NO20032271L - GABA-enhancere i behandlingen av sykdommer relatert til redusert nevrosteroidaktivitet - Google Patents

GABA-enhancere i behandlingen av sykdommer relatert til redusert nevrosteroidaktivitet

Info

Publication number
NO20032271L
NO20032271L NO20032271A NO20032271A NO20032271L NO 20032271 L NO20032271 L NO 20032271L NO 20032271 A NO20032271 A NO 20032271A NO 20032271 A NO20032271 A NO 20032271A NO 20032271 L NO20032271 L NO 20032271L
Authority
NO
Norway
Prior art keywords
treatment
gaba
diseases related
activity
enhancers
Prior art date
Application number
NO20032271A
Other languages
English (en)
Other versions
NO20032271D0 (no
Inventor
Bjarke Ebert
Peter Hongaard Andersen
Original Assignee
Lundbeck & Co As H
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=8159857&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=NO20032271(L) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Lundbeck & Co As H filed Critical Lundbeck & Co As H
Publication of NO20032271D0 publication Critical patent/NO20032271D0/no
Publication of NO20032271L publication Critical patent/NO20032271L/no

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Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/185—Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19—Carboxylic acids, e.g. valproic acid
    • A61K31/195—Carboxylic acids, e.g. valproic acid having an amino group
    • A61K31/197—Carboxylic acids, e.g. valproic acid having an amino group the amino and the carboxyl groups being attached to the same acyclic carbon chain, e.g. gamma-aminobutyric acid [GABA], beta-alanine, epsilon-aminocaproic acid or pantothenic acid
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/185—Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19—Carboxylic acids, e.g. valproic acid
    • A61K31/195—Carboxylic acids, e.g. valproic acid having an amino group
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4164—1,3-Diazoles
    • A61K31/4172—Imidazole-alkanecarboxylic acids, e.g. histidine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/42—Oxazoles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/437—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a five-membered ring having nitrogen as a ring hetero atom, e.g. indolizine, beta-carboline
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445—Non condensed piperidines, e.g. piperocaine
    • A61K31/4523—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
    • A61K31/4535—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a heterocyclic ring having sulfur as a ring hetero atom, e.g. pizotifen
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A61P15/12—Drugs for genital or sexual disorders; Contraceptives for climacteric disorders
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/22—Anxiolytics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/24—Drugs for disorders of the endocrine system of the sex hormones

Landscapes

  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Epidemiology (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Endocrinology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Reproductive Health (AREA)
  • Diabetes (AREA)
  • Psychiatry (AREA)
  • Pain & Pain Management (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Steroid Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Indole Compounds (AREA)
  • Hydrogenated Pyridines (AREA)

Abstract

Foreliggende oppfinnelse tilveiebringer anvendelsen av et ikke-steroid forbindelse som påvirker GABA-reseptor for behandling av forstyrrelser som vedrører redusert nevrosteroidaktivitet. De ikke-steroide forbindelsene kan være GABA-agonister, GABA-opptakhemmere eller enhancere av GABAergisk aktivitet.
NO20032271A 2000-11-20 2003-05-20 GABA-enhancere i behandlingen av sykdommer relatert til redusert nevrosteroidaktivitet NO20032271L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DKPA200001743 2000-11-20
PCT/DK2001/000773 WO2002040009A1 (en) 2000-11-20 2001-11-20 Gaba enhancers in the treatment of diseases relating to reduced neurosteroid activity

Publications (2)

Publication Number Publication Date
NO20032271D0 NO20032271D0 (no) 2003-05-20
NO20032271L true NO20032271L (no) 2003-05-20

Family

ID=8159857

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20032271A NO20032271L (no) 2000-11-20 2003-05-20 GABA-enhancere i behandlingen av sykdommer relatert til redusert nevrosteroidaktivitet

Country Status (34)

Country Link
US (2) US20040024038A1 (no)
EP (1) EP1337247B1 (no)
JP (1) JP4152186B2 (no)
KR (1) KR100865651B1 (no)
CN (1) CN1318027C (no)
AR (1) AR031473A1 (no)
AT (1) ATE336242T1 (no)
AU (2) AU2351402A (no)
BG (1) BG107909A (no)
BR (1) BR0115668A (no)
CA (1) CA2429220C (no)
CY (1) CY1106209T1 (no)
CZ (1) CZ20031383A3 (no)
DE (1) DE60122368T2 (no)
DK (1) DK1337247T3 (no)
EA (1) EA007287B1 (no)
ES (1) ES2266308T3 (no)
HK (1) HK1075010A1 (no)
HR (1) HRP20030404A2 (no)
HU (1) HUP0400505A3 (no)
IL (1) IL155587A0 (no)
IS (1) IS2427B (no)
ME (1) MEP6408A (no)
MX (1) MXPA03004349A (no)
NO (1) NO20032271L (no)
NZ (1) NZ525520A (no)
PL (1) PL361051A1 (no)
PT (1) PT1337247E (no)
SI (1) SI1337247T1 (no)
SK (1) SK7682003A3 (no)
UA (1) UA77403C2 (no)
WO (1) WO2002040009A1 (no)
YU (1) YU39003A (no)
ZA (1) ZA200303289B (no)

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PL1641456T3 (pl) * 2003-06-25 2010-08-31 H Lundbeck As Gaboksadol do leczenia depresji i innych zaburzeń afektywnych
GB0402118D0 (en) 2004-01-30 2004-03-03 Merck Sharp & Dohme Polymorphic forms of a GABAA agonist
MXPA06015196A (es) * 2004-06-29 2007-03-15 Lundbeck & Co As H Tratamiento del dolor neuropatico, la fibromialgia o la artritis reumatoide.
WO2006012563A2 (en) * 2004-07-23 2006-02-02 The Regents Of The University Of California Method for the treatment and diagnosis of certain psychiatric disorders related to the menstrual cycle
GB0417558D0 (en) * 2004-08-06 2004-09-08 Merck Sharp & Dohme Novel combination therapy
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KR102049526B1 (ko) * 2018-06-05 2019-11-27 충남대학교산학협력단 Gaba를 유효성분으로 하는 항결핵 약학 조성물
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Also Published As

Publication number Publication date
MXPA03004349A (es) 2003-08-19
BG107909A (bg) 2004-08-31
IS6803A (is) 2003-04-30
EA007287B1 (ru) 2006-08-25
CY1106209T1 (el) 2011-06-08
EA200300594A1 (ru) 2003-10-30
HUP0400505A3 (en) 2008-08-28
YU39003A (sh) 2006-05-25
SI1337247T1 (sl) 2006-12-31
HUP0400505A2 (hu) 2004-07-28
CA2429220C (en) 2009-09-15
BR0115668A (pt) 2003-09-02
KR20030065517A (ko) 2003-08-06
KR100865651B1 (ko) 2008-10-29
CZ20031383A3 (cs) 2003-08-13
HRP20030404A2 (en) 2005-04-30
DE60122368T2 (de) 2007-08-09
ATE336242T1 (de) 2006-09-15
US20090143435A1 (en) 2009-06-04
NO20032271D0 (no) 2003-05-20
IL155587A0 (en) 2003-11-23
SK7682003A3 (en) 2003-10-07
DK1337247T3 (da) 2006-12-04
DE60122368D1 (de) 2006-09-28
EP1337247B1 (en) 2006-08-16
CN1592616A (zh) 2005-03-09
AU2351402A (en) 2002-05-27
CN1318027C (zh) 2007-05-30
NZ525520A (en) 2005-04-29
EP1337247A1 (en) 2003-08-27
AR031473A1 (es) 2003-09-24
ZA200303289B (en) 2005-07-27
AU2002223514B2 (en) 2006-11-30
ES2266308T3 (es) 2007-03-01
PT1337247E (pt) 2006-11-30
CA2429220A1 (en) 2002-05-23
JP4152186B2 (ja) 2008-09-17
US20040024038A1 (en) 2004-02-05
PL361051A1 (en) 2004-09-20
WO2002040009A1 (en) 2002-05-23
HK1075010A1 (en) 2005-12-02
IS2427B (is) 2008-10-15
UA77403C2 (en) 2006-12-15
MEP6408A (xx) 2010-02-10
JP2004513921A (ja) 2004-05-13

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