NO20041428L - Oksazolidinon og/eller isoksazolin som antibakterielle midler. - Google Patents

Oksazolidinon og/eller isoksazolin som antibakterielle midler.

Info

Publication number
NO20041428L
NO20041428L NO20041428A NO20041428A NO20041428L NO 20041428 L NO20041428 L NO 20041428L NO 20041428 A NO20041428 A NO 20041428A NO 20041428 A NO20041428 A NO 20041428A NO 20041428 L NO20041428 L NO 20041428L
Authority
NO
Norway
Prior art keywords
isoxazoline
oxazolidinone
antibacterial agents
antibacterial
agents
Prior art date
Application number
NO20041428A
Other languages
English (en)
Other versions
NO327010B1 (no
Inventor
Michael Lingard Swain
Stuart Dennett Mills
Michael Barry Gravestock
Neil James Hales
Sheila Irene Hauck
Original Assignee
Astrazeneca Ab Global Ip
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GB0121942A external-priority patent/GB0121942D0/en
Priority claimed from GB0215420A external-priority patent/GB0215420D0/en
Application filed by Astrazeneca Ab Global Ip filed Critical Astrazeneca Ab Global Ip
Publication of NO20041428L publication Critical patent/NO20041428L/no
Publication of NO327010B1 publication Critical patent/NO327010B1/no

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D263/00Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
    • C07D263/02Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings
    • C07D263/08Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D263/16Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D263/18Oxygen atoms
    • C07D263/20Oxygen atoms attached in position 2
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/10Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing aromatic rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/14Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
NO20041428A 2001-09-11 2004-04-05 Oksazolidinon og/eller isoksazolin anvendelse derav som antibakterielle midler, farmasoytisk sammensetning og fremgangsmate for fremstilling derav NO327010B1 (no)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GB0121942A GB0121942D0 (en) 2001-09-11 2001-09-11 Chemical compounds
GB0215420A GB0215420D0 (en) 2002-07-04 2002-07-04 Chemical compounds
PCT/GB2002/004120 WO2003022824A1 (en) 2001-09-11 2002-09-09 Oxazolidinone and/or isoxazoline as antibacterial agents

Publications (2)

Publication Number Publication Date
NO20041428L true NO20041428L (no) 2004-06-08
NO327010B1 NO327010B1 (no) 2009-04-06

Family

ID=26246531

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20041428A NO327010B1 (no) 2001-09-11 2004-04-05 Oksazolidinon og/eller isoksazolin anvendelse derav som antibakterielle midler, farmasoytisk sammensetning og fremgangsmate for fremstilling derav

Country Status (26)

Country Link
US (2) US7396847B2 (no)
EP (1) EP1427711B1 (no)
JP (1) JP2005507386A (no)
KR (1) KR20040044886A (no)
CN (1) CN1639136A (no)
AR (1) AR036778A1 (no)
AT (1) ATE299502T1 (no)
AU (1) AU2002329393B2 (no)
BR (1) BR0212458A (no)
CA (1) CA2459766A1 (no)
CO (1) CO5560609A2 (no)
DE (1) DE60205030T2 (no)
DK (1) DK1427711T3 (no)
ES (1) ES2244802T3 (no)
HK (1) HK1065789A1 (no)
HU (1) HUP0401005A3 (no)
IL (1) IL160739A0 (no)
IS (1) IS7175A (no)
MX (1) MXPA04002303A (no)
NO (1) NO327010B1 (no)
NZ (1) NZ531621A (no)
PL (1) PL369183A1 (no)
PT (1) PT1427711E (no)
RU (1) RU2004111285A (no)
SI (1) SI1427711T1 (no)
WO (1) WO2003022824A1 (no)

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ES2536001T3 (es) * 2003-07-29 2015-05-19 Melinta Therapeutics, Inc. Procedimiento para la síntesis de biariloxazolidinonas
EP1713785A1 (en) 2003-12-17 2006-10-25 Rib-X Pharmaceuticals, Inc. Halogenated biaryl heterocyclic compounds and methods of making and using the same
KR100854211B1 (ko) 2003-12-18 2008-08-26 동아제약주식회사 신규한 옥사졸리디논 유도체, 그의 제조방법 및 이를유효성분으로 하는 항생제용 약학 조성물
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CN106220621B (zh) * 2008-10-10 2019-06-11 默沙东公司 制备噁唑烷酮类的方法及含有噁唑烷酮类的组合物
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US8580767B2 (en) 2009-05-28 2013-11-12 Trius Therapeutics, Inc. Oxazolidinone containing dimer compounds, compositions and methods to make and use
KR101561964B1 (ko) 2013-11-15 2015-10-20 한국과학기술연구원 옥사졸리디논 화합물 및 이를 포함하는 c형 간염 예방 또는 치료용 약학 조성물
CN114874131A (zh) * 2015-02-27 2022-08-09 海洋规划生物工厂株式会社 Kakeromycin及其衍生物的制造方法
CN106083994B (zh) * 2016-04-18 2019-12-06 南京曼杰生物科技有限公司 取代的噁唑烷酮水溶性衍生物及其应用
US20170333305A1 (en) * 2016-05-23 2017-11-23 Microban Products Company Topical skin product having retention property
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CN113149924B (zh) * 2021-03-29 2023-11-03 苏州大学 一种异噁唑啉的简单制备方法
CN113831517A (zh) * 2021-09-09 2021-12-24 万凯新材料股份有限公司 抗菌及抗紫外聚酯的制备方法

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IL163688A0 (en) 2002-02-28 2005-12-18 Astrazeneca Ab 3-Cyclyl-5-(nitrogen-containing 5-membered ring)methyl-oxazolidinone derivatives and theiruse as antibacterial agents
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Also Published As

Publication number Publication date
RU2004111285A (ru) 2005-10-10
DK1427711T3 (da) 2005-10-17
EP1427711B1 (en) 2005-07-13
CO5560609A2 (es) 2005-09-30
NZ531621A (en) 2005-06-24
CA2459766A1 (en) 2003-03-20
US20100137243A1 (en) 2010-06-03
IS7175A (is) 2004-03-10
DE60205030T2 (de) 2006-04-20
MXPA04002303A (es) 2004-06-29
PT1427711E (pt) 2005-11-30
PL369183A1 (en) 2005-04-18
CN1639136A (zh) 2005-07-13
HUP0401005A3 (en) 2007-11-28
US7396847B2 (en) 2008-07-08
HUP0401005A2 (hu) 2004-08-30
IL160739A0 (en) 2004-08-31
HK1065789A1 (en) 2005-03-04
KR20040044886A (ko) 2004-05-31
ATE299502T1 (de) 2005-07-15
EP1427711A1 (en) 2004-06-16
AR036778A1 (es) 2004-10-06
ES2244802T3 (es) 2005-12-16
BR0212458A (pt) 2004-10-19
DE60205030D1 (de) 2005-08-18
SI1427711T1 (sl) 2005-12-31
WO2003022824A1 (en) 2003-03-20
NO327010B1 (no) 2009-04-06
JP2005507386A (ja) 2005-03-17
AU2002329393B2 (en) 2008-06-12
US20050107435A1 (en) 2005-05-19

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