NO309267B1 - Substituerte oxazolidin-calpain- og/eller cathepsin B- inhibitorer og farmasöytisk preparat inneholdende disse - Google Patents
Substituerte oxazolidin-calpain- og/eller cathepsin B- inhibitorer og farmasöytisk preparat inneholdende disse Download PDFInfo
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- NO309267B1 NO309267B1 NO973216A NO973216A NO309267B1 NO 309267 B1 NO309267 B1 NO 309267B1 NO 973216 A NO973216 A NO 973216A NO 973216 A NO973216 A NO 973216A NO 309267 B1 NO309267 B1 NO 309267B1
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- compound
- compound according
- acid
- phenylmethyl
- carbonyl
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Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
- C07D263/02—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings
- C07D263/04—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/08—Vasodilators for multiple indications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
Landscapes
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Neurosurgery (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Vascular Medicine (AREA)
- Urology & Nephrology (AREA)
- Hospice & Palliative Care (AREA)
- Psychiatry (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US37119295A | 1995-01-11 | 1995-01-11 | |
| PCT/US1995/016565 WO1996021655A2 (en) | 1995-01-11 | 1995-12-15 | Substituted oxazolidine calpain and/or cathepsin b inhibitors |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| NO973216D0 NO973216D0 (no) | 1997-07-10 |
| NO973216L NO973216L (no) | 1997-09-09 |
| NO309267B1 true NO309267B1 (no) | 2001-01-08 |
Family
ID=23462894
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NO973216A NO309267B1 (no) | 1995-01-11 | 1997-07-10 | Substituerte oxazolidin-calpain- og/eller cathepsin B- inhibitorer og farmasöytisk preparat inneholdende disse |
Country Status (23)
| Country | Link |
|---|---|
| US (1) | US5691368A (es) |
| EP (1) | EP0802909B1 (es) |
| JP (1) | JP4157601B2 (es) |
| KR (1) | KR100393701B1 (es) |
| CN (1) | CN1088456C (es) |
| AR (1) | AR001787A1 (es) |
| AT (1) | ATE206413T1 (es) |
| AU (1) | AU692044B2 (es) |
| CA (1) | CA2210258C (es) |
| DE (1) | DE69523072T2 (es) |
| DK (1) | DK0802909T3 (es) |
| ES (1) | ES2165441T3 (es) |
| FI (1) | FI972935A (es) |
| HU (1) | HUT77649A (es) |
| IL (1) | IL116724A (es) |
| MX (1) | MX9705235A (es) |
| NO (1) | NO309267B1 (es) |
| NZ (1) | NZ298999A (es) |
| PT (1) | PT802909E (es) |
| SI (1) | SI0802909T1 (es) |
| TW (1) | TW454001B (es) |
| WO (1) | WO1996021655A2 (es) |
| ZA (1) | ZA96100B (es) |
Families Citing this family (38)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| IT1270882B (it) * | 1993-10-05 | 1997-05-13 | Isagro Srl | Oligopeptidi ad attivita' fungicida |
| US5925633A (en) * | 1996-03-06 | 1999-07-20 | Synphar Laboraties, Inc. | 3-Substituted-4-oxa-1-azabicyclo 3,2,0!heptan-7-one as cysteine protease inhibitors |
| WO1998038990A1 (en) * | 1997-03-07 | 1998-09-11 | Hoechst Marion Roussel, Inc. | Method of treating trauma associated with brain, spinal cord or peripheral nerve injury using carbobenzyloxy n-protected di- and tripeptide phenylalaninals |
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-
1995
- 1995-12-11 US US08/552,139 patent/US5691368A/en not_active Expired - Lifetime
- 1995-12-15 AU AU44731/96A patent/AU692044B2/en not_active Ceased
- 1995-12-15 JP JP52166996A patent/JP4157601B2/ja not_active Expired - Lifetime
- 1995-12-15 MX MX9705235A patent/MX9705235A/es unknown
- 1995-12-15 CN CN95197320A patent/CN1088456C/zh not_active Expired - Fee Related
- 1995-12-15 EP EP95943478A patent/EP0802909B1/en not_active Expired - Lifetime
- 1995-12-15 PT PT95943478T patent/PT802909E/pt unknown
- 1995-12-15 NZ NZ298999A patent/NZ298999A/xx unknown
- 1995-12-15 KR KR1019970704709A patent/KR100393701B1/ko not_active IP Right Cessation
- 1995-12-15 CA CA002210258A patent/CA2210258C/en not_active Expired - Lifetime
- 1995-12-15 DK DK95943478T patent/DK0802909T3/da active
- 1995-12-15 SI SI9530539T patent/SI0802909T1/xx unknown
- 1995-12-15 HU HU9800041A patent/HUT77649A/hu unknown
- 1995-12-15 WO PCT/US1995/016565 patent/WO1996021655A2/en active IP Right Grant
- 1995-12-15 DE DE69523072T patent/DE69523072T2/de not_active Expired - Lifetime
- 1995-12-15 AT AT95943478T patent/ATE206413T1/de not_active IP Right Cessation
- 1995-12-15 ES ES95943478T patent/ES2165441T3/es not_active Expired - Lifetime
-
1996
- 1996-01-08 ZA ZA96100A patent/ZA96100B/xx unknown
- 1996-01-09 IL IL11672496A patent/IL116724A/xx not_active IP Right Cessation
- 1996-01-09 AR AR33495896A patent/AR001787A1/es unknown
- 1996-01-10 TW TW085100250A patent/TW454001B/zh not_active IP Right Cessation
-
1997
- 1997-07-10 FI FI972935A patent/FI972935A/fi not_active IP Right Cessation
- 1997-07-10 NO NO973216A patent/NO309267B1/no not_active IP Right Cessation
Also Published As
| Publication number | Publication date |
|---|---|
| FI972935A0 (fi) | 1997-07-10 |
| CA2210258C (en) | 2002-10-01 |
| EP0802909B1 (en) | 2001-10-04 |
| DE69523072T2 (de) | 2002-06-20 |
| MX9705235A (es) | 1997-10-31 |
| KR100393701B1 (ko) | 2003-11-28 |
| NO973216D0 (no) | 1997-07-10 |
| NO973216L (no) | 1997-09-09 |
| JP4157601B2 (ja) | 2008-10-01 |
| IL116724A (en) | 2000-08-31 |
| DE69523072D1 (en) | 2001-11-08 |
| ZA96100B (en) | 1996-07-24 |
| WO1996021655A3 (en) | 1996-09-06 |
| AR001787A1 (es) | 1997-12-10 |
| AU692044B2 (en) | 1998-05-28 |
| CN1088456C (zh) | 2002-07-31 |
| US5691368A (en) | 1997-11-25 |
| AU4473196A (en) | 1996-07-31 |
| ES2165441T3 (es) | 2002-03-16 |
| WO1996021655A2 (en) | 1996-07-18 |
| SI0802909T1 (en) | 2002-02-28 |
| CN1173174A (zh) | 1998-02-11 |
| FI972935A (fi) | 1997-07-10 |
| NZ298999A (en) | 1999-01-28 |
| IL116724A0 (en) | 1996-05-14 |
| DK0802909T3 (da) | 2002-01-28 |
| PT802909E (pt) | 2002-03-28 |
| JPH10512257A (ja) | 1998-11-24 |
| HUT77649A (hu) | 1998-07-28 |
| EP0802909A2 (en) | 1997-10-29 |
| ATE206413T1 (de) | 2001-10-15 |
| CA2210258A1 (en) | 1996-07-18 |
| TW454001B (en) | 2001-09-11 |
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