AU2003271619A1 - Phenol derivatives and their use as rotamase inhibitors - Google Patents

Phenol derivatives and their use as rotamase inhibitors Download PDF

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Publication number
AU2003271619A1
AU2003271619A1 AU2003271619A AU2003271619A AU2003271619A1 AU 2003271619 A1 AU2003271619 A1 AU 2003271619A1 AU 2003271619 A AU2003271619 A AU 2003271619A AU 2003271619 A AU2003271619 A AU 2003271619A AU 2003271619 A1 AU2003271619 A1 AU 2003271619A1
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Australia
Prior art keywords
phenyl
hydroxy
chloro
urea
benzylamino
Prior art date
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Abandoned
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AU2003271619A
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English (en)
Inventor
Claudia Christner
Christoph Gibson
Gerd Hummel
Laurence Jobron
Jochen Knolle
Frank Osterkamp
Dirk Scharn
Mike Schutkowski
Roland Stragies
Thomas Tradler
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Jerini AG
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Jerini AG
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Publication of AU2003271619A1 publication Critical patent/AU2003271619A1/en
Abandoned legal-status Critical Current

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    • C07C275/34—Derivatives of urea, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups having nitrogen atoms of urea groups bound to carbon atoms of six-membered aromatic rings of a carbon skeleton being further substituted by singly-bound oxygen atoms having nitrogen atoms of urea groups and singly-bound oxygen atoms bound to carbon atoms of the same non-condensed six-membered aromatic ring
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AU2003271619A 2002-09-18 2003-09-18 Phenol derivatives and their use as rotamase inhibitors Abandoned AU2003271619A1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP20020020987 EP1402888A1 (en) 2002-09-18 2002-09-18 The use of substituted carbocyclic compounds as rotamases inhibitors
EP02020987.0 2002-09-18
PCT/EP2003/010406 WO2004026815A2 (en) 2002-09-18 2003-09-18 Phenol derivatives and their use as rotamase inhibitors

Publications (1)

Publication Number Publication Date
AU2003271619A1 true AU2003271619A1 (en) 2004-04-08

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ID=31970282

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Application Number Title Priority Date Filing Date
AU2003271619A Abandoned AU2003271619A1 (en) 2002-09-18 2003-09-18 Phenol derivatives and their use as rotamase inhibitors

Country Status (14)

Country Link
US (2) US20070054904A1 (enExample)
EP (3) EP1402888A1 (enExample)
JP (2) JP2005539072A (enExample)
KR (1) KR20050053673A (enExample)
CN (1) CN100546977C (enExample)
AU (1) AU2003271619A1 (enExample)
BR (1) BR0314544A (enExample)
CA (1) CA2498662A1 (enExample)
MX (1) MXPA05003084A (enExample)
PL (1) PL374846A1 (enExample)
RU (2) RU2005111256A (enExample)
SG (1) SG165995A1 (enExample)
WO (1) WO2004026815A2 (enExample)
ZA (1) ZA200501913B (enExample)

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AU2004210711B2 (en) * 2003-02-12 2010-07-08 Transtech Pharma, Inc. Substituted azole derivatives as therapeutic agents
WO2004089296A2 (en) 2003-04-03 2004-10-21 The Regents Of The University Of California Improved inhibitors for the soluble epoxide hydrolase
EP1701940B1 (en) * 2003-12-23 2008-05-28 H.Lundbeck A/S 2-(1h-indolylsulfanyl)-benzyl amine derivatives as ssri
WO2005075436A2 (en) * 2004-02-05 2005-08-18 Probiodrug Ag Novel inhibitors of glutaminyl cyclase
EP1765311A4 (en) 2004-03-16 2009-04-29 Univ California REDUCTION OF NEPHROPATHY WITH INHIBITORS OF SOLUBLE EPOXY HYDROLASE AND EPOXYEICOSANOIDS
CN1984899B (zh) * 2004-05-12 2011-07-27 先灵公司 Cxcr1和cxcr2趋化因子拮抗剂
US7550499B2 (en) 2004-05-12 2009-06-23 Bristol-Myers Squibb Company Urea antagonists of P2Y1 receptor useful in the treatment of thrombotic conditions
AR052308A1 (es) * 2004-07-16 2007-03-14 Lundbeck & Co As H Derivados de 2-(1h-indolilsulfanil)-arilamina y una composicion farmaceutica que contiene al compuesto
WO2006045119A2 (en) * 2004-10-20 2006-04-27 The Regents Of The University Of California Improved inhibitors for the soluble epoxide hydrolase
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