NL300105I2 - Nieuwe selectieve remstoffen van virale of bacteriële neuraminidasen. - Google Patents
Nieuwe selectieve remstoffen van virale of bacteriële neuraminidasen.Info
- Publication number
- NL300105I2 NL300105I2 NL300105C NL300105C NL300105I2 NL 300105 I2 NL300105 I2 NL 300105I2 NL 300105 C NL300105 C NL 300105C NL 300105 C NL300105 C NL 300105C NL 300105 I2 NL300105 I2 NL 300105I2
- Authority
- NL
- Netherlands
- Prior art keywords
- viral
- selective inhibitors
- neuraminidase
- compounds
- new selective
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D309/00—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings
- C07D309/16—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
- C07D309/28—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A61P31/14—Antivirals for RNA viruses
- A61P31/16—Antivirals for RNA viruses for influenza or rhinoviruses
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups
Landscapes
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Virology (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- General Chemical & Material Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Oncology (AREA)
- Communicable Diseases (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pulmonology (AREA)
- Molecular Biology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Saccharide Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Measuring Or Testing Involving Enzymes Or Micro-Organisms (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Epoxy Compounds (AREA)
- Heterocyclic Compounds That Contain Two Or More Ring Oxygen Atoms (AREA)
- Preparation Of Compounds By Using Micro-Organisms (AREA)
- Polyesters Or Polycarbonates (AREA)
- Pyrane Compounds (AREA)
Applications Claiming Priority (4)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US39524595A | 1995-02-27 | 1995-02-27 | |
US08/476,946 US5866601A (en) | 1995-02-27 | 1995-06-06 | Carbocyclic compounds |
US58056795A | 1995-12-29 | 1995-12-29 | |
PCT/US1996/002882 WO1996026933A1 (en) | 1995-02-27 | 1996-02-26 | Novel selective inhibitors of viral or bacterial neuraminidases |
Publications (2)
Publication Number | Publication Date |
---|---|
NL300105I1 NL300105I1 (nl) | 2003-01-06 |
NL300105I2 true NL300105I2 (nl) | 2003-02-03 |
Family
ID=27410155
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
NL300105C NL300105I2 (nl) | 1995-02-27 | 2002-10-29 | Nieuwe selectieve remstoffen van virale of bacteriële neuraminidasen. |
Country Status (27)
Country | Link |
---|---|
US (3) | US5952375A (nl) |
EP (1) | EP0759917B1 (nl) |
JP (3) | JP3300365B2 (nl) |
KR (1) | KR100447096B1 (nl) |
CN (2) | CN1185223C (nl) |
AT (2) | ATE191711T1 (nl) |
AU (1) | AU720933B2 (nl) |
BR (2) | BR9607098B8 (nl) |
CZ (1) | CZ297945B6 (nl) |
DE (4) | DE10299052I1 (nl) |
DK (1) | DK0759917T3 (nl) |
ES (2) | ES2249863T3 (nl) |
GR (1) | GR3033914T3 (nl) |
HK (1) | HK1026893A1 (nl) |
HU (1) | HU228450B1 (nl) |
LU (1) | LU90991I2 (nl) |
MX (1) | MX9706496A (nl) |
NL (1) | NL300105I2 (nl) |
NO (1) | NO318455B1 (nl) |
NZ (1) | NZ306625A (nl) |
PL (1) | PL194173B1 (nl) |
PT (1) | PT759917E (nl) |
RU (1) | RU2181357C2 (nl) |
SG (1) | SG45864A1 (nl) |
SI (1) | SI9620042A (nl) |
UA (1) | UA56128C2 (nl) |
WO (1) | WO1996026933A1 (nl) |
Families Citing this family (85)
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US20040053999A1 (en) * | 1997-09-17 | 2004-03-18 | Bischofberger Norbert W. | Novel compounds and methods for synthesis and therapy |
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GB9325841D0 (en) * | 1993-12-17 | 1994-02-23 | Glaxo Group Ltd | Chemical compounds |
GB9400206D0 (en) * | 1994-01-07 | 1994-03-02 | Glaxo Group Ltd | Chemical compound |
AUPM354694A0 (en) * | 1994-01-27 | 1994-02-17 | Biota Scientific Management Pty Ltd | Chemical compounds |
US5985859A (en) * | 1994-04-14 | 1999-11-16 | The University Of Alabama | Methods of inhibiting bacterial sialidase |
GB9410817D0 (en) * | 1994-05-28 | 1994-07-20 | Glaxo Group Ltd | Medicaments |
AUPM725794A0 (en) * | 1994-08-03 | 1994-08-25 | Biota Scientific Management Pty Ltd | Chemical compounds |
US5556963A (en) * | 1994-08-05 | 1996-09-17 | Oklahoma Medical Research Foundation | Synthesis of 4-alkoxy-N-acetylneuraminic acid |
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AU710492B2 (en) | 1994-11-04 | 1999-09-23 | Gilead Sciences, Inc. | Thiepane compounds inhibiting and detecting HIV protease |
US5866601A (en) * | 1995-02-27 | 1999-02-02 | Gilead Sciences, Inc. | Carbocyclic compounds |
SI9620042A (sl) * | 1995-02-27 | 1998-12-31 | Gilead Sciences, Inc. | Novi selektivni inhibitorji virusnih ali bakterijskih neuraminidaz |
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US5714509A (en) * | 1995-05-03 | 1998-02-03 | The University Of Alabama | Inhibitors of bacterial sialidase and methods of making and using the same |
GB9525389D0 (en) | 1995-12-12 | 1996-02-14 | Biota Scient Management Ltd | Chemical compounds |
GB9510141D0 (en) | 1995-05-19 | 1995-07-12 | Biota Scient Management | Chemical compounds |
CN1184473A (zh) * | 1995-05-19 | 1998-06-10 | 比奥塔科学管理有限公司 | 6-羟基酰胺-二氢吡喃衍生物 |
GB9516276D0 (en) * | 1995-08-08 | 1995-10-11 | Biota Scient Management | Chemical compounds |
US5763483A (en) * | 1995-12-29 | 1998-06-09 | Gilead Sciences, Inc. | Carbocyclic compounds |
US5859284A (en) | 1996-08-23 | 1999-01-12 | Gilead Sciences, Inc. | Preparation of carbocyclic compounds |
EP0920410B1 (en) | 1996-08-23 | 2002-03-27 | Gilead Sciences, Inc. | Preparation of cyclohexene carboxylate derivatives |
US5948816A (en) * | 1996-09-10 | 1999-09-07 | Daikin Industries, Ltd. | 4-substituted-2,7-dideoxy-7-fluoro-2,3-didehydro-sialic acid compounds |
US5886213A (en) | 1997-08-22 | 1999-03-23 | Gilead Sciences, Inc. | Preparation of carbocyclic compounds |
-
1996
- 1996-02-26 SI SI9620042A patent/SI9620042A/sl not_active IP Right Cessation
- 1996-02-26 BR BRPI9607098-6B8D patent/BR9607098B8/pt unknown
- 1996-02-26 CZ CZ0269097A patent/CZ297945B6/cs not_active IP Right Cessation
- 1996-02-26 DE DE2002199052 patent/DE10299052I1/de active Pending
- 1996-02-26 AU AU53571/96A patent/AU720933B2/en not_active Expired
- 1996-02-26 JP JP52644296A patent/JP3300365B2/ja not_active Expired - Lifetime
- 1996-02-26 HU HU9800026A patent/HU228450B1/hu unknown
- 1996-02-26 BR BR9607098A patent/BR9607098A/pt not_active IP Right Cessation
- 1996-02-26 ES ES99117934T patent/ES2249863T3/es not_active Expired - Lifetime
- 1996-02-26 SG SG1997004840A patent/SG45864A1/en unknown
- 1996-02-26 AT AT96912404T patent/ATE191711T1/de active
- 1996-02-26 CN CNB961901330A patent/CN1185223C/zh not_active Expired - Lifetime
- 1996-02-26 NZ NZ306625A patent/NZ306625A/xx not_active IP Right Cessation
- 1996-02-26 MX MX9706496A patent/MX9706496A/es unknown
- 1996-02-26 PL PL96322000A patent/PL194173B1/pl unknown
- 1996-02-26 KR KR1019970705932A patent/KR100447096B1/ko not_active IP Right Cessation
- 1996-02-26 DK DK96912404T patent/DK0759917T3/da active
- 1996-02-26 DE DE0759917T patent/DE759917T1/de active Pending
- 1996-02-26 PT PT96912404T patent/PT759917E/pt unknown
- 1996-02-26 ES ES96912404T patent/ES2118674T3/es not_active Expired - Lifetime
- 1996-02-26 DE DE69635231T patent/DE69635231T2/de not_active Expired - Lifetime
- 1996-02-26 UA UA97094796A patent/UA56128C2/uk unknown
- 1996-02-26 RU RU97116714/04A patent/RU2181357C2/ru active
- 1996-02-26 US US08/606,624 patent/US5952375A/en not_active Expired - Lifetime
- 1996-02-26 AT AT99117934T patent/ATE305453T1/de active
- 1996-02-26 EP EP96912404A patent/EP0759917B1/en not_active Expired - Lifetime
- 1996-02-26 WO PCT/US1996/002882 patent/WO1996026933A1/en active IP Right Grant
- 1996-02-26 CN CNB011247142A patent/CN100409844C/zh not_active Expired - Lifetime
- 1996-02-26 DE DE69607704T patent/DE69607704T2/de not_active Expired - Lifetime
- 1996-05-24 US US08/653,034 patent/US20050176758A1/en not_active Abandoned
-
1997
- 1997-08-26 NO NO19973908A patent/NO318455B1/no not_active IP Right Cessation
-
1999
- 1999-04-08 US US09/288,091 patent/US6225341B1/en not_active Expired - Lifetime
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2000
- 2000-07-07 GR GR20000401599T patent/GR3033914T3/el unknown
- 2000-08-02 HK HK00104830A patent/HK1026893A1/xx not_active IP Right Cessation
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2001
- 2001-08-24 JP JP2001255372A patent/JP4234917B2/ja not_active Expired - Lifetime
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2002
- 2002-10-29 NL NL300105C patent/NL300105I2/nl unknown
- 2002-12-11 LU LU90991C patent/LU90991I2/fr unknown
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2005
- 2005-07-15 JP JP2005207906A patent/JP2006036770A/ja not_active Withdrawn
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