NO309142B1 - N<alfa>-2-(4-nitrofenylsulfonyl)etoksykarbonylaminosyrer og fremgangsmåter derfor - Google Patents

N<alfa>-2-(4-nitrofenylsulfonyl)etoksykarbonylaminosyrer og fremgangsmåter derfor Download PDF

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Publication number
NO309142B1
NO309142B1 NO973752A NO973752A NO309142B1 NO 309142 B1 NO309142 B1 NO 309142B1 NO 973752 A NO973752 A NO 973752A NO 973752 A NO973752 A NO 973752A NO 309142 B1 NO309142 B1 NO 309142B1
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NO
Norway
Prior art keywords
protected
amino acid
polymer
nsc
group
Prior art date
Application number
NO973752A
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English (en)
Norwegian (no)
Other versions
NO973752L (no
NO973752D0 (no
Inventor
Vladimir Vasilyevich Samukov
Ayda Nadzhatovich Sabirov
Pavel Ivanovich Pozdnyarkov
Original Assignee
Hyundai Pharm Ind Co Ltd
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Publication date
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First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=20164784&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=NO309142(B1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Hyundai Pharm Ind Co Ltd filed Critical Hyundai Pharm Ind Co Ltd
Publication of NO973752D0 publication Critical patent/NO973752D0/no
Publication of NO973752L publication Critical patent/NO973752L/no
Publication of NO309142B1 publication Critical patent/NO309142B1/no

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C323/00Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups
    • C07C323/50Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and carboxyl groups bound to the same carbon skeleton
    • C07C323/51Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and carboxyl groups bound to the same carbon skeleton having the sulfur atoms of the thio groups bound to acyclic carbon atoms of the carbon skeleton
    • C07C323/57Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and carboxyl groups bound to the same carbon skeleton having the sulfur atoms of the thio groups bound to acyclic carbon atoms of the carbon skeleton the carbon skeleton being further substituted by nitrogen atoms, not being part of nitro or nitroso groups
    • C07C323/58Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and carboxyl groups bound to the same carbon skeleton having the sulfur atoms of the thio groups bound to acyclic carbon atoms of the carbon skeleton the carbon skeleton being further substituted by nitrogen atoms, not being part of nitro or nitroso groups with amino groups bound to the carbon skeleton
    • C07C323/59Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and carboxyl groups bound to the same carbon skeleton having the sulfur atoms of the thio groups bound to acyclic carbon atoms of the carbon skeleton the carbon skeleton being further substituted by nitrogen atoms, not being part of nitro or nitroso groups with amino groups bound to the carbon skeleton with acylated amino groups bound to the carbon skeleton
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C317/00Sulfones; Sulfoxides
    • C07C317/16Sulfones; Sulfoxides having sulfone or sulfoxide groups and singly-bound oxygen atoms bound to the same carbon skeleton
    • C07C317/18Sulfones; Sulfoxides having sulfone or sulfoxide groups and singly-bound oxygen atoms bound to the same carbon skeleton with sulfone or sulfoxide groups bound to acyclic carbon atoms of the carbon skeleton
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C317/00Sulfones; Sulfoxides
    • C07C317/44Sulfones; Sulfoxides having sulfone or sulfoxide groups and carboxyl groups bound to the same carbon skeleton
    • C07C317/48Sulfones; Sulfoxides having sulfone or sulfoxide groups and carboxyl groups bound to the same carbon skeleton the carbon skeleton being further substituted by singly-bound nitrogen atoms, not being part of nitro or nitroso groups
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D473/00Heterocyclic compounds containing purine ring systems
    • C07D473/02Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6
    • C07D473/04Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6 two oxygen atoms
    • C07D473/06Heterocyclic compounds containing purine ring systems with oxygen, sulphur, or nitrogen atoms directly attached in positions 2 and 6 two oxygen atoms with radicals containing only hydrogen and carbon atoms, attached in position 1 or 3
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K1/00General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length
    • C07K1/06General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length using protecting groups or activating agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K1/00General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length
    • C07K1/06General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length using protecting groups or activating agents
    • C07K1/061General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length using protecting groups or activating agents using protecting groups
    • C07K1/063General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length using protecting groups or activating agents using protecting groups for alpha-amino functions

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Chemistry (AREA)
  • Molecular Biology (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • General Health & Medical Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Analytical Chemistry (AREA)
  • Peptides Or Proteins (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
NO973752A 1995-02-15 1997-08-14 N<alfa>-2-(4-nitrofenylsulfonyl)etoksykarbonylaminosyrer og fremgangsmåter derfor NO309142B1 (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
RU9595102102A RU2079491C1 (ru) 1995-02-15 1995-02-15 Nα -2-(4-НИТРОФЕНИЛСУЛЬФОНИЛ)ЭТОКСИКАРБОНИЛ-АМИНОКИСЛОТЫ В КАЧЕСТВЕ Nα -ЗАЩИЩЕННЫХ АМИНОКИСЛОТ ДЛЯ ТВЕРДОФАЗНОГО СИНТЕЗА ПЕПТИДОВ
PCT/KR1996/000012 WO1996025394A1 (en) 1995-02-15 1996-01-27 Nα-2-(4-NITROPHENULSULFONYL)ETHOXYCARBONYL-AMINO ACIDS

Publications (3)

Publication Number Publication Date
NO973752D0 NO973752D0 (no) 1997-08-14
NO973752L NO973752L (no) 1997-10-14
NO309142B1 true NO309142B1 (no) 2000-12-18

Family

ID=20164784

Family Applications (1)

Application Number Title Priority Date Filing Date
NO973752A NO309142B1 (no) 1995-02-15 1997-08-14 N<alfa>-2-(4-nitrofenylsulfonyl)etoksykarbonylaminosyrer og fremgangsmåter derfor

Country Status (19)

Country Link
US (1) US5616788A (ru)
EP (1) EP0765307B1 (ru)
JP (1) JP2888991B2 (ru)
KR (1) KR100241948B1 (ru)
CN (1) CN1058260C (ru)
AT (1) ATE185796T1 (ru)
AU (1) AU705716B2 (ru)
CA (1) CA2212052C (ru)
CZ (1) CZ289747B6 (ru)
DE (1) DE69604759T2 (ru)
DK (1) DK0765307T3 (ru)
ES (1) ES2140061T3 (ru)
FI (1) FI973338A (ru)
GR (1) GR3031832T3 (ru)
HU (1) HUP9801150A3 (ru)
NO (1) NO309142B1 (ru)
PL (1) PL184205B1 (ru)
RU (1) RU2079491C1 (ru)
WO (1) WO1996025394A1 (ru)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN1090615C (zh) * 1996-10-19 2002-09-11 Hyundai药物工业株式会社 Nα-2-(4-硝基苯基磺酰基)乙氧羰基氨基酸
JP2001502686A (ja) 1996-10-19 2001-02-27 ヒュンダイ ファーマスティカル インダストリアル カンパニー リミテッド N▲下α▼―2―(4―ニトロフェニルスルホニル)エトキシカルボニル―アミノ酸
KR100378252B1 (ko) * 1999-11-12 2003-03-29 학교법인 포항공과대학교 니트로술포닐에톡시카르보닐-아미노산을 이용한 합성테트라펩티드 라이브러리의 제조방법
AU1894000A (en) * 1999-12-24 2001-07-24 Hyundai Pharmaceutical Ind. Co., Ltd. Nalpha-2-(4-nitrophenylsulfonyl)ethoxycarbonyl-amino acid fluorides and process for the preparation thereof
KR100418962B1 (ko) * 2001-06-07 2004-02-14 김학주 2-(4-나이트로페닐설포닐)에톡시카르보닐-아미노산류를사용하여 펩티드를 고수율 및 고순도로 제조하는 방법
WO2009014177A1 (ja) * 2007-07-25 2009-01-29 Ajinomoto Co., Inc. ジベンゾフルベン誘導体の淘汰方法
CN103421087A (zh) * 2013-04-12 2013-12-04 上海捌加壹医药科技有限公司 一种多肽的液相合成方法
WO2024079043A1 (en) 2022-10-10 2024-04-18 Bachem Holding Ag Method of manufacturing a peptide with a lysine derivative

Also Published As

Publication number Publication date
NO973752L (no) 1997-10-14
FI973338A0 (fi) 1997-08-14
EP0765307B1 (en) 1999-10-20
WO1996025394A1 (en) 1996-08-22
HUP9801150A3 (en) 2000-07-28
CN1058260C (zh) 2000-11-08
CZ247797A3 (cs) 1998-02-18
CN1173865A (zh) 1998-02-18
DE69604759D1 (de) 1999-11-25
JP2888991B2 (ja) 1999-05-10
CA2212052A1 (en) 1996-08-22
CZ289747B6 (cs) 2002-03-13
AU705716B2 (en) 1999-05-27
PL321864A1 (en) 1997-12-22
JPH10503216A (ja) 1998-03-24
AU4549696A (en) 1996-09-04
RU95102102A (ru) 1996-11-20
FI973338A (fi) 1997-10-14
KR19980702267A (ko) 1998-07-15
PL184205B1 (pl) 2002-09-30
RU2079491C1 (ru) 1997-05-20
HUP9801150A2 (hu) 1998-09-28
DE69604759T2 (de) 2000-06-21
DK0765307T3 (da) 1999-12-27
CA2212052C (en) 2002-09-03
EP0765307A1 (en) 1997-04-02
GR3031832T3 (en) 2000-02-29
ES2140061T3 (es) 2000-02-16
NO973752D0 (no) 1997-08-14
US5616788A (en) 1997-04-01
KR100241948B1 (ko) 2000-02-01
ATE185796T1 (de) 1999-11-15

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