NO20013179L - Aromatiske heterocyklusforbindelser som har HIV integrase- inhiberende aktiviteter - Google Patents

Aromatiske heterocyklusforbindelser som har HIV integrase- inhiberende aktiviteter

Info

Publication number
NO20013179L
NO20013179L NO20013179A NO20013179A NO20013179L NO 20013179 L NO20013179 L NO 20013179L NO 20013179 A NO20013179 A NO 20013179A NO 20013179 A NO20013179 A NO 20013179A NO 20013179 L NO20013179 L NO 20013179L
Authority
NO
Norway
Prior art keywords
aromatic heterocycle
hiv integrase
inhibitory activities
heterocycle compounds
integrase inhibitory
Prior art date
Application number
NO20013179A
Other languages
English (en)
Norwegian (no)
Other versions
NO20013179D0 (no
Inventor
Toshio Fujishita
Tomokazu Yoshinaga
Akihiko Sato
Original Assignee
Shionogi & Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Shionogi & Co filed Critical Shionogi & Co
Publication of NO20013179D0 publication Critical patent/NO20013179D0/no
Publication of NO20013179L publication Critical patent/NO20013179L/no

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/41961,2,4-Triazoles
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D403/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/06Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/14Antivirals for RNA viruses
    • A61P31/18Antivirals for RNA viruses for HIV
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D333/00Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/02Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
    • C07D333/04Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
    • C07D333/06Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to the ring carbon atoms
    • C07D333/24Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D333/00Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/02Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
    • C07D333/04Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
    • C07D333/26Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D333/30Hetero atoms other than halogen
    • C07D333/34Sulfur atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Virology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • AIDS & HIV (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Molecular Biology (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
NO20013179A 1998-12-25 2001-06-22 Aromatiske heterocyklusforbindelser som har HIV integrase- inhiberende aktiviteter NO20013179L (no)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
JP37127098 1998-12-25
JP24747999 1999-09-01
PCT/JP1999/007101 WO2000039086A1 (fr) 1998-12-25 1999-12-17 Composes heterocycliques aromatiques possedant des activites inhibitrices de l'integrase du vih

Publications (2)

Publication Number Publication Date
NO20013179D0 NO20013179D0 (no) 2001-06-22
NO20013179L true NO20013179L (no) 2001-08-27

Family

ID=26538287

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20013179A NO20013179L (no) 1998-12-25 2001-06-22 Aromatiske heterocyklusforbindelser som har HIV integrase- inhiberende aktiviteter

Country Status (22)

Country Link
US (3) US6620841B1 (id)
EP (1) EP1142872B1 (id)
JP (1) JP3929244B2 (id)
KR (1) KR20010089708A (id)
CN (1) CN1178913C (id)
AP (1) AP2001002169A0 (id)
AT (1) ATE411286T1 (id)
AU (1) AU763040B2 (id)
BR (1) BR9916583A (id)
CA (1) CA2353961A1 (id)
CZ (1) CZ20012160A3 (id)
DE (1) DE69939749D1 (id)
HK (1) HK1042701A1 (id)
HU (1) HUP0201472A3 (id)
ID (1) ID29027A (id)
IL (1) IL143958A0 (id)
NO (1) NO20013179L (id)
NZ (1) NZ512184A (id)
PL (1) PL348596A1 (id)
RU (1) RU2225860C2 (id)
TR (1) TR200101886T2 (id)
WO (1) WO2000039086A1 (id)

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WO2008041882A1 (fr) * 2006-10-03 2008-04-10 Viktor Veniaminovich Tets Procédé pour agir sur les virus au moyen d'une substance à base de 2,8-dithioxo-1h- pyrano[2,3-d;6,5-d'] dipyrimidine et de leurs analogues 10-aza (et variantes)
CN102670628B (zh) 2008-01-25 2015-11-25 奇默里克斯公司 治疗病毒感染的方法
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TWI695003B (zh) 2014-12-23 2020-06-01 美商基利科學股份有限公司 多環胺甲醯基吡啶酮化合物及其醫藥用途
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Also Published As

Publication number Publication date
RU2225860C2 (ru) 2004-03-20
JP3929244B2 (ja) 2007-06-13
HK1042701A1 (zh) 2002-08-23
EP1142872B1 (en) 2008-10-15
WO2000039086A1 (fr) 2000-07-06
HUP0201472A2 (hu) 2003-10-28
US6620841B1 (en) 2003-09-16
AP2001002169A0 (en) 2001-06-30
PL348596A1 (en) 2002-06-03
ID29027A (id) 2001-07-26
DE69939749D1 (de) 2008-11-27
NZ512184A (en) 2003-08-29
US7098201B2 (en) 2006-08-29
KR20010089708A (ko) 2001-10-08
BR9916583A (pt) 2001-09-25
TR200101886T2 (tr) 2001-12-21
IL143958A0 (en) 2002-04-21
RU2001120016A (ru) 2003-12-10
EP1142872A4 (en) 2002-04-17
CN1178913C (zh) 2004-12-08
ATE411286T1 (de) 2008-10-15
AU1797900A (en) 2000-07-31
NO20013179D0 (no) 2001-06-22
AU763040B2 (en) 2003-07-10
EP1142872A1 (en) 2001-10-10
US6645956B1 (en) 2003-11-11
HUP0201472A3 (en) 2006-03-28
CZ20012160A3 (cs) 2001-10-17
CA2353961A1 (en) 2000-07-06
US20040002485A1 (en) 2004-01-01
CN1335834A (zh) 2002-02-13

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