MX358512B - Uso de (r)-7cloro-n-(quinuclidin-3-il) benzo[b] tiofeno-2-carboxamida o una sal farmacéuticamente aceptable de la misma para preparar una composición farmacéutica en el tratamiento de una disfunción cognitiva. - Google Patents

Uso de (r)-7cloro-n-(quinuclidin-3-il) benzo[b] tiofeno-2-carboxamida o una sal farmacéuticamente aceptable de la misma para preparar una composición farmacéutica en el tratamiento de una disfunción cognitiva.

Info

Publication number
MX358512B
MX358512B MX2014013491A MX2014013491A MX358512B MX 358512 B MX358512 B MX 358512B MX 2014013491 A MX2014013491 A MX 2014013491A MX 2014013491 A MX2014013491 A MX 2014013491A MX 358512 B MX358512 B MX 358512B
Authority
MX
Mexico
Prior art keywords
treating
maintaining
cognitive function
methods
improving cognitive
Prior art date
Application number
MX2014013491A
Other languages
English (en)
Other versions
MX2014013491A (es
Inventor
Koenig Gerhard
C Hilt Dana
Original Assignee
Forum Pharmaceuticals Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Forum Pharmaceuticals Inc filed Critical Forum Pharmaceuticals Inc
Publication of MX2014013491A publication Critical patent/MX2014013491A/es
Publication of MX358512B publication Critical patent/MX358512B/es

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/439—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom the ring forming part of a bridged ring system, e.g. quinuclidine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K2121/00—Preparations for use in therapy

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Hospice & Palliative Care (AREA)
  • Psychiatry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

Un método de administración de una cantidad efectiva de (R)-7-cloro-N-(quinuclidin-3-il) benzo[b]tiofeno-2-carboxamida, o una sal farmacéuticamente aceptable de la misma, a un paciente que necesita de la misma. Una modalidad de la invención proporciona un método para mantener, tratar, curar y/o mejorar al menos una función cognitiva en un paciente que necesita de la misma, que comprende: administrar al paciente, durante un período prolongado, una dosis efectiva de (R)-7-cloro-N-(quinuclidin-3-il) benzo[b]tiofeno-2-carboxamida, o una sal farmacéuticamente aceptable de la misma.
MX2014013491A 2012-05-08 2013-05-06 Uso de (r)-7cloro-n-(quinuclidin-3-il) benzo[b] tiofeno-2-carboxamida o una sal farmacéuticamente aceptable de la misma para preparar una composición farmacéutica en el tratamiento de una disfunción cognitiva. MX358512B (es)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201261644113P 2012-05-08 2012-05-08
US201261670087P 2012-07-10 2012-07-10
PCT/US2013/039692 WO2013169646A1 (en) 2012-05-08 2013-05-06 Methods of maintaining, treating or improving cognitive function

Publications (2)

Publication Number Publication Date
MX2014013491A MX2014013491A (es) 2015-10-22
MX358512B true MX358512B (es) 2018-08-24

Family

ID=49551186

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2014013491A MX358512B (es) 2012-05-08 2013-05-06 Uso de (r)-7cloro-n-(quinuclidin-3-il) benzo[b] tiofeno-2-carboxamida o una sal farmacéuticamente aceptable de la misma para preparar una composición farmacéutica en el tratamiento de una disfunción cognitiva.

Country Status (9)

Country Link
US (2) US9585877B2 (es)
EP (3) EP3461481A1 (es)
AU (3) AU2013259871A1 (es)
CA (1) CA2872005A1 (es)
HK (1) HK1208356A1 (es)
IL (1) IL235469A0 (es)
MX (1) MX358512B (es)
RU (2) RU2635522C2 (es)
WO (1) WO2013169646A1 (es)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2017060290A1 (en) * 2015-10-06 2017-04-13 Sandoz Ag Crystalline encenicline hydrochloride
EP3153513A1 (en) * 2015-10-06 2017-04-12 Sandoz Ag Crystalline encenicline hydrochloride

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