MXPA05003084A - Nuevos compuestos para la inhibicion de rotamasas y usos de los mismos. - Google Patents

Nuevos compuestos para la inhibicion de rotamasas y usos de los mismos.

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Publication number
MXPA05003084A
MXPA05003084A MXPA05003084A MXPA05003084A MXPA05003084A MX PA05003084 A MXPA05003084 A MX PA05003084A MX PA05003084 A MXPA05003084 A MX PA05003084A MX PA05003084 A MXPA05003084 A MX PA05003084A MX PA05003084 A MXPA05003084 A MX PA05003084A
Authority
MX
Mexico
Prior art keywords
phenyl
hydroxy
chloro
phenol
urea
Prior art date
Application number
MXPA05003084A
Other languages
English (en)
Spanish (es)
Inventor
Osterkamp Frank
Original Assignee
Jerini Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Jerini Ag filed Critical Jerini Ag
Publication of MXPA05003084A publication Critical patent/MXPA05003084A/es

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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/13—Amines
    • A61K31/155—Amidines (), e.g. guanidine (H2N—C(=NH)—NH2), isourea (N=C(OH)—NH2), isothiourea (—N=C(SH)—NH2)
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
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    • C07C275/28—Derivatives of urea, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups having nitrogen atoms of urea groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton
    • C07C275/32—Derivatives of urea, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups having nitrogen atoms of urea groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton being further substituted by singly-bound oxygen atoms
    • C07C275/34—Derivatives of urea, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups having nitrogen atoms of urea groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton being further substituted by singly-bound oxygen atoms having nitrogen atoms of urea groups and singly-bound oxygen atoms bound to carbon atoms of the same non-condensed six-membered aromatic ring
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    • A61K31/17—Amides, e.g. hydroxamic acids having the group >N—C(O)—N< or >N—C(S)—N<, e.g. urea, thiourea, carmustine
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  • Public Health (AREA)
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  • Animal Behavior & Ethology (AREA)
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  • Dermatology (AREA)
  • Cardiology (AREA)
  • Diabetes (AREA)
  • Psychology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
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MXPA05003084A 2002-09-18 2003-09-18 Nuevos compuestos para la inhibicion de rotamasas y usos de los mismos. MXPA05003084A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP20020020987 EP1402888A1 (en) 2002-09-18 2002-09-18 The use of substituted carbocyclic compounds as rotamases inhibitors
PCT/EP2003/010406 WO2004026815A2 (en) 2002-09-18 2003-09-18 Phenol derivatives and their use as rotamase inhibitors

Publications (1)

Publication Number Publication Date
MXPA05003084A true MXPA05003084A (es) 2005-11-17

Family

ID=31970282

Family Applications (1)

Application Number Title Priority Date Filing Date
MXPA05003084A MXPA05003084A (es) 2002-09-18 2003-09-18 Nuevos compuestos para la inhibicion de rotamasas y usos de los mismos.

Country Status (14)

Country Link
US (2) US20070054904A1 (enExample)
EP (3) EP1402888A1 (enExample)
JP (2) JP2005539072A (enExample)
KR (1) KR20050053673A (enExample)
CN (1) CN100546977C (enExample)
AU (1) AU2003271619A1 (enExample)
BR (1) BR0314544A (enExample)
CA (1) CA2498662A1 (enExample)
MX (1) MXPA05003084A (enExample)
PL (1) PL374846A1 (enExample)
RU (2) RU2005111256A (enExample)
SG (1) SG165995A1 (enExample)
WO (1) WO2004026815A2 (enExample)
ZA (1) ZA200501913B (enExample)

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WO2004071447A2 (en) * 2003-02-12 2004-08-26 Transtech Pharma Inc. Substituted azole derivatives as therapeutic agents
EP1608319A4 (en) 2003-04-03 2007-02-28 Univ California IMPROVED HEMMER FOR SOLUBLE EPOXY HYDROLASE
AU2004303461B2 (en) * 2003-12-23 2011-04-28 H. Lundbeck A/S 2-(1H-indolylsulfanyl)-benzyl amine derivatives as SSRI
EP1713780B1 (en) * 2004-02-05 2012-01-18 Probiodrug AG Novel inhibitors of glutaminyl cyclase
CA2559665A1 (en) 2004-03-16 2005-09-29 The Regents Of The University Of California Reducing nephropathy with inhibitors of soluble epoxide hydrolase and epoxyeicosanoids
KR20070011475A (ko) * 2004-05-12 2007-01-24 쉐링 코포레이션 Ｃｘｃｒ1 및 ｃｘｃｒ2 케모카인 길항제
US7550499B2 (en) 2004-05-12 2009-06-23 Bristol-Myers Squibb Company Urea antagonists of P2Y1 receptor useful in the treatment of thrombotic conditions
AR052308A1 (es) * 2004-07-16 2007-03-14 Lundbeck & Co As H Derivados de 2-(1h-indolilsulfanil)-arilamina y una composicion farmaceutica que contiene al compuesto
CN101084216B (zh) 2004-10-20 2011-09-14 加利福尼亚大学董事会 可溶性环氧化物水解酶的改进抑制剂
AU2006206611A1 (en) 2005-01-19 2006-07-27 Bristol-Myers Squibb Company 2-phenoxy-N- (1, 3 , 4-thiadizol-2-yl) pyridin-3-amine derivatives and related compounds as P2Y1 receptor inhibitors for the treatment of thromboembolic disorders
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