NL194616C - Werkwijze voor het winnen van een (2R,3S)-3-(4-methoxyfenyl)- glycidinezuur ester. - Google Patents

Werkwijze voor het winnen van een (2R,3S)-3-(4-methoxyfenyl)- glycidinezuur ester. Download PDF

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Publication number
NL194616C
NL194616C NL9100854A NL9100854A NL194616C NL 194616 C NL194616 C NL 194616C NL 9100854 A NL9100854 A NL 9100854A NL 9100854 A NL9100854 A NL 9100854A NL 194616 C NL194616 C NL 194616C
Authority
NL
Netherlands
Prior art keywords
methoxyphenyl
ester
glycidic acid
trans
mixture
Prior art date
Application number
NL9100854A
Other languages
English (en)
Dutch (nl)
Other versions
NL194616B (nl
NL9100854A (nl
Inventor
Claudio Giordano
Luca Ghirotto
Stefano Servi
Claudio Fuganti
Angelo Gentile
Original Assignee
Zambon Spa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Zambon Spa filed Critical Zambon Spa
Publication of NL9100854A publication Critical patent/NL9100854A/nl
Publication of NL194616B publication Critical patent/NL194616B/xx
Application granted granted Critical
Publication of NL194616C publication Critical patent/NL194616C/nl

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D407/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen atoms as the only ring hetero atoms, not provided for by group C07D405/00
    • C07D407/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen atoms as the only ring hetero atoms, not provided for by group C07D405/00 containing two hetero rings
    • C07D407/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen atoms as the only ring hetero atoms, not provided for by group C07D405/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D281/00—Heterocyclic compounds containing rings of more than six members having one nitrogen atom and one sulfur atom as the only ring hetero atoms
    • C07D281/02—Seven-membered rings
    • C07D281/04—Seven-membered rings having the hetero atoms in positions 1 and 4
    • C07D281/08—Seven-membered rings having the hetero atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
    • C07D281/10—Seven-membered rings having the hetero atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems condensed with one six-membered ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D303/00—Compounds containing three-membered rings having one oxygen atom as the only ring hetero atom
    • C07D303/02—Compounds containing oxirane rings
    • C07D303/48—Compounds containing oxirane rings with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms, e.g. ester or nitrile radicals
    • C—CHEMISTRY; METALLURGY
    • C12—BIOCHEMISTRY; BEER; SPIRITS; WINE; VINEGAR; MICROBIOLOGY; ENZYMOLOGY; MUTATION OR GENETIC ENGINEERING
    • C12P—FERMENTATION OR ENZYME-USING PROCESSES TO SYNTHESISE A DESIRED CHEMICAL COMPOUND OR COMPOSITION OR TO SEPARATE OPTICAL ISOMERS FROM A RACEMIC MIXTURE
    • C12P17/00—Preparation of heterocyclic carbon compounds with only O, N, S, Se or Te as ring hetero atoms
    • C12P17/02—Oxygen as only ring hetero atoms
    • C—CHEMISTRY; METALLURGY
    • C12—BIOCHEMISTRY; BEER; SPIRITS; WINE; VINEGAR; MICROBIOLOGY; ENZYMOLOGY; MUTATION OR GENETIC ENGINEERING
    • C12P—FERMENTATION OR ENZYME-USING PROCESSES TO SYNTHESISE A DESIRED CHEMICAL COMPOUND OR COMPOSITION OR TO SEPARATE OPTICAL ISOMERS FROM A RACEMIC MIXTURE
    • C12P41/00—Processes using enzymes or microorganisms to separate optical isomers from a racemic mixture
    • C12P41/003—Processes using enzymes or microorganisms to separate optical isomers from a racemic mixture by ester formation, lactone formation or the inverse reactions
    • C12P41/005—Processes using enzymes or microorganisms to separate optical isomers from a racemic mixture by ester formation, lactone formation or the inverse reactions by esterification of carboxylic acid groups in the enantiomers or the inverse reaction

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Wood Science & Technology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Zoology (AREA)
  • Health & Medical Sciences (AREA)
  • General Engineering & Computer Science (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Biotechnology (AREA)
  • Biochemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Microbiology (AREA)
  • General Health & Medical Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Analytical Chemistry (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Epoxy Compounds (AREA)
NL9100854A 1990-05-17 1991-05-16 Werkwijze voor het winnen van een (2R,3S)-3-(4-methoxyfenyl)- glycidinezuur ester. NL194616C (nl)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
IT2034890 1990-05-17
IT02034890A IT1249777B (it) 1990-05-17 1990-05-17 Processo per la preparazione di intermedi per la sintesi del diltiazem

Publications (3)

Publication Number Publication Date
NL9100854A NL9100854A (nl) 1991-12-16
NL194616B NL194616B (nl) 2002-05-01
NL194616C true NL194616C (nl) 2002-09-03

Family

ID=11165937

Family Applications (1)

Application Number Title Priority Date Filing Date
NL9100854A NL194616C (nl) 1990-05-17 1991-05-16 Werkwijze voor het winnen van een (2R,3S)-3-(4-methoxyfenyl)- glycidinezuur ester.

Country Status (13)

Country Link
US (2) US5571704A (ja)
JP (2) JP3060187B2 (ja)
AT (1) AT400446B (ja)
BE (1) BE1005406A0 (ja)
CA (1) CA2042535C (ja)
CH (1) CH682670A5 (ja)
DE (1) DE4115697C2 (ja)
ES (1) ES2033203B1 (ja)
FR (1) FR2662178B1 (ja)
GB (2) GB2246351B (ja)
IT (1) IT1249777B (ja)
NL (1) NL194616C (ja)
SE (1) SE509297C2 (ja)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2687789B2 (ja) * 1991-08-13 1997-12-08 田辺製薬株式会社 光学活性３−フェニルグリシッド酸エステル類化合物の製法
ES2050067B1 (es) * 1992-06-08 1994-12-16 Menarini Lab Proceso para la produccion de acido s-(+)-2-(3-benzoilfenil) propionico por transesterificacion enantioselectiva con un alcohol bifuncional catalizada enzimaticamente en medio organico.
ES2048653B1 (es) * 1992-06-08 1994-12-16 Menarini Lab Proceso para la produccion de acido s-(+)-2-(3-benzoilfenil) propionico por transesterificacion enantioselectiva catalizada enzimaticamente en un disolvente organico.
US6020174A (en) * 1992-07-27 2000-02-01 The Board Of Governors For Higher Education Chemoenzymatic synthesis of the taxol C-13 side chain N-benzolyl- (2R,3S)-Phenylisoserine
DE4225155C1 (ja) * 1992-07-30 1993-08-05 Hoechst Ag, 6230 Frankfurt, De
SG72731A1 (en) * 1996-03-15 2000-05-23 Nabe Seiyaku Co Ltd Process for preparing optically active trans-3-phenylglycidamide compounds
TW438787B (en) * 1997-02-27 2001-06-07 Tanabe Seiyaku Co Process for preparing optically active trans-3-substituted glycidic acid ester
AU7551998A (en) * 1997-06-11 1998-12-30 Tanabe Seiyaku Co., Ltd. Process for preparing optically active phenyloxirane compounds
IT1302261B1 (it) 1998-09-24 2000-09-05 Zambon Spa Processo per la risoluzione cinetica enzimatica di 3-fenilglicidatiper transesterificazione con amminoalcoli
DE19901925A1 (de) * 1999-01-19 2000-07-27 Aventis Res & Tech Gmbh & Co Verfahren zur Trennung optischer Isomerer durch simultane Durchführung einer enzymatischen Reaktion und einer chromatographischen Trennung
WO2003066873A1 (en) * 2002-02-06 2003-08-14 Commonwealth Scientific And Industrial Research Organisation Esterases with lipase activity
TWM583351U (zh) 2019-05-10 2019-09-11 北聯研磨科技股份有限公司 砂輪中心孔保護墊

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NL8801311A (nl) * 1988-05-20 1989-12-18 Stamicarbon Fenylglycidaatstereoisomeren, omzettingsprodukten daarvan met 2-nitrothiofenol en de bereiding van diltiazem.
IT1217765B (it) * 1988-06-02 1990-03-30 Montedison Spa Processo per la risoluzione enzimatica degli isomeri ottici di derivati racemi esterei dell,acido 3 mercapto 2 alchilpropionico
FI95931C (fi) * 1988-09-02 1996-04-10 Tanabe Seiyaku Co Menetelmä (2R,3S)-3-(4-metoksifenyyli)glysidiinihapon alemman alkyyliesterin valmistamiseksi
DE3833774C1 (ja) * 1988-10-05 1990-04-26 Fischer-Werke Artur Fischer Gmbh & Co Kg, 7244 Waldachtal, De
US5108916A (en) * 1989-06-05 1992-04-28 Rhone-Poulenc Rorer, S.A. Process for stereoselectively hydrolyzing, transesterifying or esterifying with immobilized isozyme of lipase from candida rugosa
US5244803A (en) * 1989-09-13 1993-09-14 Tanabe Seiyaku Co., Ltd. Process for preparing optically active 3-phenylglycidic acid esters
JPH0779706B2 (ja) * 1990-03-22 1995-08-30 田辺製薬株式会社 ２―クロロ―３―ヒドロキシ―３―フエニルプロピオン酸エステル類の製法
IT1240651B (it) * 1990-05-17 1993-12-17 Zambon Spa Processo per la risoluzione di derivati glicidici
FR2672600B1 (fr) * 1991-02-08 1994-10-14 Synthelabo Procede de preparation du (-)-(2r,3s)-2,3-epoxy-3-(4-methoxyphenyl) propionate de methyle.
NL9202208A (nl) * 1992-12-18 1994-07-18 Dsm Nv Werkwijze voor de enzymatische bereiding van optisch aktieve glycidezure esters.

Also Published As

Publication number Publication date
GB2246351B (en) 1993-12-15
SE9101482D0 (sv) 1991-05-16
JP2000139492A (ja) 2000-05-23
BE1005406A0 (fr) 1993-07-13
IT1249777B (it) 1995-03-18
FR2662178B1 (fr) 1995-05-05
JPH04228095A (ja) 1992-08-18
DE4115697C2 (de) 2000-09-07
DE4115697A1 (de) 1991-11-21
ES2033203A1 (es) 1993-03-01
IT9020348A0 (it) 1990-05-17
JP3223317B2 (ja) 2001-10-29
GB9120710D0 (en) 1991-11-13
GB2247020B (en) 1993-12-15
CH682670A5 (it) 1993-10-29
GB2246351A (en) 1992-01-29
GB9110610D0 (en) 1991-07-03
CA2042535C (en) 1998-06-16
AT400446B (de) 1995-12-27
GB2247020A (en) 1992-02-19
CA2042535A1 (en) 1991-11-18
NL194616B (nl) 2002-05-01
IT9020348A1 (it) 1991-11-17
FR2662178A1 (fr) 1991-11-22
JP3060187B2 (ja) 2000-07-10
SE509297C2 (sv) 1999-01-11
ES2033203B1 (es) 1993-12-16
SE9101482L (sv) 1991-11-18
NL9100854A (nl) 1991-12-16
US5571704A (en) 1996-11-05
US6346632B1 (en) 2002-02-12
ATA99591A (de) 1995-05-15

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BB A search report has been drawn up
BC A request for examination has been filed
V1 Lapsed because of non-payment of the annual fee

Effective date: 20051201