NL8201022A - Azaspiroalkaandionen; werkwijze voor het bereiden daarvan; farmaceutische preparaten; werkwijze voor het oproepen van een tranquilizereffect. - Google Patents

Azaspiroalkaandionen; werkwijze voor het bereiden daarvan; farmaceutische preparaten; werkwijze voor het oproepen van een tranquilizereffect. Download PDF

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Publication number
NL8201022A
NL8201022A NL8201022A NL8201022A NL8201022A NL 8201022 A NL8201022 A NL 8201022A NL 8201022 A NL8201022 A NL 8201022A NL 8201022 A NL8201022 A NL 8201022A NL 8201022 A NL8201022 A NL 8201022A
Authority
NL
Netherlands
Prior art keywords
formula
pharmaceutically acceptable
compound
butyl
acid addition
Prior art date
Application number
NL8201022A
Other languages
English (en)
Dutch (nl)
Original Assignee
Bristol Myers Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bristol Myers Co filed Critical Bristol Myers Co
Publication of NL8201022A publication Critical patent/NL8201022A/nl

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D221/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00
    • C07D221/02—Heterocyclic compounds containing six-membered rings having one nitrogen atom as the only ring hetero atom, not provided for by groups C07D211/00 - C07D219/00 condensed with carbocyclic rings or ring systems
    • C07D221/20—Spiro-condensed ring systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/20—Hypnotics; Sedatives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/26—Psychostimulants, e.g. nicotine, cocaine

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Public Health (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Psychiatry (AREA)
  • Pain & Pain Management (AREA)
  • Anesthesiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Other In-Based Heterocyclic Compounds (AREA)
  • Indole Compounds (AREA)
NL8201022A 1981-03-16 1982-03-11 Azaspiroalkaandionen; werkwijze voor het bereiden daarvan; farmaceutische preparaten; werkwijze voor het oproepen van een tranquilizereffect. NL8201022A (nl)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US24442681 1981-03-16
US06/244,426 US4320131A (en) 1981-03-16 1981-03-16 N-[(4-Phenyl-1,2,3,6-tetrahydropyridin-1-yl)alkylene]azaspiroalkanediones and N-[(4-hydroxy-4-phenylpiperidin-1-yl)alkylene]azaspiroalkanediones

Publications (1)

Publication Number Publication Date
NL8201022A true NL8201022A (nl) 1982-10-18

Family

ID=22922718

Family Applications (1)

Application Number Title Priority Date Filing Date
NL8201022A NL8201022A (nl) 1981-03-16 1982-03-11 Azaspiroalkaandionen; werkwijze voor het bereiden daarvan; farmaceutische preparaten; werkwijze voor het oproepen van een tranquilizereffect.

Country Status (31)

Country Link
US (1) US4320131A (fr)
JP (1) JPS57165384A (fr)
KR (1) KR880001557B1 (fr)
AT (1) AT381939B (fr)
AU (1) AU535385B2 (fr)
BE (1) BE892502A (fr)
CA (1) CA1192556A (fr)
CH (2) CH652123A5 (fr)
CY (1) CY1372A (fr)
DE (1) DE3209534A1 (fr)
DK (1) DK161322C (fr)
ES (1) ES8305753A1 (fr)
FI (1) FI71317C (fr)
FR (1) FR2501689B1 (fr)
GB (1) GB2094801B (fr)
GR (1) GR76113B (fr)
HK (1) HK4688A (fr)
HU (2) HU193379B (fr)
IE (1) IE52789B1 (fr)
IL (1) IL65254A0 (fr)
IT (1) IT1148145B (fr)
KE (1) KE3710A (fr)
LU (1) LU84012A1 (fr)
NL (1) NL8201022A (fr)
NZ (1) NZ199944A (fr)
PH (1) PH18182A (fr)
PT (1) PT74584B (fr)
SE (2) SE449100B (fr)
SG (1) SG30887G (fr)
YU (1) YU43789B (fr)
ZA (1) ZA821541B (fr)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2660407B2 (ja) * 1986-09-26 1997-10-08 住友製薬株式会社 新規なイミド誘導体
HU207310B (en) * 1988-12-02 1993-03-29 Pfizer Process for producing aryl-piperidine derivatives
US5137894A (en) * 1991-12-05 1992-08-11 New James S 4-(4-Piperidinyl-thieno[3,2-c]pyridine derivatives of n-alkylglutarimides

Family Cites Families (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US355877A (en) * 1887-01-11 Waltee n
FR3013E (fr) * 1902-04-03 1904-08-12 William Henry Hoyle Perfectionnements au procédé et aux machines pour la fabrication de matières fibreuses connues sous le nom de fils "frottés"
US3106552A (en) * 1960-07-19 1963-10-08 Geschickter Fund Med Res Nu-substituted azaspiranes and azaspirane-diones and processes for their preparation
US3432499A (en) * 1965-04-02 1969-03-11 Geschickter Fund Med Res Trifluoromethylazaspiranes and azaspirane diones
US3398151A (en) * 1966-02-01 1968-08-20 Mead Johnson & Co Azaspirodecanediones and azaspiroundecanediones
US3558777A (en) * 1968-06-21 1971-01-26 Mead Johnson & Co Pharmacologic processes and compositions containing azaspirodecanediones and azaspiroundecanediones
BE759371A (fr) * 1969-11-24 1971-05-24 Bristol Myers Co Azaspirodecanediones heterocycliques et procedes pour leur preparation
CH547802A (de) * 1970-06-19 1974-04-11 Hoffmann La Roche Verfahren zur herstellung von tetrahydropyridinderivaten.
US3976776A (en) * 1972-12-06 1976-08-24 Mead Johnson & Company Tranquilizer process employing N-(heteroarcyclic)piperazinylalkylazaspiroalkanediones
US4250175A (en) * 1977-10-31 1981-02-10 Mccall John M Methods of treating psychosis
US4179510A (en) * 1977-10-31 1979-12-18 The Upjohn Company Methods of treating psychosis
US4218456A (en) * 1978-07-10 1980-08-19 Warner-Lambert Company 1-(4-Fluorophenyl)-4-(1,2,3,6-tetrahydro-4-phenoxy-1-pyridinyl)-butanones
US4261990A (en) * 1979-03-09 1981-04-14 Ciba-Geigy Corporation N-alkyleneiminoalkyl-dicarboximides as antiallergics and antiasthmatics
US4221714A (en) * 1979-08-03 1980-09-09 American Cyanamid Company 11-(1,2,3,6-Tetrahydro-substituted-4-pyridyl)-dibenz[b,f][1,4]oxazepines
US4305944A (en) * 1980-09-08 1981-12-15 Mead Johnson & Company N-[(4-[3-cyano substituted pyridyl]piperazino)alkyl]-azaspirodecanediones

Also Published As

Publication number Publication date
CA1192556A (fr) 1985-08-27
DK161322C (da) 1991-12-09
IL65254A0 (en) 1982-05-31
LU84012A1 (fr) 1983-02-22
PH18182A (en) 1985-04-12
PT74584A (en) 1982-04-01
GB2094801B (en) 1985-04-24
ES510448A0 (es) 1983-04-16
US4320131A (en) 1982-03-16
CH652123A5 (de) 1985-10-31
AT381939B (de) 1986-12-10
HU190793B (en) 1986-11-28
KR830008680A (ko) 1983-12-14
FI820855L (fi) 1982-09-17
KR880001557B1 (ko) 1988-08-22
DE3209534A1 (de) 1982-09-23
PT74584B (pt) 1984-11-27
IE820590L (en) 1982-09-16
CY1372A (en) 1987-08-07
HK4688A (en) 1988-01-29
SE8201630L (sv) 1982-09-17
YU55882A (en) 1984-10-31
FI71317B (fi) 1986-09-09
GB2094801A (en) 1982-09-22
CH657365A5 (de) 1986-08-29
FR2501689B1 (fr) 1985-07-19
SE460606B (sv) 1989-10-30
IE52789B1 (en) 1988-03-02
SG30887G (en) 1987-07-17
AU8133582A (en) 1982-11-04
HU193379B (en) 1987-09-28
YU43789B (en) 1989-12-31
JPH0345072B2 (fr) 1991-07-09
DK112682A (da) 1982-09-17
ES8305753A1 (es) 1983-04-16
HUT40797A (en) 1987-02-27
NZ199944A (en) 1986-06-11
BE892502A (fr) 1982-09-15
AU535385B2 (en) 1984-03-15
IT1148145B (it) 1986-11-26
DE3209534C2 (fr) 1993-03-11
SE449100B (sv) 1987-04-06
FR2501689A1 (fr) 1982-09-17
SE8603177D0 (sv) 1986-07-21
ZA821541B (en) 1983-01-26
ATA104682A (de) 1986-05-15
JPS57165384A (en) 1982-10-12
IT8247992A0 (it) 1982-03-15
KE3710A (en) 1987-04-16
FI71317C (fi) 1986-12-19
GR76113B (fr) 1984-08-03
SE8603177L (sv) 1986-07-21
DK161322B (da) 1991-06-24

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Legal Events

Date Code Title Description
A85 Still pending on 85-01-01
BA A request for search or an international-type search has been filed
BB A search report has been drawn up
BC A request for examination has been filed
DNT Communications of changes of names of applicants whose applications have been laid open to public inspection

Free format text: BRISTOL-MYERS SQUIBB COMPANY

BV The patent application has lapsed