NL300105I2 - Nieuwe selectieve remstoffen van virale of bacteriële neuraminidasen. - Google Patents

Nieuwe selectieve remstoffen van virale of bacteriële neuraminidasen.

Info

Publication number
NL300105I2
NL300105I2 NL300105C NL300105C NL300105I2 NL 300105 I2 NL300105 I2 NL 300105I2 NL 300105 C NL300105 C NL 300105C NL 300105 C NL300105 C NL 300105C NL 300105 I2 NL300105 I2 NL 300105I2
Authority
NL
Netherlands
Prior art keywords
viral
selective inhibitors
neuraminidase
compounds
new selective
Prior art date
Application number
NL300105C
Other languages
English (en)
Dutch (nl)
Other versions
NL300105I1 (nl
Original Assignee
Gilead Sciences
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=27410155&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=NL300105(I2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Priority claimed from US08/476,946 external-priority patent/US5866601A/en
Application filed by Gilead Sciences filed Critical Gilead Sciences
Publication of NL300105I1 publication Critical patent/NL300105I1/nl
Publication of NL300105I2 publication Critical patent/NL300105I2/nl

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D309/00Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings
    • C07D309/16Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D309/28Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • A61P31/14Antivirals for RNA viruses
    • A61P31/16Antivirals for RNA viruses for influenza or rhinoviruses
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02PCLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00Technologies relating to chemical industry
    • Y02P20/50Improvements relating to the production of bulk chemicals
    • Y02P20/55Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Virology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Pulmonology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Molecular Biology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Saccharide Compounds (AREA)
  • Measuring Or Testing Involving Enzymes Or Micro-Organisms (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Heterocyclic Compounds That Contain Two Or More Ring Oxygen Atoms (AREA)
  • Pyrane Compounds (AREA)
  • Epoxy Compounds (AREA)
  • Pyridine Compounds (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Pyrrole Compounds (AREA)
  • Polyesters Or Polycarbonates (AREA)
NL300105C 1995-02-27 2002-10-29 Nieuwe selectieve remstoffen van virale of bacteriële neuraminidasen. NL300105I2 (nl)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US39524595A 1995-02-27 1995-02-27
US08/476,946 US5866601A (en) 1995-02-27 1995-06-06 Carbocyclic compounds
US58056795A 1995-12-29 1995-12-29
PCT/US1996/002882 WO1996026933A1 (en) 1995-02-27 1996-02-26 Novel selective inhibitors of viral or bacterial neuraminidases

Publications (2)

Publication Number Publication Date
NL300105I1 NL300105I1 (nl) 2003-01-06
NL300105I2 true NL300105I2 (nl) 2003-02-03

Family

ID=27410155

Family Applications (1)

Application Number Title Priority Date Filing Date
NL300105C NL300105I2 (nl) 1995-02-27 2002-10-29 Nieuwe selectieve remstoffen van virale of bacteriële neuraminidasen.

Country Status (26)

Country Link
US (3) US5952375A (enExample)
EP (1) EP0759917B1 (enExample)
JP (3) JP3300365B2 (enExample)
KR (1) KR100447096B1 (enExample)
CN (2) CN100409844C (enExample)
AT (2) ATE305453T1 (enExample)
AU (1) AU720933B2 (enExample)
BR (2) BR9607098B8 (enExample)
CZ (1) CZ297945B6 (enExample)
DE (4) DE759917T1 (enExample)
DK (1) DK0759917T3 (enExample)
ES (2) ES2118674T3 (enExample)
GR (1) GR3033914T3 (enExample)
HU (1) HU228450B1 (enExample)
LU (1) LU90991I2 (enExample)
MX (1) MX9706496A (enExample)
NL (1) NL300105I2 (enExample)
NO (1) NO318455B1 (enExample)
NZ (1) NZ306625A (enExample)
PL (1) PL194173B1 (enExample)
PT (1) PT759917E (enExample)
RU (1) RU2181357C2 (enExample)
SG (1) SG45864A1 (enExample)
SI (1) SI9620042A (enExample)
UA (1) UA56128C2 (enExample)
WO (1) WO1996026933A1 (enExample)

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CN1185223C (zh) 2005-01-19
PT759917E (pt) 2000-10-31
US6225341B1 (en) 2001-05-01
SI9620042A (sl) 1998-12-31
DE69607704D1 (de) 2000-05-18
JPH11501908A (ja) 1999-02-16
NO318455B1 (no) 2005-03-21
UA56128C2 (uk) 2003-05-15
NO973908D0 (no) 1997-08-26
US5952375A (en) 1999-09-14
BR9607098A (pt) 1997-11-04
BR9607098B8 (pt) 2014-11-18
HUP9800026A2 (hu) 1999-09-28
KR19980703600A (ko) 1998-12-05
EP0759917B1 (en) 2000-04-12
HUP9800026A3 (en) 2002-04-29
JP3300365B2 (ja) 2002-07-08
CZ297945B6 (cs) 2007-05-02
ES2118674T1 (es) 1998-10-01
DE69635231D1 (de) 2006-02-09
GR3033914T3 (en) 2000-11-30
CN1147813A (zh) 1997-04-16
DE69635231T2 (de) 2006-07-13
PL194173B1 (pl) 2007-05-31
HU228450B1 (en) 2013-03-28
DK0759917T3 (da) 2000-07-31
AU5357196A (en) 1996-09-18
HK1026893A1 (en) 2000-12-29
JP2006036770A (ja) 2006-02-09
CZ269097A3 (en) 1997-11-12
CN1347693A (zh) 2002-05-08
NL300105I1 (nl) 2003-01-06
ES2249863T3 (es) 2006-04-01
ATE305453T1 (de) 2005-10-15
DE69607704T2 (de) 2000-12-28
DE10299052I1 (de) 2003-05-22
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ES2118674T3 (es) 2000-08-16
MX9706496A (es) 1997-11-29
PL322000A1 (en) 1998-01-05
NZ306625A (en) 2001-04-27
LU90991I2 (fr) 2003-02-11
ATE191711T1 (de) 2000-04-15
EP0759917A1 (en) 1997-03-05
JP4234917B2 (ja) 2009-03-04
DE759917T1 (de) 1998-10-22
NO973908L (no) 1997-10-27
CN100409844C (zh) 2008-08-13
KR100447096B1 (ko) 2005-10-11
WO1996026933A1 (en) 1996-09-06
US20050176758A1 (en) 2005-08-11
JP2002161074A (ja) 2002-06-04

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