TW200420286A - Improved process for the preparation of aryl fused polycyclic lactams - Google Patents

Improved process for the preparation of aryl fused polycyclic lactams

Info

Publication number
TW200420286A
TW200420286A TW093100889A TW93100889A TW200420286A TW 200420286 A TW200420286 A TW 200420286A TW 093100889 A TW093100889 A TW 093100889A TW 93100889 A TW93100889 A TW 93100889A TW 200420286 A TW200420286 A TW 200420286A
Authority
TW
Taiwan
Prior art keywords
preparation
aryl fused
fused polycyclic
improved process
lactams
Prior art date
Application number
TW093100889A
Other languages
English (en)
Inventor
Robert Eugene Handfield Jr
Timothy James Norman Watson
Original Assignee
Pfizer Prod Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc
Publication of TW200420286A publication Critical patent/TW200420286A/zh

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D221/00Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00
    • C07D221/02Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00 condensed with carbocyclic rings or ring systems
    • C07D221/22Bridged ring systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D221/00Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00
    • C07D221/02Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00 condensed with carbocyclic rings or ring systems
    • C07D221/22Bridged ring systems
    • C07D221/26Benzomorphans
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Hydrogenated Pyridines (AREA)
  • Other In-Based Heterocyclic Compounds (AREA)
TW093100889A 2003-01-15 2004-01-14 Improved process for the preparation of aryl fused polycyclic lactams TW200420286A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US44026603P 2003-01-15 2003-01-15

Publications (1)

Publication Number Publication Date
TW200420286A true TW200420286A (en) 2004-10-16

Family

ID=32713537

Family Applications (1)

Application Number Title Priority Date Filing Date
TW093100889A TW200420286A (en) 2003-01-15 2004-01-14 Improved process for the preparation of aryl fused polycyclic lactams

Country Status (19)

Country Link
US (1) US20070066827A1 (zh)
EP (1) EP1587794A1 (zh)
JP (1) JP2006517202A (zh)
KR (2) KR20070087258A (zh)
CN (1) CN100363350C (zh)
AR (1) AR042855A1 (zh)
AU (1) AU2004203983A1 (zh)
BR (1) BRPI0406670A (zh)
CA (1) CA2513293A1 (zh)
CL (1) CL2004000041A1 (zh)
HK (1) HK1085204A1 (zh)
IL (1) IL169479A0 (zh)
MX (1) MXPA05007565A (zh)
PL (1) PL379373A1 (zh)
RS (1) RS20050513A (zh)
RU (1) RU2291862C2 (zh)
TW (1) TW200420286A (zh)
WO (1) WO2004063164A1 (zh)
ZA (1) ZA200505103B (zh)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN1714075A (zh) 2002-11-25 2005-12-28 辉瑞产品公司 1,3-取代的茚类的改进制备方法
US8039620B2 (en) 2008-05-22 2011-10-18 Teva Pharmaceutical Industries Ltd. Varenicline tosylate, an intermediate in the preparation process of varenicline L-tartrate
US20090318695A1 (en) * 2008-06-19 2009-12-24 Vinod Kumar Kansal Processes for the preparation of varenicline and intermediates thereof
WO2010151524A1 (en) 2009-06-22 2010-12-29 Teva Pharmaceutical Industries Ltd Solid states forms of varenicline salts and processes for preparation thereof

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6605610B1 (en) * 1997-12-31 2003-08-12 Pfizer Inc Aryl fused azapolycyclic compounds
DK1044189T4 (en) * 1997-12-31 2015-03-30 Pfizer Prod Inc Aryl-fused fused azapolycyclic connections
MXPA03009527A (es) * 2001-04-20 2004-02-12 Pfizer Prod Inc PROCEDIMIENTO PARA LA PREPARACIoN DE INDENOS 1,3-SUSTITUIDOS Y COMPUESTOS AZAPOLICICLICOS CONDENSADOS CON ARILO.

Also Published As

Publication number Publication date
IL169479A0 (en) 2007-07-04
ZA200505103B (en) 2006-11-29
RU2291862C2 (ru) 2007-01-20
CN1738803A (zh) 2006-02-22
EP1587794A1 (en) 2005-10-26
RS20050513A (en) 2007-11-15
CL2004000041A1 (es) 2005-04-22
AR042855A1 (es) 2005-07-06
WO2004063164A1 (en) 2004-07-29
HK1085204A1 (en) 2006-08-18
WO2004063164A8 (en) 2005-05-26
KR20050101177A (ko) 2005-10-20
AU2004203983A1 (en) 2004-07-29
RU2005122406A (ru) 2006-01-27
BRPI0406670A (pt) 2005-12-20
CA2513293A1 (en) 2004-07-29
KR20070087258A (ko) 2007-08-27
PL379373A1 (pl) 2006-08-21
JP2006517202A (ja) 2006-07-20
CN100363350C (zh) 2008-01-23
MXPA05007565A (es) 2005-09-21
US20070066827A1 (en) 2007-03-22

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