OA OA1200200256A patent/OA12181A/en unknown
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- 2001-02-08 SK SK1204-2002A patent/SK12042002A3/sk not_active Application Discontinuation
- 2001-02-08 DK DK01953630T patent/DK1259489T3/da active
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- 2001-02-08 DZ DZ013328A patent/DZ3328A1/fr active
- 2001-02-08 BR BR0108610-3A patent/BR0108610A/pt not_active Application Discontinuation
- 2001-02-08 EA EA200200716A patent/EA005316B1/ru not_active IP Right Cessation
- 2001-02-08 ES ES05106835T patent/ES2336800T3/es not_active Expired - Lifetime
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- 2001-02-08 AU AU28748/01A patent/AU784081B2/en not_active Ceased
- 2001-02-08 PL PL01365163A patent/PL365163A1/xx not_active Application Discontinuation
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- 2001-02-08 WO PCT/IB2001/000153 patent/WO2001062736A1/en active IP Right Grant
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- 2001-02-08 ES ES01953630T patent/ES2263640T3/es not_active Expired - Lifetime
- 2001-02-08 EP EP01953630A patent/EP1259489B1/en not_active Expired - Lifetime
- 2001-02-08 AT AT01953630T patent/ATE328872T1/de active
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- 2001-02-08 JP JP2001562518A patent/JP2003524002A/ja active Pending
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- 2001-02-08 AP APAP/P/2002/002604A patent/AP1860A/en active
- 2001-02-08 KR KR10-2002-7011140A patent/KR100537976B1/ko not_active IP Right Cessation
- 2001-08-02 UA UA2002075792A patent/UA74813C2/uk unknown
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- 2002-07-08 IL IL150639A patent/IL150639A/en not_active IP Right Cessation
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- 2002-08-13 MA MA26775A patent/MA26875A1/fr unknown
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EP1044189B2 (en) | Aryl fused azapolycyclic compounds | |
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