MXPA05007565A - Procedimiento mejorado de preparacion de lactamas policiclicas fusionadas con arilos. - Google Patents

Procedimiento mejorado de preparacion de lactamas policiclicas fusionadas con arilos.

Info

Publication number
MXPA05007565A
MXPA05007565A MXPA05007565A MXPA05007565A MXPA05007565A MX PA05007565 A MXPA05007565 A MX PA05007565A MX PA05007565 A MXPA05007565 A MX PA05007565A MX PA05007565 A MXPA05007565 A MX PA05007565A MX PA05007565 A MXPA05007565 A MX PA05007565A
Authority
MX
Mexico
Prior art keywords
preparation
aryl fused
fused polycyclic
lactams
polycyclic lactams
Prior art date
Application number
MXPA05007565A
Other languages
English (en)
Inventor
Robert Eugene Handfield Jr
Original Assignee
Pfizer Prod Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc
Publication of MXPA05007565A publication Critical patent/MXPA05007565A/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D221/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00
    • C07D221/02—Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00 condensed with carbocyclic rings or ring systems
    • C07D221/22—Bridged ring systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D221/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00
    • C07D221/02—Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00 condensed with carbocyclic rings or ring systems
    • C07D221/22—Bridged ring systems
    • C07D221/26—Benzomorphans
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system

Abstract

La presente invencion se refiere a un procedimiento de preparacion de lactamas policiclicas fusionadas con arilos de formula I (ver formula (I)) que son intermedios utiles en la sintesis de compuestos azapoliciclicos fusionados con arilos como agentes para el tratamiento de trastornos neurologicos y psicologicos.
MXPA05007565A 2003-01-15 2004-01-08 Procedimiento mejorado de preparacion de lactamas policiclicas fusionadas con arilos. MXPA05007565A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US44026603P 2003-01-15 2003-01-15
PCT/IB2004/000152 WO2004063164A1 (en) 2003-01-15 2004-01-08 Process for the preparation of aryl fused polycyclic lactams

Publications (1)

Publication Number Publication Date
MXPA05007565A true MXPA05007565A (es) 2005-09-21

Family

ID=32713537

Family Applications (1)

Application Number Title Priority Date Filing Date
MXPA05007565A MXPA05007565A (es) 2003-01-15 2004-01-08 Procedimiento mejorado de preparacion de lactamas policiclicas fusionadas con arilos.

Country Status (19)

Country Link
US (1) US20070066827A1 (es)
EP (1) EP1587794A1 (es)
JP (1) JP2006517202A (es)
KR (2) KR20050101177A (es)
CN (1) CN100363350C (es)
AR (1) AR042855A1 (es)
AU (1) AU2004203983A1 (es)
BR (1) BRPI0406670A (es)
CA (1) CA2513293A1 (es)
CL (1) CL2004000041A1 (es)
HK (1) HK1085204A1 (es)
IL (1) IL169479A0 (es)
MX (1) MXPA05007565A (es)
PL (1) PL379373A1 (es)
RS (1) RS20050513A (es)
RU (1) RU2291862C2 (es)
TW (1) TW200420286A (es)
WO (1) WO2004063164A1 (es)
ZA (1) ZA200505103B (es)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2004048318A1 (en) 2002-11-25 2004-06-10 Pfizer Products Inc. Improved process for the preparation of 1,3-substituted indenes
CA2709774C (en) * 2008-05-22 2012-10-02 Teva Pharmaceutical Industries Ltd. Varenicline tosylate, an intermediate in the preparation process of varenicline l-tartrate
WO2009155403A2 (en) * 2008-06-19 2009-12-23 Teva Pharmaceutical Industries Ltd. Processes for the preparation of varenicline and intermediates thereof
EP2438054A1 (en) * 2009-06-22 2012-04-11 Teva Pharmaceutical Industries Ltd. Solid states forms of varenicline salts and processes for preparation thereof

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6605610B1 (en) * 1997-12-31 2003-08-12 Pfizer Inc Aryl fused azapolycyclic compounds
SI1044189T2 (sl) * 1997-12-31 2015-05-29 Pfizer Products Inc. Z arilom kondenzirane azapoliciklične spojine
DE60225433T2 (de) * 2001-04-20 2008-06-12 Pfizer Products Inc., Groton Verfahren zur herstellung von 1,3-substituierte indene und aryl-annellierte azapolycyclische verbindungen

Also Published As

Publication number Publication date
RU2005122406A (ru) 2006-01-27
US20070066827A1 (en) 2007-03-22
IL169479A0 (en) 2007-07-04
CL2004000041A1 (es) 2005-04-22
TW200420286A (en) 2004-10-16
CN1738803A (zh) 2006-02-22
AU2004203983A1 (en) 2004-07-29
BRPI0406670A (pt) 2005-12-20
RU2291862C2 (ru) 2007-01-20
EP1587794A1 (en) 2005-10-26
KR20070087258A (ko) 2007-08-27
PL379373A1 (pl) 2006-08-21
CN100363350C (zh) 2008-01-23
CA2513293A1 (en) 2004-07-29
AR042855A1 (es) 2005-07-06
WO2004063164A1 (en) 2004-07-29
JP2006517202A (ja) 2006-07-20
HK1085204A1 (en) 2006-08-18
WO2004063164A8 (en) 2005-05-26
RS20050513A (en) 2007-11-15
ZA200505103B (en) 2006-11-29
KR20050101177A (ko) 2005-10-20

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