LV10434A - 3-Amidopirazola atvasinajumi to iegusanas panemiens un farmaceitiskais sastavs uz to bazes - Google Patents

3-Amidopirazola atvasinajumi to iegusanas panemiens un farmaceitiskais sastavs uz to bazes

Info

Publication number
LV10434A
LV10434A LV930138A LV930138A LV10434A LV 10434 A LV10434 A LV 10434A LV 930138 A LV930138 A LV 930138A LV 930138 A LV930138 A LV 930138A LV 10434 A LV10434 A LV 10434A
Authority
LV
Latvia
Prior art keywords
amidopyrazole
depletion
derivatives
pharmaceutical composition
pharmaceutical
Prior art date
Application number
LV930138A
Other languages
English (en)
Other versions
LV10434B (en
Inventor
Robert Boigegrain
Danielle Gully
Francis Jeanjean
Jean-Charles Molimard
Original Assignee
Sanofi Elf
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sanofi Elf filed Critical Sanofi Elf
Publication of LV10434A publication Critical patent/LV10434A/lv
Publication of LV10434B publication Critical patent/LV10434B/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D231/28—Two oxygen or sulfur atoms
    • C07D231/30—Two oxygen or sulfur atoms attached in positions 3 and 5
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/08—Vasodilators for multiple indications
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D231/16—Halogen atoms or nitro radicals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/54—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings condensed with carbocyclic rings or ring systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups
LVP-93-138A 1990-08-20 1993-02-25 3-amidopyrazole derivatives, process for preparing these and pharmaceutical compositions containing them LV10434B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR9010486A FR2665898B1 (fr) 1990-08-20 1990-08-20 Derives d'amido-3 pyrazole, procede pour leur preparation et compositions pharmaceutiques les contenant.

Publications (2)

Publication Number Publication Date
LV10434A true LV10434A (lv) 1995-02-20
LV10434B LV10434B (en) 1995-10-20

Family

ID=9399742

Family Applications (1)

Application Number Title Priority Date Filing Date
LVP-93-138A LV10434B (en) 1990-08-20 1993-02-25 3-amidopyrazole derivatives, process for preparing these and pharmaceutical compositions containing them

Country Status (32)

Country Link
US (6) US5420141A (lv)
EP (1) EP0477049B1 (lv)
JP (1) JP2694932B2 (lv)
KR (1) KR100223074B1 (lv)
AR (1) AR248133A1 (lv)
AT (1) ATE187167T1 (lv)
AU (1) AU646683B2 (lv)
BR (1) BR9103550A (lv)
CA (4) CA2049514C (lv)
CZ (1) CZ281864B6 (lv)
DE (1) DE69131813T2 (lv)
DK (1) DK0477049T3 (lv)
ES (1) ES2142798T3 (lv)
FI (1) FI104170B1 (lv)
FR (1) FR2665898B1 (lv)
GR (1) GR3032732T3 (lv)
HK (1) HK1005136A1 (lv)
HU (2) HU217435B (lv)
IE (1) IE912932A1 (lv)
IL (1) IL99225A (lv)
LT (1) LT3520B (lv)
LV (1) LV10434B (lv)
MX (1) MX9203576A (lv)
MY (1) MY121908A (lv)
NO (1) NO300212B1 (lv)
NZ (1) NZ239476A (lv)
PL (1) PL169085B1 (lv)
PT (1) PT98717B (lv)
RU (1) RU2066317C1 (lv)
SG (1) SG52322A1 (lv)
TW (1) TW366337B (lv)
ZA (1) ZA916583B (lv)

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JPH04244065A (ja) 1992-09-01
PL291463A1 (en) 1992-07-13
EP0477049B1 (fr) 1999-12-01
HU211970A9 (en) 1996-01-29
CZ281864B6 (cs) 1997-03-12
BR9103550A (pt) 1992-04-07
LT3520B (en) 1995-11-27
CA2166902A1 (en) 1992-02-21
IL99225A0 (en) 1992-07-15
FI913917A0 (fi) 1991-08-19
IE912932A1 (en) 1992-02-26
US5635526A (en) 1997-06-03
IL99225A (en) 1995-10-31
CA2166901C (en) 1999-01-26
NO913234D0 (no) 1991-08-19
AR248133A1 (es) 1995-06-30
CA2049514A1 (en) 1992-02-21
CA2166903A1 (en) 1992-02-21
FI913917A (fi) 1992-02-21
US5744491A (en) 1998-04-28
US5744493A (en) 1998-04-28
DE69131813D1 (de) 2000-01-05
LV10434B (en) 1995-10-20
US5616592A (en) 1997-04-01
LTIP656A (en) 1995-01-31
MX9203576A (es) 1992-07-01
CA2166903C (en) 1998-09-01
SG52322A1 (en) 1998-09-28
FI104170B (fi) 1999-11-30
DK0477049T3 (da) 2000-04-25
CA2166902C (en) 1999-01-19
CA2049514C (en) 1997-02-25
CS257491A3 (en) 1992-06-17
US5607958A (en) 1997-03-04
US5420141A (en) 1995-05-30
DE69131813T2 (de) 2000-05-31
KR920004354A (ko) 1992-03-27
KR100223074B1 (ko) 1999-10-15
ES2142798T3 (es) 2000-05-01
FR2665898B1 (fr) 1994-03-11
TW366337B (en) 1999-08-11
RU2066317C1 (ru) 1996-09-10
HUT59106A (en) 1992-04-28
FI104170B1 (fi) 1999-11-30
GR3032732T3 (en) 2000-06-30
PT98717B (pt) 1999-01-29
EP0477049A1 (fr) 1992-03-25
ATE187167T1 (de) 1999-12-15
FR2665898A1 (fr) 1992-02-21
NZ239476A (en) 1993-11-25
ZA916583B (en) 1992-05-27
NO300212B1 (no) 1997-04-28
CA2166901A1 (en) 1992-02-21
HK1005136A1 (en) 1998-12-24
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AU8259691A (en) 1992-02-27
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